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抗乳腺癌化合物库

抗乳腺癌化合物库

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产品编号 L2191 Anti-Breast Cancer Compound Library
  库化合物信息   Excel SDF

乳腺癌是乳腺恶性肿瘤,是全球女性发病率较高的癌症,约占女性癌症患者的20%,也是100多个国家癌症死亡的主要原因。近年来全球乳腺癌发病率一直呈上升趋势。 乳腺癌根据病理分型可分为非浸润性癌,早期浸润性癌,浸润性癌。根据分子分型可分为雌激素受体阳性乳腺癌(ER+PR+HER2-),HER2阳性乳腺癌(ER-PR-HER2+),三阴性乳腺癌(ER-PR-HER2-)。不同类型的乳腺癌,从治疗方法到预后都是非常不同,需要针对已经明确的致癌位点,探索相关靶点来设计相应的药物。 TargetMol 抗乳腺癌库收集了1965 种与乳腺癌相关的化合物,包含了已经报道的有乳腺癌治疗作用的化合物,以及相关的靶点通路(HER-2, VEGF, EGFR, PARP, CDK4/6, HSP, PD-1, SET7/9, BRCA 等),是乳腺癌药物研发的良好工具。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
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产品描述

  • 1965种与乳腺癌相关的化合物,可以用于抗乳腺癌药物研发和药理研究;
  • 靶点包含HER-2, VEGF, EGFR, PARP, CDK4/6, HSP, PD-1, SET7/9, BRCA等;
  • 部分化合物已上市或已进入临床期;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L2191)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

Apoptosis (357)
Autophagy (266)
NF-κB (228)
CDK (186)
PI3K (173)
Reactive Oxygen Species (165)
EGFR (160)
VEGFR (149)
PPAR (118)
HDAC (105)
Endogenous Metabolite (97)
Akt (94)
mTOR (91)
FGFR (75)
AMPK (73)
Antibacterial (70)
PDGFR (65)
HSP (58)
GSK-3 (57)
PARP (56)
COX (53)
TGF-beta/Smad (52)
FLT (45)
ERK (43)
c-Kit (43)
IκB/IKK (40)
Src (39)
DNA-PK (37)
TNF (32)
p38 MAPK (32)
Parasite (32)
S6 Kinase (30)
Ferroptosis (30)
DNA/RNA Synthesis (30)
HER (30)
STAT (27)
c-Met/HGFR (25)
JNK (25)
HIV Protease (24)
Aurora Kinase (24)
NOD (23)
Mitophagy (23)
Estrogen/progestogen Receptor (23)
RIP kinase (23)
ATM/ATR (23)
Antibiotic (23)
PKC (22)
Estrogen Receptor/ERR (21)
Influenza Virus (21)
IL Receptor (20)
JAK (20)
Bcr-Abl (20)
Antifungal (20)
Caspase (19)
ALK (19)
Topoisomerase (19)
Gamma-secretase (19)
PDK (19)
Wnt/beta-catenin (18)
c-RET (18)
Antioxidant (18)
IRAK (17)
P450 (17)
Potassium Channel (17)
NO Synthase (16)
Calcium Channel (16)
ROS (16)
Raf (16)
Microtubule Associated (15)
MEK (15)
PKA (15)
Lipoxygenase (14)
BCL (14)
PI4K (14)
Dehydrogenase (13)
MMP (13)
NOD-like Receptor (NLR) (13)
IGF-1R (13)
PD-1/PD-L1 (12)
Tyrosinase (12)
Casein Kinase (11)
TAM Receptor (11)
Beta Amyloid (11)
Mitochondrial Metabolism (11)
Interleukin (11)
Chk (11)
Nrf2 (11)
p53 (10)
MAPK (10)
c-Fms (10)
Prostaglandin Receptor (10)
PDE (9)
Trk receptor (9)
Tyrosine Kinases (9)
HIF/HIF Prolyl-Hydroxylase (9)
Sodium Channel (9)
FAK (9)
Virus Protease (8)
NOS (8)
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PTEN (8)
GABA Receptor (8)
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transporter (7)
ROCK (7)
PLK (7)
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SIK (6)
TLR (6)
AChR (6)
P-gp (6)
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CaMK (5)
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Cannabinoid Receptor (4)
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Leukotriene Receptor (3)
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PERK (3)
PGE Synthase (3)
Serine Protease (3)
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cholecystokinin (2)
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GTPase (2)
ABC (2)
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Histone Methyltransferase (2)
MRP (2)
TOPK (2)
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HBV (2)
BACE (2)
BCRP (2)
Survivin (2)
Rho (2)
Glutathione reductase (2)
Reverse Transcriptase (2)
GNRH Receptor (2)
Aminopeptidase (1)
SGLT (1)
CRISPR/Cas9 (1)
Beta-Secretase (1)
Adenosine deaminase (1)
c-Myc (1)
AhR (1)
UGT (1)
cGAS (1)
cAMP (1)
Somatostatin (1)
RSV (1)
cell cycle arrest (1)
ATP Citrate Lyase (1)
Antifolate (1)
CFTR (1)
Thrombin (1)
Smo (1)
Telomerase (1)
PKM (1)
Reductase (1)
Monoamine Oxidase (1)
OCT (1)
NUDIX hydrolase (1)
GST (1)
NPC1L1 (1)
Haspin Kinase (1)
NADPH-oxidase (1)
Hexokinase (1)
Myosin (1)
MNK (1)
Glutaminase (1)
Histone Acetyltransferase (1)
Melatonin Receptor (1)
Mdm2 (1)
Indoleamine 2,3-Dioxygenase (IDO) (1)
LTR (1)
LPL Receptor (1)
Liver X Receptor (1)
Lipase (1)
OXPHOS (1)
GluR (1)
RAR/RXR  (1)
Endothelin Receptor (1)
DAPK (1)
DHFR (1)
Proton pump (1)
DNA Alkylator/Crosslinker (1)
Dopamine Receptor (1)
DUB (1)
Platelet aggregation (1)
KSP (1)
Epoxide Hydrolase (1)
PAD (1)
FAAH (1)
Phospholipase (1)
FLAP (1)
FXR (1)
Gap Junction Protein (1)
Glucokinase (1)
PAK (1)
PAI-1 (1)
YAP (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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