Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TP1940 | Ac-RYYRIK-NH2 | ||
High affinity ligand for the NOP site (Ki = 1.5 nM). Antagonizes nociceptin-stimulated GTP binding in rat brain and the chronotropic effect of nociceptin on rat cardiomyocytes. However, displays potent agonist properties in vivo, inhibiting locomotor acti |