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Cat. No. | Product Name | ||
---|---|---|---|
L7110 | 抗高血压化合物库 | 719 compounds | |
719 种高血压相关的小分子,用于高通量和高内涵筛选; |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T0706 |
Lisinopril dihydrate
Lisinopril,Renacor,赖诺普利二水合物,MK-521 (dihydrate) |
RAAS; MRP | Endocrinology/Hormones; Immunology/Inflammation |
Lisinopril dihydrate (MK-521) 是一种血管紧张素转化酶抑制剂。Lisinopri dihydrate 能够作用于高血压,充血性心力衰竭和心脏病等。 | |||
T32790 |
Lisinopril R,S,S-diketopiperazine
Lisinopril specified impurity D |
||
Lisinopril R,S,S-diketopiperazine is a bioactive chemical. | |||
T71028 | Lisinopril, epsilon-biotinamidocaproyl- | ||
Lisinopril, epsilon-biotinamidocaproyl- is an angiotensin converting enzyme (ACE) inhibitor. | |||
T71026 | MC2050 HCl | ||
MC2050 is a potent PARP-1 inhibitor. The IC50 for inhibition of PARP-1 activity is 119 nM, compared to 1.8 μM for PARP-2. MC2050 inhibits apoptosis and blocks poly ADP-ribosylation of histone H1 in hydrogen peroxide treated SH-SY5Y neuroblastoma cells. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T21418 |
Lisinopril
Linopril,赖诺普利,Zestril,Prinivil,Lisipril |
RAAS | Endocrinology/Hormones |
Lisinopril (Prinivil) 是一种血管紧张素转化酶抑制剂,能够作用于高血压,充血性心力衰竭和心脏病等。 |
Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPJ-00386 |
ACE2/ACEH Protein, Human, Recombinant (HEK293, His & Avi), Biotinylated
Metalloprotease MPROT15,ACEH,Angiotensin-Converting Enzyme H... |
Human | Human Cells |
Angiotensin-Converting Enzyme 2 (ACE-2) is an integral membrane protein and a zinc metalloprotease of the ACE family, the ACE family includes somatic and germinal ACE. ACE-2 cleaves angiotensins I and II as a carboxypeptidase, ACE-2 converts angiotensin I to angiotensin 1-9, and angiotensin II to angiotensin 1-7. ACE-2 is also able to hydrolyze apelin-13 and dynorphin-13 with high efficiency. ACE-2 can be high expressed in testis, kidney and heart, in colon, small intestine and ovary at moderate... |