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Search Results for "BPK-29"
Targets Recommended: Others

2

抑制剂 & 化合物

62

化合物库

3

TargetMol 试剂盒

1

仪器耗材

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Cat. No. Product Name
L1710 抗COVID-19化合物库

1160 compounds
1160种对SARS-CoV-2有抑制作用或潜在抑制作用的化合物集合,可用于高通量和高内涵筛选;
L6720 抗COVID-19中药单体库

1162 compounds
根据抗新冠肺炎疫情过程中应用于临床治疗的中药方剂,收集了1162种相关中药来源的单体化合物,可用于高通量和高内涵筛选,是抗新冠病毒药物研发的良好工具;
NY1000 天然产物衍生物库

4000 compounds
22个天然产物骨架,4000个天然产物衍生物;
L4900 心血管毒性化合物库

127 compounds
127种心血管毒性化合物的独特集合,可用于毒理学研究;
L2520 糖代谢化合物库

708 compounds
708种糖代谢相关的化合物,可用于高通量和高内涵筛选;
L9411 半胱氨酸共价化合物库

72 compounds
半胱氨酸共价库包含72个化合物。
L9230 ReFRAME 化合物库

3274 compounds
3274化合物的独特集合,可用于高通量筛选和高内涵筛选
DC1140 特权片段注释化合物库-Ligand-gated

9028 compounds
DC1180 特权片段注释化合物库-Lyases

19530 compounds
DC1150 特权片段注释化合物库-GPCR Family B

9320 compounds
DC1170 特权片段注释化合物库-Oxidoreductases

8812 compounds
DC1190 特权片段注释化合物库-Sigma Opioid receptors

8724 compounds
DC1040 特权片段注释化合物库-Transferases

23001 compounds
DC1030 特权片段注释化合物库-Epigenetics

9196 compounds
DC1100 特权片段注释化合物库-GPCR Frizzled family

3434 compounds
DC1200 特权片段注释化合物库-Isomerases

1206 compounds
DC1050 特权片段注释化合物库-Voltage-gated

17952 compounds
DC1110 特权片段注释化合物库-Proteases

22863 compounds
DC1010 特权片段注释化合物库-GPCR Family A

24763 compounds
DC1000 特权片段注释化合物库

190000 compounds
The database contains 190k small molecules divided into 23 sub libraries each focused at a specific target. According to the recent studies, molecules acting on a particular target or class of targets usually have characteristic moieties (PF) containing key binding points responsible for activity, e.g. hinge-binding fragments. We used this principle for the statistical analysis of the reported active molecules and corresponding targets for the annotation of pre-filtered ChemDiv in house colle...
DC1130 特权片段注释化合物库-Phosphodiesterases

13154 compounds
DC1060 特权片段注释化合物库-Kinases

18350 compounds
DC1220 特权片段注释化合物库-Aminoacyltransferases

3008 compounds
DC1210 特权片段注释化合物库-Phosphatases

15354 compounds
DC1160 特权片段注释化合物库-Toll-like and Il-1 receptors

3536 compounds
DC1090 特权片段注释化合物库-Ligases

11828 compounds
DQ3000 Factor XIa化合物库

6500 compounds
DC1080 特权片段注释化合物库-GPCR Taste family

2675 compounds
DC1120 特权片段注释化合物库-Thrombopoietin receptors

4908 compounds
DC1230 特权片段注释化合物库-Beta amyloid A4 protein

4617 compounds
DC1070 特权片段注释化合物库-GPCR Family C

5071 compounds
DC1020 特权片段注释化合物库-Spiro Library

20563 compounds
L3980 DNA损伤/修复库Plus

667 compounds
667种DNA损伤/修复靶向、结构新颖的化合物;
L4700 免疫/炎症分子化合物库

3483 compounds
3483种具有抗炎症活性的化合物的特有集合,可用于高通量筛选和高内涵筛选;
L2200 酪氨酸激酶分子库

746 compounds
746种酪氨酸激酶抑制剂的独特集合,可用于高通量筛选和高内涵筛选;
L5100 含氟化合物库

583 compounds
583个含氟化合物的独特集合,可用于高通量筛选和高内涵筛选;
L4400 抗生素库

708 compounds
708个具有抗菌活性化合物的独特集合,是医药研究的优良工具库和药物筛选的有效载体;
L2130 抗癌细胞代谢库

1280 compounds
1280种癌细胞代谢相关的生物活性小分子化合物的特有集合,用于肿瘤相关的研究以及抗肿瘤药物的筛选,用于高通量、高内涵筛选;
L6130 萜类天然产物库

