antiserotonergic

Cyproheptadine hydrochloride (Periactin hydrochloride) 是一种 5-HT2A 受体拮抗剂，具有抗抑郁和抗血清素作用。它具有抗血小板活性，可用于血栓栓塞性疾病的研究。

Telotristat Etiprate (LX 1606 Hippurate) 是一种色氨酸羟化酶抑制剂，可抑制血清素的产生。

Pirenperone 是5-HT2血清素受体拮抗剂，具有一定抗焦虑作用。

Telotristat 是色氨酸羟化酶 (tryptophan hydroxylase) 抑制剂，在体内的IC50值为0.028 μM。

Cyproheptadine 是一种有效的口服活性5-HT2A 受体拮抗剂。Cyproheptadine 具有抗抑郁和抗血清素作用。Cyproheptadine 还具有抗血小板和血栓保护活性，可用于研究血栓栓塞性疾病。

Citatepine is a tetracyclic dopamine antagonist acting strongly antidopaminergic opposed to antiserotonergic. Some anticholinergic activity.

Dothiepin HCl is a Tricyclic antidepressant (TCA), acting as a serotonin–norepinephrine reuptake inhibitor (SNRI) and also having other activities including antihistamine, antiadrenergic, antiserotonergic, anticholinergic, and sodium channel-blocking effects.

Levomepromazine Maleate is a Tricyclic antidepressant (TCA), acting as a serotonin–norepinephrine reuptake inhibitor (SNRI) and also having other activities including antihistamine, antiadrenergic, antiserotonergic, anticholinergic, and sodium channel-blocking effects.

6-Gingediol (compound 13) 作为一种从生姜中提取的化合物,展示了潜在的抗血清素效果和对胃粘膜的保护能力.在浓度不超过 10 μM 的情况下,该化合物不具备刺激性气味;然而,其浓度一旦超过 100 μM,乃至达到 1000 μM,刺激性气味则变得非常明显.