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抗肝癌化合物库

抗肝癌化合物库

产品编号 L2193 Anti-Liver Cancer Compound Library
  库化合物信息   Excel SDF

在全球范围内,肝癌占癌症死亡率第三位。肝癌的主要病因包括乙肝、丙肝、酒精性脂肪性肝炎和非酒精性脂肪性肝炎(NASH)。许多细胞信号通路与肝癌的发生有关,如 PI3K/Akt/mTOR 信号通路,表皮生长因子受体(EGFR)、血管内皮生长因子受体(VEGFR)等

TargetMol 抗肝癌化合物库收集了 1816 种与肝癌相关的化合物,包括已经报道具有肝癌治疗作用的化合物,以及靶向肝癌相关靶点潜在治疗肝癌的化合物,是抗肝癌药物研发的良好工具。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
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产品描述

  • 1816种与肝癌相关的化合物,可以用于抗肝癌药物研发和药理研究;
  • 通路靶点包含PI3K/Akt/mTOR,EGFR, FGFR,Met等;
  • 部分化合物已上市或进入临床期;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L2193)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

Apoptosis (355)
Autophagy (281)
NF-κB (206)
Reactive Oxygen Species (163)
PI3K (156)
EGFR (144)
VEGFR (141)
Endogenous Metabolite (90)
JAK (88)
mTOR (85)
Akt (85)
ERK (82)
p38 MAPK (81)
STAT (79)
FGFR (73)
Antibacterial (71)
PDGFR (67)
Raf (66)
c-Met/HGFR (64)
AMPK (60)
CDK (59)
Ras (59)
TGF-beta/Smad (52)
GSK-3 (52)
FLT (51)
c-Kit (49)
JNK (45)
Src (44)
COX (44)
MEK (42)
MAPK (41)
IκB/IKK (38)
HER (37)
DNA/RNA Synthesis (37)
DNA-PK (36)
TNF (34)
S6 Kinase (30)
Parasite (30)
Ferroptosis (30)
Tyrosine Kinases (28)
Antibiotic (28)
HIV Protease (27)
IL Receptor (25)
Mitophagy (24)
c-RET (23)
ALK (23)
RIP kinase (22)
ATM/ATR (22)
Antifungal (21)
Potassium Channel (21)
Bcr-Abl (21)
Caspase (21)
NOD (20)
PKC (20)
Influenza Virus (19)
PDK (19)
Aurora Kinase (17)
ROS (17)
P450 (17)
Antioxidant (17)
IRAK (16)
Calcium Channel (15)
Pim (15)
Topoisomerase (15)
IGF-1R (14)
Casein Kinase (14)
TAM Receptor (14)
PI4K (13)
PKA (13)
Trk receptor (13)
NO Synthase (13)
NOD-like Receptor (NLR) (13)
PPAR (13)
Rho (12)
Microtubule Associated (12)
c-Fms (12)
MMP (12)
Mitochondrial Metabolism (12)
Dehydrogenase (12)
Interleukin (12)
PD-1/PD-L1 (11)
Lipoxygenase (11)
Nucleoside Antimetabolite/Analog (11)
Sodium Channel (10)
HDAC (10)
HCV Protease (10)
Virus Protease (10)
5-HT Receptor (10)
FAK (9)
HIF/HIF Prolyl-Hydroxylase (9)
Chk (9)
Nrf2 (9)
AChR (9)
HBV (9)
ROCK (9)
Tyrosinase (8)
Adrenergic Receptor (8)
BCL (8)
HSP (8)
Estrogen/progestogen Receptor (8)
Syk (8)
Proteasome (8)
PTEN (8)
Wnt/beta-catenin (8)
PDE (7)
HSV (7)
TLR (7)
p53 (7)
Reverse Transcriptase (7)
SARS-CoV (7)
Beta Amyloid (7)
NOS (7)
BTK (6)
PLK (6)
GABA Receptor (6)
DNA Alkylator/Crosslinker (6)
E1/E2/E3 Enzyme (6)
Drug Metabolite (5)
MELK (5)
