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TargetMol产品目录中 "

thromboxane

"的结果
  • 抑制剂&激动剂
    133
    TargetMol | Inhibitors_Agonists
  • 化合物库
    1
    TargetMol | Compound_Libraries
  • 重组蛋白
    1
    TargetMol | Recombinant_Protein
  • 多肽产品
    1
    TargetMol | Peptide_Products
  • 天然产物
    9
    TargetMol | Natural_Products
  • 同位素
    3
    TargetMol | Isotope_Products
  • 分子与细胞研究
    1
    TargetMol | Inhibitors_Agonists
  • NTP42
    T122682055599-51-2
    NTP42 是血栓素 A2 (TXA2) 受体的拮抗剂,IC50为 3.278 nM,可用于肺动脉高压的相关研究。
    • ¥ 493
    In stock
    规格
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  • Thromboxane A2
    Rabbit aorta contracting substance,TXA-2,TXA2,TXA 2
    T3486257576-52-0
    Thromboxane A2, as an unstable intermediate between the prostaglandin endoperoxides and thromboxane B2, is a potent inducer of platelet aggregation and causes vasoconstriction.
    • 待询
    8-10周
    规格
    数量
  • 15(R)-Pinane Thromboxane A2
    15(R)-Pinane Thromboxane A2
    T3620871154-83-1
    15(R)-Pinane thromboxane A2 is the (R)-epimer of pinane thromboxane A2 . 15(R)-PTA2 does not inhibit collagen-induced platelet aggregation (IC50s = 120-130 μM). It does not affect gastric tone in isolated rat gastric fundus when used at concentrations of 0.5 or 1.5 μg ml and is less effective than PTA2 at inhibiting prostaglandin-induced contraction of isolated rat stomach muscle.
    • 待估
    35日内发货
    规格
    数量
  • 2,3-dinor Thromboxane B1
    2,3-dinor Thromboxane B1
    T36220196493-76-2
    Thromboxane B2 (TXB2) is released in substantial quantities from aggregating platelets and metabolized during circulation to 11-dehydro TXB2 and 2,3-dinor TXB2. In rats and rabbits, 2,3-dinor TXB1 has been identified as another urinary metabolite of TXB2. However in human urine, only trace amounts of 2,3-dinor TXB1 have been identified. In rats, 2,3-dinor TXB1 is excreted at a much higher rate than 2,3-dinor TXB2 (19.2 ± 4.9 ng/24 hr and 1.6 ± 0.3 ng/24 hr, respectively). Therefore, urinary 2,3-dinor TXB1 is a suitable marker of thromboxane biosynthesis in rats.
    • 待估
    35日内发货
    规格
    数量
  • Carbocyclic Thromboxane A2
    T3654874034-56-3
    Carbocyclic Thromboxane A2 可用于生命科学领域的相关研究。其产品编号为 T36548,CAS号为 74034-56-3。
    • 待询
    规格
    数量
  • Thromboxane B2
    T4124654397-85-2
    Thromboxane B2 是一种在过敏反应期间释放的前列腺素衍生物。Thromboxane B2 诱导动脉收缩和血小板聚集。
    • 待询
    6-8周
    规格
    数量
  • Thromboxane B1
    T7385564626-32-0
    Thromboxane B1 (TXB1) 是TXB家族中的一员,属于类花生酸脂质家族。该家族因参与血栓形成而得名。
    • 待估
    35日内发货
    规格
    数量
  • Thromboxane B3
    Δ17-TXB2
    T8456971953-80-5
    Thromboxane B3 (TXB3), the stable hydrolysis product of TXA3, is synthesized from eicosapentaenoic acid (EPA) through the action of COX and thromboxane synthase enzymes. This compound is biosynthesized in several tissues, including seminal vesicles, lungs, polymorphonuclear leukocytes (PMNL), and ocular tissues.
    • 待询
    8-10周
    规格
    数量
  • 11-dehydro Thromboxane B3
    11-dehydro TXB3
    T84570129228-55-3
    11-Dehydro Thromboxane B3 (11-dehydro TXB3) serves as a urinary metabolite of TXA3 in humans following an increased dietary intake of EPA.
    • 待询
    8-10周
    规格
    数量
  • 2,3-dinor Thromboxane B2
    2,3-dinor TXB2
    T8462663250-09-9
    Thromboxane B2 (TXB2) is a compound significantly released from aggregating platelets and undergoes metabolic transformation during circulation into 11-dehydro TXB2 and 2,3-dinor TXB2. The latter, 2,3-dinor TXB2, serves as a prevalent urinary metabolite of TXB2 and acts as an indicator for in vivo TXA2 synthesis. Studies have shown that in healthy male volunteers, the median excretion rate of 2,3-dinor TXB2 is measured at 10.3 ng hour, equivalent to 138 pg mg of creatinine.
    • 待询
    8-10周
    规格
    数量
  • 11-dehydro-2,3-dinor Thromboxane B2
    11-dehydro-2,3-dinor TXB2
    T8462779250-60-5
    11-Dehydro-2,3-dinor Thromboxane B2 (11-dehydro-2,3-dinor TXB2) is a metabolite derived from the inactive TXA2 metabolite, TXB2. Its formation involves the action of cytosolic aldehyde dehydrogenase (ALDH) and β-oxidation processes. Remarkably, levels of 11-dehydro-2,3-dinor TXB2 have been observed to increase by 5.2-fold in a surgery-induced rat model of tendon overuse, highlighting its potential role in physiological stress responses.
