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TargetMol | Compound Library

细胞焦亡化合物库现货

Pyroptosis Compound Library

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产品编号 L8720

细胞焦亡,又称细胞炎性坏死,是一种程序性坏死;表现为细胞不断胀大直至细胞膜破裂,导致细胞内容物的释放进而激活强烈的炎症反应。按激活机制,可分为 Caspase-1依赖的经典途径和 Caspase-1不依赖(caspase-4/5/11)的非经典途径,caspase-1和 caspase-4/5/11通过切割 Gasdermin-D(GSDMD)蛋白,释放其 N 端结构域,该结构域结合膜脂并在细胞膜上打孔,导致细胞渗透压变化而发生胀大直至细胞膜破裂。两种途径都能同时诱导IL-1β和IL-18的前体进行切割,形成成熟的IL-1β和IL-18,并释放到胞外,造成炎症反应。细胞焦亡在感染性疾病、代谢疾病、神经系统疾病、心血管疾病、癌症等疾病中有广泛的研究,对细胞焦亡的研究有助于认识其在相关疾病的发生发展。 TargetMol 细胞焦亡化合物库收集了1066 种细胞焦亡相关的化合物,可以用于细胞焦亡相关研究。

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产品编号 L8720

细胞焦亡化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 1066种与细胞焦亡相关的活性小分子,可用于高通量和高内涵筛选;
  • 靶点包括Caspase-1、Caspase-4、Caspase-5、Caspase-11、NLRP3、gasdermin D等;
  • 部分化合物已被FDA批准上市;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;

Packaging And Storage | TargetMol 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。

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Library Customization | TargetMol 化合物库组成

NF-κB
Apoptosis
Autophagy
Reactive Oxygen Species
COX
p38 MAPK
mTOR
Caspase
AMPK
TNF
IL Receptor
Endogenous Metabolite
Antibacterial
TLR
PI3K
ROS
JNK
IκB/IKK
p53
Akt
ERK
NOD
HIV Protease
RIP kinase
Interleukin
NO Synthase
Ferroptosis
Antioxidant
E1/E2/E3 Enzyme
Mdm2
Antifungal
PPAR
Parasite
STAT
Cytochromes P450
DNA-PK
Bcl-2 Family
IRAK
Antibiotic
NOS
Mitophagy
PARP
Influenza Virus
Calcium Channel
Mitochondrial Metabolism
NOD-like Receptor (NLR)
MMP
Lipoxygenase
CDK
DNA/RNA Synthesis
MAPK
SARS-CoV
Nrf2
ROS Kinase
Virus Protease
JAK
Potassium Channel
Dehydrogenase
Topoisomerase
EGFR
Sirtuin
Beta Amyloid
VEGFR
PKC
Cholinesterase (ChE)
ASK
ATM/ATR
GABA Receptor
S6 Kinase
Tyrosinase
HIF/HIF Prolyl-Hydroxylase
Proteasome
Estrogen/progestogen Receptor
Wnt/beta-catenin
IAP
HSV
TGF-beta/Smad
PGE Synthase
Prostaglandin Receptor
ALK
HDAC
5-HT Receptor
AChR
c-Met/HGFR
HBV
PDE
Xanthine Oxidase
P-gp
HSP
Pyroptosis
Casein Kinase
MEK
Anti-infection
Sodium Channel
Src
Adenosine Receptor
NADPH
PKA
TRP/TRPV Channel
Glucocorticoid Receptor
Aurora Kinase
Trk receptor
Free radical scavengers
transporter
Ligand for E3 Ligase
PDK
FLT
ATPase
Chloride channel
Carbonic Anhydrase
HCV Protease
RAAS
Histamine Receptor
Glutathione Peroxidase
GSK-3
Serine Protease
Leukotriene Receptor
Aryl Hydrocarbon Receptor
MAO
Immunology/Inflammation related
Raf
Molecular Glues
Opioid Receptor
IGF-1R
Antiviral
Reverse Transcriptase
FGFR
Microtubule Associated
Transferase
Integrin
DNA Alkylator/Crosslinker
Reductase
BACE
IFNAR
PERK
Tie-2
Phosphatase
MRP
Estrogen Receptor/ERR
Tyrosine Kinases
RANKL/RANK
Bcr-Abl
Antifection
Epigenetic Reader Domain
CaMK
DNA
DUB
AIM2
Retinoid Receptor
c-Fms
Aromatase
Phospholipase
HIF
Cannabinoid Receptor
Complement System
Syk
c-Kit
FAK
MLK
ADC Cytotoxin
FOXO3
PROTACs
NPC1L1
RAR/RXR
ROR
Dynamin
MyD88
LTR
Na+/Ca2+ Exchanger
Lipase
gp120/CD4
Progesterone Receptor
OCT
c-Myc
Rho
Serine/threonin kinase
Liver X Receptor
Nucleoside Antimetabolite/Analog
Cysteine Protease
FXR
Glucokinase
ROCK
Adrenergic Receptor
Amylase
iGluR
SIK
Annexin A
FLAP
UGT
PAFR
Haspin Kinase
LDL
Gamma-secretase
Drug Metabolite
Glucagon Receptor
NMDAR
Glucosidase
PAK
PDGFR
Hedgehog/Smoothened
FAAH
CCR
CXCR
PTEN
Somatostatin
Chk
PAD
cAMP
Indoleamine 2,3-Dioxygenase (IDO)
Androgen Receptor
SGLT
ATP Citrate Lyase
OXPHOS
Beta-Secretase
Glutathione reductase
STING
LRRK2
Aminopeptidase
cGAS
PAI-1
RSV
GST
PI4K
Adenosine Deaminase
c-RET
Discoidin Domain Receptor (DDR)
Gap Junction Protein
Platelet aggregation
NADPH-oxidase
AhR
CFTR
PKM
S1P Receptor
HER
Monoamine Oxidase
BTK

Keywords