CSF-1R (5)
TOPK (5)
Adenosine Receptor (5)
MLK (5)
HIF (5)
Histone Methyltransferase (5)
PARP (5)
AChE (5)
ASK (5)
Antiviral (5)
MNK (5)
SGK (5)
Estrogen Receptor/ERR (5)
SIK (5)
Ephrin Receptor (5)
Phosphatase (5)
Transferase (5)
Histamine Receptor (5)
CaMK (4)
NADPH (4)
Serine Protease (4)
DNA Alkylation (4)
P-gp (4)
Aryl Hydrocarbon Receptor (4)
Tie-2 (4)
Prostaglandin Receptor (4)
RAAS (4)
ATPase (4)
Integrin (4)
Histone Acetyltransferase (3)
CCR (3)
Glucosidase (3)
Glutathione Peroxidase (3)
ROS Kinase (3)
Proton pump (3)
Carbonic Anhydrase (3)
KLF (3)
Epigenetic Reader Domain (3)
BACE (3)
IFNAR (3)
Chloride channel (3)
Sirtuin (3)
Cannabinoid Receptor (3)
Glucocorticoid Receptor (3)
Discoidin Domain Receptor (DDR) (3)
Antifection (3)
Free radical scavengers (3)
Anti-infection (3)
PGE Synthase (3)
LRRK2 (3)
Opioid Receptor (3)
cholecystokinin (3)
Phospholipase (2)
Retinoid Receptor (2)
RSV (2)
ROR (2)
Aromatase (2)
PERK (2)
Beta-Secretase (2)
Fatty Acid Synthase (2)
Somatostatin (2)
S1P Receptor (2)
Kinesin (2)
Glutathione reductase (2)
TRP/TRPV Channel (2)
GST (2)
GTPase (2)
transporter (2)
Hck (2)
Hedgehog/Smoothened (2)
HMG-CoA Reductase (2)
DPP-4 (2)
IRE1 (2)
c-Myc (2)
RANKL/RANK (2)
Leukotriene Receptor (2)
MAO (2)
DHFR (2)
Antifolate (2)
NADPH-oxidase (2)
Aminopeptidase (1)
Serotonin Transporter (1)
Wee1 (1)
UGT (1)
ACK (1)
Reductase (1)
Serine/threonin kinase (1)
Sigma receptor (1)
SGLT (1)
Adenosine deaminase (1)
Telomerase (1)
ATP Citrate Lyase (1)
Thrombopoietin Receptor (1)
Androgen Receptor (1)
STING (1)
AhR (1)
Thrombin (1)
cGAS (1)
RAR/RXR  (1)
Hydroxylase (1)
Liver X Receptor (1)
LDL (1)
KSP (1)
DNA Methyltransferase (1)
Dopamine Receptor (1)
ABC (1)
Indoleamine 2,3-Dioxygenase (IDO) (1)
DUB (1)
DYRK (1)
IAP (1)
Hippo pathway (1)
DNA (1)
hCE (1)
Haspin Kinase (1)
GPX (1)
GPR (1)
GluR (1)
Glucokinase (1)
Gap Junction Protein (1)
Gamma-secretase (1)
FXR (1)
FAAH (1)
LTR (1)
Mdm2 (1)
Pyroptosis (1)
OXPHOS (1)
PYK2 (1)
Progesterone Receptor (1)
Platelet aggregation (1)
PKM (1)
BCRP (1)
BMI-1 (1)
cAMP (1)
PAK (1)
PAI-1 (1)
CFTR (1)
OCT (1)
Melanin-concentrating Hormone Receptor (MCHR) (1)
NPC1L1 (1)
Complement System (1)
NEDD8 (1)
Na+/Ca2+ Exchanger (1)
Myosin (1)
CRISPR/Cas9 (1)
MRP (1)
Monoamine Oxidase (1)
Cysteine Protease (1)
DAPK (1)
YAP (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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