首页 工具
登录
购物车
临床前化合物库

临床前化合物库

现 货
产品编号 L3410 Preclinical Compound Library
  库化合物信息   Excel SDF

709 个临床前小分子化合物的独特集合,靶点明确,有详细的临床分期和适应症信息,可用于高通量、高内涵筛选。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
咨询化合物库
获取报价
点击图片重新获取验证码

产品描述

  • 709种临床前小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 拥有明确的靶点信息;有详细的临床分期和适应症信息;
  • 是新药研发过程中的热门先导化合物;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR和HPLC检测技术保证产品高纯度和高质量;
  • 所有化合物现货供应。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L3410)
点击图片重新获取验证码

客户使用化合物库发表的文献

收起

化合物库组成

Apoptosis (130)
Autophagy (112)
Endogenous Metabolite (37)
Antibacterial (35)
Antibiotic (33)
CDK (25)
VEGFR (25)
PDGFR (20)
PI3K (20)
HIV Protease (20)
FGFR (19)
DNA/RNA Synthesis (18)
EGFR (18)
NF-κB (17)
Influenza Virus (17)
JAK (16)
Adrenergic Receptor (13)
FLT (13)
Dopamine Receptor (12)
c-Kit (12)
Src (12)
5-HT Receptor (12)
Epigenetic Reader Domain (12)
Calcium Channel (12)
Histamine Receptor (12)
Microtubule Associated (12)
mTOR (12)
Parasite (11)
Sodium Channel (11)
HDAC (11)
PDE (10)
c-RET (10)
c-Met/HGFR (10)
Ferroptosis (10)
AChR (10)
Adenosine Receptor (9)
Potassium Channel (9)
PPAR (9)
Bcr-Abl (9)
HSP (9)
Mitophagy (9)
Phosphatase (9)
BCL (9)
Aurora Kinase (9)
E1/E2/E3 Enzyme (9)
Reactive Oxygen Species (9)
Raf (9)
ATM/ATR (9)
DNA-PK (8)
ALK (8)
SARS-CoV (8)
iGluR (8)
PLK (8)
PKC (8)
COX (8)
MEK (8)
p53 (8)
GluR (8)
IGF-1R (7)
Dehydrogenase (7)
DNA Alkylator/Crosslinker (7)
Antifungal (7)
p38 MAPK (7)
STAT (7)
GSK-3 (7)
ROS (7)
Trk receptor (7)
NMDAR (7)
Topoisomerase (6)
Histone Methyltransferase (6)
Tyrosine Kinases (6)
P450 (6)
Akt (6)
Casein Kinase (6)
Mdm2 (6)
Beta Amyloid (6)
FXR (5)
HBV (5)
TAM Receptor (5)
Ras (5)
Opioid Receptor (5)
Proteasome (5)
GABA Receptor (5)
TGF-beta/Smad (5)
Reverse Transcriptase (5)
Chk (5)
AMPK (5)
Lipoxygenase (5)
PDK (5)
Pim (4)
TRP/TRPV Channel (4)
HIF/HIF Prolyl-Hydroxylase (4)
HER (4)
Hydroxylase (4)
Wnt/beta-catenin (4)
PARP (4)
LPL Receptor (4)
IL Receptor (4)
Cannabinoid Receptor (4)
RAAS (4)
Gamma-secretase (4)
Estrogen/progestogen Receptor (4)
S6 Kinase (4)
FAK (4)
TNF (4)
Sirtuin (4)
ERK (4)
BTK (4)
Retinoid Receptor (4)
Sigma receptor (4)
Syk (4)
Serine Protease (4)
Endothelin Receptor (4)
CRM1 (3)
MAPK (3)
LPA Receptor (3)
Cysteine Protease (3)
Serine/threonin kinase (3)
Smo (3)
Proton pump (3)
Complement System (3)
MELK (3)
Virus Protease (3)
c-Fms (3)
