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中药单体化合物库

中药单体化合物库

产品编号 L6810 Traditional Chinese Medicine Monomer Library
  库化合物信息   Excel SDF

中药的有效性已经在数千年的实践中得到了验证,为挽救人类的生命做出了重大贡献,但由于其成分过于复杂,难以通过实验证明其作用机理,使中药在现代医学中的应用受到了极大限制。实际上中药具有一定的药理作用主要是因为其中含有的活性化合物,如黄花蒿具有抗疟药效是因为其中含有抗疟活性成分青蒿素,人参被称之为 “百草之王”,具有多种药理活性,也是因为其中含有多种人参皂苷成分。随着国家对中药现代化的重视日益加深,中药单体的研究已经成为研究中药抗病机理的主要途径。

与人工合成的化合物相比,中药单体往往具有更高的生物学活性和结构多样性,更易进入细胞发挥药效,拥有更高的生物学活性。此外,针对一些特殊的困难靶点,从中药单体中筛选得到其调节剂的概率更大。

TargetMol 精选2688 种中药来源的单体化合物,来源包括三七、甘草、当归、陈皮、黄连、人参等近800种传统中药,含有黄酮、生物碱、萜类、糖苷等多种结构类型,是抗癌、抗炎、抗菌、细胞凋亡、细胞自噬研究领域的有力工具。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
我们的产品含有多种规格,如需了解具体的规格以及价格信息,请联系我们咨询订购,对于大额的订购,我们还有额外的优惠!
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如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
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产品描述

  • 2688种中药来源的单体化合物,是药物开发、药理研究等领域的有力工具;
  • 来源包括三七、甘草、当归、陈皮、黄连、人参等近800种传统中药;
  • 结构多样,包含黄酮、生物碱、萜类、糖苷等多种类别,分类详细;
  • HNMR/HPLC检测保障化合物品质;
  • 所有化合物现货供应,到货快。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L6810)
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化合物库组成

