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糖酵解化合物库

糖酵解化合物库

产品编号 L2521 Glycolysis Compound Library
  库化合物信息   Excel SDF

糖酵解途径又称 EMP 途径(Embden-Meyerhof-Parnas pathway),指在无氧条件下葡萄糖通过一系列步骤,降解成丙酮酸并生成 ATP 的过程,糖酵解发生在所有活细胞中。研究发现即使在有氧状态下,肿瘤细胞仍会优先选择糖酵解途径提供能量,称为有氧糖酵解(Warburg 效应)。与正常细胞比较,肿瘤细胞会消耗更多的葡萄糖,所以通过定位消耗大量葡萄糖的区域可以帮助识别癌症。因此靶向肿瘤细胞的糖酵解有望成为治疗肿瘤的一个重要治疗策略。

TargetMol 收集了 555 种靶向糖酵解相关的活性化合物,可用于抗肿瘤和糖代谢相关药物开发。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
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产品描述

  • 555种糖酵解相关的活性化合物,可用于高通量和高内涵筛选;
  • 作用靶点包含己糖激酶(hexokinase);丙酮酸激(pyruvate kinase);葡萄糖激酶(glucokinase)等糖酵解关键酶;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;
  • NMR和HPLC检测技术保证产品高纯度和高质量;
  • 所有化合物现货供应。

化合物库定制

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包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L2521)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

PI3K (157)
Autophagy (103)
Apoptosis (103)
Akt (85)
mTOR (84)
AMPK (60)
GSK-3 (52)
HIF/HIF Prolyl-Hydroxylase (40)
DNA-PK (37)
HIF (29)
S6 Kinase (29)
CDK (26)
ATM/ATR (22)
Endogenous Metabolite (21)
Glucokinase (20)
PDK (19)
Antibacterial (18)
NF-κB (16)
c-Myc (16)
ERK (15)
Reactive Oxygen Species (15)
transporter (15)
PI4K (13)
PKC (11)
PKA (10)
Parasite (10)
p38 MAPK (10)
VEGFR (9)
Mitophagy (8)
Src (8)
PKM (8)
TNF (7)
Dehydrogenase (7)
HIV Protease (7)
PTEN (7)
Chk (7)
JNK (7)
Casein Kinase (6)
Influenza Virus (6)
Caspase (6)
ROCK (6)
STAT (6)
MAPK (6)
PPAR (6)
Antibiotic (6)
SIK (5)
Phosphatase (5)
MELK (5)
MEK (5)
COX (5)
FLT (5)
IL Receptor (5)
HSV (4)
MMP (4)
Potassium Channel (4)
P450 (4)
Calcium Channel (3)
Raf (3)
Microtubule Associated (3)
HCV Protease (3)
PDGFR (3)
JAK (3)
IGF-1R (3)
SGK (3)
Hexokinase (3)
Mitochondrial Metabolism (3)
Interleukin (3)
Lipoxygenase (3)
PDE (3)
Virus Protease (3)
PLK (2)
DNA/RNA Synthesis (2)
Antiviral (2)
Tyrosinase (2)
Epigenetic Reader Domain (2)
HDAC (2)
ATP Citrate Lyase (2)
TGF-beta/Smad (2)
Cannabinoid Receptor (2)
SGLT (2)
FGFR (2)
EGFR (2)
c-RET (2)
Prostaglandin Receptor (2)
Beta Amyloid (2)
Chloride channel (2)
Wnt/beta-catenin (2)
Glucosidase (2)
Tyrosine Kinases (2)
Integrin (2)
Adenosine Receptor (2)
Carbonic Anhydrase (2)
Ferroptosis (2)
Bcr-Abl (2)
PARP (2)
BCL (2)
Aurora Kinase (2)
Fatty Acid Synthase (2)
Adrenergic Receptor (2)
MRP (1)
GABA Receptor (1)
RAAS (1)
PERK (1)
DYRK (1)
IFNAR (1)
BACE (1)
Antioxidant (1)
HBV (1)
c-Met/HGFR (1)
Antifungal (1)
Estrogen/progestogen Receptor (1)
YAP (1)
AChR (1)
DAPK (1)
c-Kit (1)
cholecystokinin (1)
NPC1L1 (1)
NOS (1)
Proton pump (1)
FAK (1)
CFTR (1)
p53 (1)
PD-1/PD-L1 (1)
Kinesin (1)
ATPase (1)
NO Synthase (1)
Estrogen Receptor/ERR (1)
GluR (1)
CRISPR/Cas9 (1)
P-gp (1)
CXCR (1)
CaMK (1)
Guanylate cyclase (1)
Androgen Receptor (1)
Phosphorylase (1)
Drug Metabolite (1)
Gamma-secretase (1)
E1/E2/E3 Enzyme (1)
BCRP (1)
Myosin (1)
Topoisomerase (1)
Beta-Secretase (1)
MAO (1)
AChE (1)
OAT (1)
KLF (1)
Serine Protease (1)
c-Fms (1)
Pim (1)
Reverse Transcriptase (1)
Rho (1)
Hck (1)
IκB/IKK (1)
cell cycle arrest (1)
Aryl Hydrocarbon Receptor (1)
Serine/threonin kinase (1)
Nrf2 (1)
FXR (1)
Sirtuin (1)
Trk receptor (1)
Glutaminase (1)
S1P Receptor (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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