349 compounds
349种萜类天然产物的独特集合,可用于高通量筛选和高内涵筛选;
L3600 细胞因子抑制剂库

613 compounds
613个与细胞因子紧密相关的化合物集合,是高通量、高内涵筛选的良好载体;
L8500 HIF-1化合物库

1352 compounds
1352个HIF-1相关小分子的独特集合,可用于缺血性疾病、癌症等相关领域的药物开发和药理研究;
L6700 抗癌天然产物库

1471 compounds
1471种已知活性天然产物的独特集合,是肿瘤药物开发、抗癌先导化合物筛选等领域的有力工具,可用于HTS和HCS。
L2191 抗乳腺癌化合物库

1965 compounds
1965种与乳腺癌相关的化合物,可以用于抗乳腺癌药物研发和药理研究;
L7600 趋化因子抑制剂库

59 compounds
59种趋化因子或其受体抑制剂的独特集合,可用于高通量筛选和高内涵筛选;
DP9100 CB1-2化合物库

CL0140 BTK inhibitor kit

CL0122 ACE inhibitor kit

CL0115 Proton Pump inhibitor kit

CL0127 NOS inhibitor kit

CL0098 HER2 inhibitor kit

CL0128 HMGCR inhibitor kit

CL0150 DNA Methyltransferase/Demethylase inhibitor kit

CL0138 Carbonic Anhydrase inhibitor kit

CL0134 p53 inhibitor/reactivator kit

CL0147 c-FMS inhibitor kit

CL0099 RAR/RXR agonist kit

CL0117 DPP4 inhibitor kit

CL0136 ATM/ATR inhibitor kit

CL0088 Angiotensin Receptor inhibitor kit

CL0148 LPL Receptor antagonist/agonist kit

L1010 FDA上市及药典收录分子库

3158 compounds
3158个上市及药典分子集合,可用于高通量筛选和高内涵筛选;
L9860 抗抑郁症化合物库

1181 compounds
1181种与抑郁症相关的化合物,可以用于高通量和高内涵筛选

化合物库

抗COVID-19化合物库
L1710
Compounds: 1160
抗COVID-19中药单体库
L6720
Compounds: 1162
天然产物衍生物库
NY1000
Compounds: 4000
心血管毒性化合物库
L4900
Compounds: 127
糖代谢化合物库
L2520
Compounds: 708
半胱氨酸共价化合物库
L9411
Compounds: 72
ReFRAME 化合物库
L9230
Compounds: 3274
特权片段注释化合物库-Ligand-gated
DC1140
Compounds: 9028
特权片段注释化合物库-Lyases
DC1180
Compounds: 19530
特权片段注释化合物库-GPCR Family B
DC1150
Compounds: 9320
特权片段注释化合物库-Oxidoreductases
DC1170
Compounds: 8812
特权片段注释化合物库-Sigma Opioid receptors
DC1190
Compounds: 8724
特权片段注释化合物库-Transferases
DC1040
Compounds: 23001
特权片段注释化合物库-Epigenetics
DC1030
Compounds: 9196
特权片段注释化合物库-GPCR Frizzled family
DC1100
Compounds: 3434
特权片段注释化合物库-Isomerases
DC1200
Compounds: 1206
特权片段注释化合物库-Voltage-gated
DC1050
Compounds: 17952
特权片段注释化合物库-Proteases
DC1110
Compounds: 22863
特权片段注释化合物库-GPCR Family A
DC1010
Compounds: 24763
特权片段注释化合物库
DC1000
Compounds: 190000
特权片段注释化合物库-Phosphodiesterases
DC1130
Compounds: 13154
特权片段注释化合物库-Kinases
DC1060
Compounds: 18350
特权片段注释化合物库-Aminoacyltransferases
DC1220
Compounds: 3008
特权片段注释化合物库-Phosphatases
DC1210
Compounds: 15354
特权片段注释化合物库-Toll-like and Il-1 receptors
DC1160
Compounds: 3536
特权片段注释化合物库-Ligases
DC1090
Compounds: 11828
Factor XIa化合物库
DQ3000
Compounds: 6500
特权片段注释化合物库-GPCR Taste family
DC1080
Compounds: 2675
特权片段注释化合物库-Thrombopoietin receptors
DC1120
Compounds: 4908
特权片段注释化合物库-Beta amyloid A4 protein
DC1230
Compounds: 4617
特权片段注释化合物库-GPCR Family C