    • 待询
    8-10周
    规格
    数量
  • Imitrodast
    咪曲司特
    T68086114686-12-3In house
    Imitrodast是一种小分子血栓素A2合成酶(TXA2 synthase)抑制剂,可用于治疗免疫系统疾病、呼吸系统疾病和心血管疾病,可用于研究动脉血栓形成、哮喘和冠状血管痉挛。
    • ¥ 893
    In stock
    规格
    数量
    TargetMol | Inhibitor Sale
  • Ozagrel
    奥扎格雷, OKY-046, Domenan
    T623682571-53-7
    Ozagrel (Domenan) 是血栓烷 A2(TXA2) 合酶抑制剂,可抑制哮喘。它也是一种抗血小板剂,可选择性抑制人血小板聚集,IC50为 53.12 μM。
    • ¥ 145
    In stock
    规格
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  • p-Hydroxycinnamic acid
    对羟基肉桂酸, p-Hydroxy-cinnamic acid, p-Cumaric acid, p-Coumaric acid, NSC 59260
    T70537400-08-0
    p-Hydroxycinnamic acid (NSC-59260) 是常见的食用酚,可抑制血小板活性,对血栓素 B2 和前列腺素 E2 的 IC50值分别为 371 和 126 μM。
    • ¥ 140
    In stock
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  • RS-601
    T12771207987-59-5In house
    RS-601 是一种有效的 leukotriene D4 thromboxane A2 双重抑制剂,对抗原诱导的气道高反应性 (AHR)有抑制作用且在豚鼠哮喘模型中显示出平喘作用。
    • ¥ 4900
    In stock
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  • AZ-1355
    T1356375451-07-9In house
    AZ-1355是一种新型二苯并恶西平衍生物,具有降脂效果。
    • ¥ 630
    In stock
    规格
    数量
    TargetMol | Inhibitor Sale
  • Terbogrel
    BIBV 308SE, 特波格雷
    T17039149979-74-8In house
    Terbogrel 是一种可口服的 、具有选择性 thromboxane A2 受体拮抗剂(IC50 约为 10 nM),是一种 thromboxane A2 synthase 抑制剂(IC50 约为 10 nM)。Terbogrel 是一种抗血小板化合物,可抑制血小板聚集,是预防血栓的潜在化合物。
    • ¥ 780
    In stock
    规格
    数量
    TargetMol | Inhibitor Sale
  • Isbogrel
    CV4151, CV-4151, CV 4151, 伊波格雷
    T2763089667-40-3In house
    Isbogrel (CV4151)是一种小分子血栓素A2合成酶(TXA2 synthase)抑制剂,可用来研究心律失常、短暂性脑缺血发作和血栓形成。
    • ¥ 2350
    In stock
    规格
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  • Dazmegrel HCl
    UK-38,485 HCl, Dazmegrel HCl(76894-77-4 Free base)
    T31213L In house
    Dazmegrel HCl 是一种血小板血栓素抑制剂,可用于研究心肌梗死和心律失常。
    • ¥ 1300
    In stock
    规格
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  • Pirmagrel
    吡吗格雷
    T6795885691-74-3In house
    pirmagrel 是一种强效的血栓素合酶抑制剂。
    • ¥ 525
    In stock
    规格
    数量
  • Pirodomast
    吡咯司特
    T67959108310-20-9In house
    Pirodomast 是血栓素 A(TXA2)合成酶抑制剂。Pirodomast 能抑制白三烯(LT)D4、C4、E4 的形成和血栓素 B2(TXB2)的活性,但对组胺、甲氧胆碱、血清素、LTC4 或血小板活化因子诱导的豚鼠支气管痉挛的拮抗作用较弱或无效。Pirodomast 在体外对豚鼠气管只有微弱的松弛活性。Pirodomast 是一种潜在的抗过敏化合物,在体外可抑制胰蛋白酶的蛋白水解活性,在体内可阻止抗原诱发过敏绵羊的即时和晚期哮喘反应,抑制抗原诱导的过敏绵羊对组胺和卡巴胆碱的气道高反应性。
    • ¥ 678
    In stock
    规格
    数量
    TargetMol | Inhibitor Sale
  • Ozagrel hydrochloride
    Ozagrel HCl, 盐酸奥扎格雷, OKY-046 HCl
    T662578712-43-3
    Ozagrel hydrochloride (OKY-046 HCl) 是一种选择性血栓素 A(2) 合成酶抑制剂,用于改善术后脑血管收缩和伴随的脑缺血。它是一种抗血小板剂,可选择性抑制人血小板聚集,IC50为 53.12 μM。
    • ¥ 148
    In stock
    规格
    数量
  • NP-313
    NSC-4264, NSC4264, NSC 4264, NP 313
    T245425397-78-4
    NP-313 (NSC-4264) 是一种有效的抗血栓剂,对血栓素 A 2 合成和选择性抑制由 SOCC 介导的 Ca 2+ 内流有抑制作用,可以抑制血小板的聚集和活化。
    • ¥ 497
    In stock
    规格
    数量
    TargetMol | Inhibitor Sale
  • Astragalus polyphenols
    芪多酚, Astragalus polyphenols, 2,3,5,4'-Tetrahydroxystilbene-2-O-b-D-glucopyranoside, 2,3,5,4'-Tetrahydroxystilbene 2-O-β-D-glucoside, 2,3,4',5-Tetrahydroxystilbene 2-O-D-glucoside
    T296482373-94-2
    2,3,5,4'-Tetrahydroxystilbene 2-O-β-D-glucoside (Astragalus polyphenols) 是分离自蓼属植物物种的根中,对5-HETE、HHT、thromboxane B2的形成具有抑制作用。
    • ¥ 123
    In stock
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