cck 1

CCK-A receptor inhibitor 1 是一种有效的缩胆囊素 A (CCK-A) 受体抑制剂(IC50：340 nM）。CCK-A receptor inhibitor 1 可用于研究与消化系统相关的疾病。

Gastrin CCK antagonist 1 是一种有效的 gastrin CCK 拮抗剂，可用于研究代谢系统相关疾病。

Lintitript (SR 27897) 是 CCK1的选择性拮抗剂，对 CCK1和 CCK2的 EC50s 为6 nM 和200 nM。对 CCK1的 Ki 值为0.2 nM。

CCK-B Receptor Antagonist 1 is a cholecystokinin B (CCK-B) receptor agonist and has the potential of reducing the secretion of gastric acid.

CCK2R Ligand-Linker Conjugate 1 is a hydrophilic peptide linker that conjugates to the cytotoxic antimicrotubule agents Desacetyl Vinblastine Hydrazide (DAVBH) and Tubulysin B Hydrazide (TubBH) as ligand-linker conjugates[1].

Cholecystokinin (1-21)，作为一种胆囊收缩素 (CCK) 片段，能够激活人体脂肪组织的脂肪分解作用。

GV-150013X ((S)-1-(1-(adamantan-1-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepin-3-yl)-3-phenylurea) 是一种有效的CCKB 拮抗剂，pKi= 9.02。

Sograzepide (Netazepide) 是一种具有口服活性选择性和高效性的 Gastrin/CCK-B 拮抗剂，抑制 Gastrin/CCK-A 活性，抑制 1 型胃神经内分泌肿瘤中 Pappalysin 2 的表达，可诱导 1 型胃神经内分泌肿瘤消退。

Loxiglumide (CR-1505) 是一种缩胆囊素受体拮抗剂。

Pinolenic acid is a polyunsaturated fatty acid found in Korean pine (Pinus orientalis) and maritime pine (Pinus pinaster) seed oils. Both oils have been found to have lipid-lowering properties. A diet containing maritime pine seed oil (MPSO) lowered high-density lipoprotein and ApoA1 levels in transgenic mice expressing human ApoA1. MPSO was found to diminish cholesterol efflux in vitro. Korean pine seed oil supplements may help in obesity by reduction of appetite. People taking this oil had an increase in the satiety hormones CCK and GLP-1 and a reduced desire to eat. The activity of the oil is attributed to pinolenic acid. Pinolenic acid is not converted to arachidonic acid metabolically and can reduce arachidonic acid levels in the phosphatidylinositol fraction of HepG2 cells from 15.9% to 7.0%. Pinolenic acid ethyl ester is a neutral, more lipophilic form of the free acid.

Givinostat(ITF-2357)是一种非选择性和口服活性的HDAC抑制剂，能够抑制STAT5磷酸化，对crlf2重排的BCP-ALL具有抗肿瘤活性并诱导凋亡。Givinostat具有抗炎活性，在endotoxin刺激的PBMCs中抑制TNF-α和IL-1β，还能够促进β细胞的存活，可用于糖尿病、急性淋巴细胞白血病和关节炎。

CCK (27-33) is a C-terminal fragment of CCK , a peptide hormone found in the intestine and brain that stimulates digestion, mediates satiety, and is involved in anxiety. Non-sulfated CCK (27-33) inhibits binding of [3H]naloxone in rat cerebellum membranes (IC50 = 4 uM) and inhibits electrically-stimulated contraction of isolated guinea pig ileum (IC50 = 17 uM), an effect that can be reversed by naloxone. Unlike sulfated CCK (27-33), the non-sulfated form does not reduce exploratory behavior in mice when administered at doses up to 1 uMol/kg.

Butabindide (UCL-1397) 是三肽肽酶II (TPP II)的选择性抑制剂，对 TPP I 和TPP II 的Ki 值分别为 10 μM 和 7 nM。Butabindide 抑制 TPP II 以保护 CCK-8 免于失活。

CE-326597 is a potent and selective CCK1R agonist. The type 1 cholecystokinin receptor (CCK1R) has multiple physiologic roles relating to nutrient homeostasis,including mediation of postcibal satiety. The type 1 cholecystokinin (CCK) receptor (CCK1R) is a key mediator of postcibal satiety and a potential target for drugs that may be useful to prevent and or treat obesity.

L-Phenylalanine (Standard)（L-苯丙氨酸标准品）是一种人体必需的α-氨基酸，作为标准品可用于定量分析。L-苯丙氨酸是 GPR142 的激动剂，促进胰岛素分泌，与糖代谢和糖尿病研究密切相关。可作为钙敏感受体（CaSR）的激活剂促进胆囊收缩素（CCK）和胰高血糖素样肽-1（GLP-1）的分泌，从而影响食欲和代谢。可通过影响多巴胺水平间接调节N-甲基-D-天冬氨酸受体（NMDA受体）。

[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate ([D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate (96736-12-8 free base)) 是广谱神经肽反向激动剂和拮抗剂。 ghrelin 受体的强效完全反向激动剂(EC50 = 5.2 nM)；减少组成型生长素释放肽受体信号传导。它也是速激肽、缓激肽、CCK 和铃蟾肽受体的拮抗剂。在体外诱导细胞凋亡并抑制癌细胞生长。

Cholecystokinin-33 (swine) 是胆囊收缩素 (CCK) 片段，可以减少食物摄入量和胆囊收缩。