DC1070
Compounds: 5071
特权片段注释化合物库-Spiro Library
DC1020
Compounds: 20563
DNA损伤/修复库Plus
L3980
Compounds: 667
免疫/炎症分子化合物库
L4700
Compounds: 3483
酪氨酸激酶分子库
L2200
Compounds: 746
含氟化合物库
L5100
Compounds: 583
抗生素库
L4400
Compounds: 708
抗癌细胞代谢库
L2130
Compounds: 1280
萜类天然产物库
L6130
Compounds: 349
细胞因子抑制剂库
L3600
Compounds: 613
HIF-1化合物库
L8500
Compounds: 1352
抗癌天然产物库
L6700
Compounds: 1471
抗乳腺癌化合物库
L2191
Compounds: 1965
趋化因子抑制剂库
L7600
Compounds: 59
CB1-2化合物库
DP9100
Compounds: 0
BTK inhibitor kit
CL0140
Compounds: 0
ACE inhibitor kit
CL0122
Compounds: 0
Proton Pump inhibitor kit
CL0115
Compounds: 0
NOS inhibitor kit
CL0127
Compounds: 0
HER2 inhibitor kit
CL0098
Compounds: 0
HMGCR inhibitor kit
CL0128
Compounds: 0
DNA Methyltransferase/Demethylase inhibitor kit
CL0150
Compounds: 0
Carbonic Anhydrase inhibitor kit
CL0138
Compounds: 0
p53 inhibitor/reactivator kit
CL0134
Compounds: 0
c-FMS inhibitor kit
CL0147
Compounds: 0
RAR/RXR agonist kit
CL0099
Compounds: 0
DPP4 inhibitor kit
CL0117
Compounds: 0
ATM/ATR inhibitor kit
CL0136
Compounds: 0
Angiotensin Receptor inhibitor kit
CL0088
Compounds: 0
LPL Receptor antagonist/agonist kit
CL0148
Compounds: 0
FDA上市及药典收录分子库
L1010
Compounds: 3158
抗抑郁症化合物库
L9860
Compounds: 1181
Cat. No. Product Name Form Specificity Of Inhibition
C0005 Cell Counting Kit-8 (CCK-8)

Cell Counting Kit-8 (CCK-8)

Solution in bottle
C0003 Phosphatase Inhibitor Cocktail II (100× DMSO)

磷酸酶抑制剂 Cocktail II

Solution (100× in DMSO) Alkaline phosphatases, Ser/Thr phosphatases, Acid and PP1 and PP2A
C0002 Phosphatase Inhibitor Cocktail I (100× ddH2O)

磷酸酶抑制剂 Cocktail I

Solution (100× in ddH2O) Acid Phosphatase, Alkaline phosphatase, PTPs, ATPases

TargetMol 试剂盒

Cell Counting Kit-8 (CCK-8)
C0005
磷酸酶抑制剂 Cocktail II
C0003
磷酸酶抑制剂 Cocktail I
C0002
Cat. No. Product Name
EC3000 TargetMol® 24 道磁力架

强力钕磁铁部件,吸附效率高,可兼容所有磁珠。助力核酸分离、蛋白纯化、细胞分选!可同时分离 24管样品,节省实验时间;操作简单,架身美观小巧,价格优惠。

仪器耗材

TargetMol® 24 道磁力架
EC3000
Cat. No. Product Name Target Signaling Pathways
T13586 BPK-29

Others Others
BPK-29 is a specific ligand that disrupts the atypical orphan nuclear receptor NR0B1-protein interactions by covalently modifying C274. It impairs the anchorage-independent growth of KEAP1-mutant cancer cells.
T13586L BPK-29 hydrochloride

Others Others
BPK-29 hydrochloride 是特殊配体,能够共价修饰 C274 ,破坏非典型孤核受体NR0B1与RBM45、SNW1蛋白质的相互作用。它能够损害KEAP1突变癌细胞的锚定独立生长。

化合物

BPK-29
T13586
synonym:
Target: Others
BPK-29 hydrochloride
T13586L
synonym:
Target: Others