Endogenous Metabolite (462)
Apoptosis (320)
Antibacterial (205)
Autophagy (196)
NF-κB (170)
Antioxidant (102)
Antifungal (91)
COX (85)
Reactive Oxygen Species (82)
P450 (65)
Parasite (61)
TNF (61)
Influenza Virus (58)
AChR (50)
p38 MAPK (46)
AChE (45)
ERK (43)
Anti-infection (43)
IL Receptor (42)
NO Synthase (42)
HIV Protease (41)
Akt (38)
STAT (37)
Calcium Channel (36)
Antibiotic (35)
GABA Receptor (35)
Caspase (34)
DNA/RNA Synthesis (34)
Tyrosinase (34)
AMPK (33)
PPAR (33)
JNK (28)
MMP (28)
ROS (28)
Virus Protease (28)
Ferroptosis (26)
Topoisomerase (26)
PI3K (25)
5-HT Receptor (25)
BCL (25)
Nrf2 (24)
Lipoxygenase (23)
Estrogen Receptor/ERR (23)
TRP/TRPV Channel (22)
Immunology/Inflammation related (22)
Estrogen/progestogen Receptor (21)
NOS (21)
Antifection (20)
HSV (20)
PKC (20)
Prostaglandin Receptor (20)
ATPase (19)
Potassium Channel (19)
Dehydrogenase (19)
Mitophagy (18)
Glucosidase (18)
Beta Amyloid (17)
Microtubule Associated (17)
Adrenergic Receptor (16)
P-gp (16)
HBV (16)
Antiviral (16)
PDE (15)
EGFR (14)
Dopamine Receptor (14)
MAO (14)
PARP (14)
Wnt/beta-catenin (14)
Sodium Channel (13)
JAK (13)
Interleukin (13)
mTOR (12)
HIF/HIF Prolyl-Hydroxylase (11)
TLR (11)
TGF-beta/Smad (10)
MAPK (10)
Phosphatase (10)
Sirtuin (10)
Mitochondrial Metabolism (10)
Reductase (10)
SARS-CoV (9)
Phospholipase (9)
HCV Protease (9)
Fatty Acid Synthase (9)
Androgen Receptor (8)
iGluR (8)
VEGFR (8)
Opioid Receptor (8)
Monoamine Oxidase (8)
CDK (8)
Drug Metabolite (8)
RAAS (8)
HDAC (7)
HSP (7)
Adenosine Receptor (7)
UGT (7)
Cannabinoid Receptor (7)
BACE (7)
IκB/IKK (7)
MEK (7)
transporter (6)
p53 (6)
Platelet aggregation (6)
Histamine Receptor (6)
HER (6)
PAFR (6)
LDL (6)
Indoleamine 2,3-Dioxygenase (IDO) (6)
GluR (6)
Chloride channel (6)
Carbonic Anhydrase (6)
Gamma-secretase (5)
NMDAR (5)
Epigenetic Reader Domain (5)
Proteasome (5)
Beta-Secretase (5)
CaMK (5)
Amino Acids and Derivatives (5)
cAMP (5)
HIF (5)
NOD (4)
PKA (4)
Free radical scavengers (4)
Nucleoside Antimetabolite/Analog (4)
PGE Synthase (4)
PTEN (4)
CXCR (4)
Reverse Transcriptase (4)
Hedgehog/Smoothened (4)
FAK (4)
Serine Protease (4)
SGLT (4)
FGFR (4)
Xanthine Oxidase (4)
S6 Kinase (4)
IGF-1R (4)
HMG-CoA Reductase (4)
Integrin (4)
IAP (4)
GSK-3 (4)
Aromatase (4)
GPR (4)
E1/E2/E3 Enzyme (3)
DNA (3)
Tyrosine Kinases (3)
Acyltransferase (3)
Progesterone Receptor (3)
Histone Acetyltransferase (3)
MRP (3)
CCR (3)
cell cycle arrest (3)
Proton pump (3)
NOD-like Receptor (NLR) (3)
PDGFR (3)
Telomerase (3)
FAAH (3)
ROR (3)
Syk (3)
Glucocorticoid Receptor (3)
Liver X Receptor (3)
Arginase (3)
c-Met/HGFR (3)
Serotonin Transporter (3)
Src (3)
GST (3)
Casein Kinase (2)
Pim (2)
PKM (2)
Smo (2)
Adiponectin receptor (2)
Trk receptor (2)
Transferase (2)
Bombesin Receptor (2)
Aminopeptidase (2)
Thrombin (2)
Pyroptosis (2)
Bcr-Abl (2)
RANKL/RANK (2)
Ras (2)
Aurora Kinase (2)
ATM/ATR (2)
Serine/threonin kinase (2)
Aryl Hydrocarbon Receptor (2)
PAI-1 (2)
hCE (2)
c-Myc (2)
DYRK (2)
NADPH-oxidase (2)
DPP-4 (2)
Monoamine Transporter (2)
OAT (2)
ABC (2)
Glutathione Peroxidase (2)
Glucokinase (2)
NADPH (2)
Cysteine Protease (2)
IRAK (2)
Leukotriene Receptor (2)
Lipase (2)
Lipid (2)
FXR (1)
FLT (1)
Stearoyl-CoA Desaturase (SCD) (1)
stilbene oxidase (1)
Survivin (1)
Imidazoline Receptor (1)
Fas/FasL (1)
Glucagon Receptor (1)
Antifolate (1)
Factor Xa (1)
advanced glycation end products (1)
aconitase (1)
Histone Demethylase (1)
Adenosine deaminase (1)
Adenylyl cyclase (1)
Histone Methyltransferase (1)
GlyT (1)
Glutathione reductase (1)
IFNAR (1)
AhR (1)
Transaminase (1)
ALK (1)
Hydroxylase (1)
IDO (1)
Thrombopoietin Receptor (1)
LTR (1)
CRISPR/Cas9 (1)
RSV (1)
DNA gyrase (1)
P2Y Receptor (1)
PD-1/PD-L1 (1)
CFTR (1)
P2X Receptor (1)
PDK (1)
PERK (1)
Oxytocin Receptor (1)
Decarboxylase (1)
CaSR (1)
Phosphorylase (1)
OCT (1)
DHFR (1)
NPC1L1 (1)
Norepinephrine (1)
PLK (1)
ROS Kinase (1)
Epoxide Hydrolase (1)
ATP Citrate Lyase (1)
CYP19A1 (1)
ribosome (1)
Melatonin Receptor (1)
Retinoid Receptor (1)
ATTECs (1)
Dynamin (1)
DNA Methyltransferase (1)
Raf (1)
Monocarboxylate transporter (1)
MT Receptor (1)
MTH1 (1)
MyD88 (1)
Prolyl Endopeptidase (PREP) (1)
Mdm2 (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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