MMP (3)
TLR (3)
MRP (3)
Nucleoside Antimetabolite/Analog (3)
NADPH (3)
Nrf2 (3)
Norepinephrine (3)
Mitochondrial Metabolism (3)
Phospholipase (3)
Guanylate cyclase (3)
Hedgehog/Smoothened (3)
Glucocorticoid Receptor (3)
HIF (3)
Glucokinase (3)
JNK (3)
ROCK (3)
Estrogen Receptor/ERR (3)
Aminopeptidase (3)
Integrin (3)
Interleukin (3)
ATPase (3)
PKA (3)
DUB (3)
HCV Protease (3)
ROS Kinase (3)
Prostaglandin Receptor (3)
STING (2)
Reductase (2)
NOS (2)
S1P Receptor (2)
PROTACs (2)
Oxytocin Receptor (2)
transporter (2)
Transferase (2)
Progesterone Receptor (2)
TOPK (2)
ROR (2)
PAI-1 (2)
Vasopressin Receptor (2)
ribosome (2)
Kinesin (2)
Xanthine Oxidase (2)
IRE1 (2)
Ligands for Target Protein for PROTAC (2)
FAAH (2)
Ligand for E3 Ligase (2)
Leukotriene Receptor (2)
Acetyl-CoA Carboxylase (2)
IκB/IKK (2)
IFNAR (2)
Liver X Receptor (2)
CRISPR/Cas9 (2)
HSV (2)
HMG-CoA Reductase (2)
Histone Demethylase (2)
Histone Acetyltransferase (2)
GPR (2)
Caspase (2)
CaSR (2)
NADPH-oxidase (2)
Androgen Receptor (2)
Tie-2 (1)
Adenylyl cyclase (1)
Adenosine deaminase (1)
Wee1 (1)
CSF-1R (1)
AChE (1)
SIK (1)
CXCR (1)
Discoidin Domain Receptor (DDR) (1)
DNA (1)
DNA Alkylation (1)
DNA Methyltransferase (1)
DPP-4 (1)
DprE1 (1)
Ephrin Receptor (1)
advanced glycation end products (1)
Chloride channel (1)
UGT (1)
BCRP (1)
Carbonic Anhydrase (1)
Telomerase (1)
Taste receptor (1)
Carboxypeptidase (1)
Bradykinin Receptor (1)
BMI-1 (1)
ASK (1)
Thrombin (1)
CCR (1)
Aryl Hydrocarbon Receptor (1)
Antioxidant (1)
Antifolate (1)
cell cycle arrest (1)
Amino Acids and Derivatives (1)
Somatostatin (1)
Epoxide Hydrolase (1)
Neurokinin receptor (1)
RIP kinase (1)
OXPHOS (1)
PAFR (1)
Melanocortin Receptor (1)
MLK (1)
MNK (1)
P2Y Receptor (1)
P2X Receptor (1)
Molecular Glues (1)
OX Receptor (1)
PAK (1)
Monoamine Transporter (1)
Monocarboxylate transporter (1)
Na+/Ca2+ Exchanger (1)
NPC1L1 (1)
NAMPT (1)
NEDD8 (1)
NOD-like Receptor (NLR) (1)
NOD (1)
MALT (1)
lysosomal autophagy (1)
Factor Xa (1)
GPCR19 (1)
Rho (1)
FLAP (1)
Gap Junction Protein (1)
Glutathione Peroxidase (1)
GlyT (1)
NO Synthase (1)
gp120/CD4 (1)
PYK2 (1)
LTR (1)
Hippo pathway (1)
IAP (1)
Platelet aggregation (1)
PKM (1)
Isocitrate Dehydrogenase (IDH) (1)
P-gp (1)
PERK (1)
Lipid (1)
GNRH Receptor (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
陶术
生物
TargetMol®中国区唯一合作伙伴
点击进入陶术生物官网陶术生物
联系我们
400-820-0310

上海市静安区江场三路238号8楼