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Antiproliferative agent-15是一种具有抗癌活性的试剂。Antiproliferative agent-15对人结肠癌(HCT116和HCT15)和脑癌(LN-229和GBM-10)具有抗增殖活性。


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Antiproliferative agent-15是一种具有抗癌活性的试剂。Antiproliferative agent-15对人结肠癌(HCT116和HCT15)和脑癌(LN-229和GBM-10)具有抗增殖活性。
| 规格 | 价格 | 库存 | 数量 |
|---|---|---|---|
| 5 mg | ¥ 139 | In stock | |
| 10 mg | ¥ 203 | In stock | |
| 25 mg | ¥ 328 | In stock | |
| 50 mg | ¥ 585 | In stock | |
| 100 mg | ¥ 1,030 | In stock | |
| 200 mg | ¥ 1,560 | In stock |
| 产品描述 | Antiproliferative agent-15 is a reagent with anticancer activity. Antiproliferative agent-15 showed antiproliferative activity against human colon cancer (HCT116 and HCT15) and brain cancer (LN-229 and GBM-10). |
| 靶点活性 | HCT15 cells:4.8 μM, LN-229 cells:18.3 μM, HCT116 cells:8.3 μM, GBM10:12 μM |
| 体外活性 | Antiproliferative agent-15针对人类结肠癌细胞系(HCT116和HCT15)及脑癌细胞系(LN-229和GBM-10)显示出抗增殖活性,其IC50值分别为8.3 μM、4.8 μM、18.3 μM和12 μM [1]。 |
| 别名 | 抗增值剂15 |
| 分子量 | 282.36 |
| 分子式 | C16H14N2OS |
| CAS No. | 19819-18-2 |
| Smiles | O=C1C2=C(SC3=C2CCCC3)NC(=N1)C4=CC=CC=C4 |
| 密度 | no data available |
| 存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |
| 溶解度信息 | DMSO: Slightly soluble |
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