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    TargetMol | Inhibitors_Agonists
  • telaglenastat
    CB-839, CB839, CB 839
    T67971439399-58-2
    Telaglenastat (CB 839) 是一种谷氨酰胺酶 1 (GLS1) 抑制剂，具有选择性、可逆性和口服活性。Telaglenastat 具有抗肿瘤活性，可以诱导细胞自噬。
    transporterGlutaminaseAutophagy
    • ¥ 221
    In stock
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  • Telaglenastat hydrochloride
    CB-839 hydrochloride
    T393091874231-60-3
    Telaglenastat (CB-839) hydrochloride is a first-in-class, reversible, and orally active inhibitor of glutaminase 1 (GLS1). It selectively inhibits the splice variants of GLS1, specifically KGA (kidney-type glutaminase) and GAC (glutaminase C), as compared to GLS2. Telaglenastat hydrochloride has an IC50 of 23 nM for endogenous glutaminase in mouse kidney and 28 nM in the brain. In addition, it induces autophagy and exhibits antitumor activity.
    Others
    • ¥ 10600
    1-2周
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