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细胞焦亡化合物库

细胞焦亡化合物库

现 货
产品编号 L8720 Pyroptosis Compound Library
  库化合物信息   Excel SDF

细胞焦亡,又称细胞炎性坏死,是一种程序性坏死;表现为细胞不断胀大直至细胞膜破裂,导致细胞内容物的释放进而激活强烈的炎症反应。按激活机制,可分为 Caspase-1依赖的经典途径和 Caspase-1不依赖(caspase-4/5/11)的非经典途径,caspase-1和 caspase-4/5/11通过切割 Gasdermin-D(GSDMD)蛋白,释放其 N 端结构域,该结构域结合膜脂并在细胞膜上打孔,导致细胞渗透压变化而发生胀大直至细胞膜破裂。两种途径都能同时诱导IL-1β和IL-18的前体进行切割,形成成熟的IL-1β和IL-18,并释放到胞外,造成炎症反应。细胞焦亡在感染性疾病、代谢疾病、神经系统疾病、心血管疾病、癌症等疾病中有广泛的研究,对细胞焦亡的研究有助于认识其在相关疾病的发生发展。

TargetMol 细胞焦亡化合物库收集了1077 种细胞焦亡相关的化合物,可以用于细胞焦亡相关研究。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
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产品描述

  • 1077种与细胞焦亡相关的活性小分子,可用于高通量和高内涵筛选;
  • 靶点包括Caspase-1、Caspase-4、Caspase-5、Caspase-11、NLRP3、gasdermin D等;
  • 部分化合物已被FDA批准上市;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L8720)
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客户使用化合物库发表的文献

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化合物库组成

NF-κB (219)
Apoptosis (206)
Autophagy (176)
Reactive Oxygen Species (165)
COX (136)
mTOR (86)
p38 MAPK (83)
TNF (78)
Endogenous Metabolite (77)
Caspase (75)
IL Receptor (71)
Antibacterial (59)
TLR (56)
PI3K (53)
ROS (53)
AMPK (48)
JNK (46)
IκB/IKK (38)
Akt (37)
p53 (37)
ERK (34)
Interleukin (24)
HIV Protease (24)
Ferroptosis (24)
NOD (22)
NO Synthase (21)
RIP kinase (21)
E1/E2/E3 Enzyme (21)
Antifungal (21)
PPAR (21)
Antioxidant (20)
STAT (20)
Parasite (19)
Mdm2 (19)
BCL (18)
Influenza Virus (17)
DNA-PK (16)
NOD-like Receptor (NLR) (16)
IRAK (16)
Antibiotic (16)
P450 (16)
NOS (15)
PARP (15)
Mitochondrial Metabolism (14)
Calcium Channel (13)
Mitophagy (13)
MMP (12)
Lipoxygenase (11)
DNA/RNA Synthesis (11)
ROS Kinase (10)
MAPK (10)
CDK (10)
SARS-CoV (10)
Nrf2 (10)
EGFR (9)
Dehydrogenase (8)
Beta Amyloid (8)
Potassium Channel (8)
PKC (8)
JAK (8)
Virus Protease (8)
Tyrosinase (7)
Topoisomerase (7)
Src (7)
VEGFR (7)
ASK (7)
S6 Kinase (7)
ATM/ATR (7)
HIF/HIF Prolyl-Hydroxylase (7)
GABA Receptor (6)
Sirtuin (6)
Proteasome (6)
AChE (6)
Prostaglandin Receptor (6)
P-gp (6)
PGE Synthase (6)
IAP (6)
Wnt/beta-catenin (6)
5-HT Receptor (6)
AChR (6)
Estrogen/progestogen Receptor (6)
ALK (6)
Xanthine Oxidase (5)
TGF-beta/Smad (5)
Sodium Channel (5)
NADPH (5)
Anti-infection (5)
HSV (5)
HSP (5)
PDE (5)
c-Met/HGFR (5)
Casein Kinase (5)
MEK (4)
Antiviral (4)
transporter (4)
Free radical scavengers (4)
Trk receptor (4)
HDAC (4)
ATPase (4)
HBV (4)
PDK (4)
Glucocorticoid Receptor (4)
PKA (4)
Pyroptosis (4)
Antifection (3)
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Indoleamine 2,3-Dioxygenase (IDO) (1)
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NPC1L1 (1)
c-Myc (1)
NMDAR (1)
c-RET (1)
Na+/Ca2+ Exchanger (1)
MyD88 (1)
OXPHOS (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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