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表型筛选靶点鉴定库

表型筛选靶点鉴定库

现 货
产品编号 L9500 Target-Focused Phenotypic Screening Library
  库化合物信息   Excel SDF

TargetMol 表型筛选靶点鉴定库是专为表型筛选的科研工作者提供的,众所周知,表型筛选中的体外筛选,通常以细胞作为筛选工具,优点是对于靶点还不明晰,或靶点与疾病之间的关系还不明确时的药物开发,具有非常好的效果,常用于 First-in-class 药物的研发。而活性化合物的发现与靶标的鉴定两者间实现无缝对接,是学术界和产业界关注的焦点和难点。

选用靶点明确的已知活性化合物进行表型筛选,可以缩小后期靶点确认的范围,是一种较好的基于表型进行靶点鉴定的方式。该库针对表型筛选后难以确定靶点作用机制的痛点,精选了对600多个药物靶点有明确活性的 1832 个小分子组成了该化合物库。每个靶点采取2-4个结构差异较大的化合物,把表型筛选和靶点作用机制判断融为一体,是表型筛选的有力工具。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
咨询化合物库
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产品描述

  • 1832种靶点明确的已知活性化合物,适合表型筛选;
  • 覆盖600多个药物靶点,多样性好,覆盖度广,使用方便;
  • 每个靶点对应2-4个结构差异较大的化合物,提高靶点确认的成功率;
  • 详细的说明书,化合物结构、靶点信息、活性描述,方便科学家对结果进行分析;
  • NMR、HPLC/LCMS多重严苛出厂检测,保证产品结构准确,纯度高,保障实验顺利进行。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L9500)
点击图片重新获取验证码

客户使用化合物库发表的文献

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化合物库组成

Apoptosis (272)
Autophagy (260)
Endogenous Metabolite (93)
Antibacterial (91)
5-HT Receptor (71)
Antibiotic (59)
AChR (53)
DNA/RNA Synthesis (52)
Adrenergic Receptor (50)
P450 (45)
VEGFR (45)
Dopamine Receptor (44)
HIV Protease (40)
PI3K (36)
Epigenetic Reader Domain (36)
PDE (34)
COX (32)
FGFR (32)
PDGFR (31)
Influenza Virus (31)
Histamine Receptor (31)
CDK (30)
Ferroptosis (30)
Parasite (29)
FLT (28)
NF-κB (28)
Potassium Channel (27)
c-Kit (27)
TRP/TRPV Channel (27)
Src (27)
PPAR (24)
Histone Methyltransferase (24)
HCV Protease (24)
GluR (24)
Raf (24)
Reactive Oxygen Species (23)
EGFR (23)
Calcium Channel (23)
Dehydrogenase (23)
TGF-beta/Smad (22)
Mitophagy (22)
Microtubule Associated (22)
JAK (21)
SARS-CoV (20)
HDAC (20)
Topoisomerase (20)
BCL (20)
Estrogen/progestogen Receptor (19)
mTOR (19)
Adenosine Receptor (19)
GABA Receptor (19)
GPR (18)
Sodium Channel (18)
Beta Amyloid (18)
Bcr-Abl (18)
c-Met/HGFR (18)
MAO (17)
p38 MAPK (17)
PKC (17)
Antifungal (17)
IL Receptor (16)
Wnt/beta-catenin (16)
ALK (16)
RAAS (16)
Opioid Receptor (16)
Proteasome (16)
Retinoid Receptor (16)
Estrogen Receptor/ERR (15)
TNF (15)
Carbonic Anhydrase (15)
E1/E2/E3 Enzyme (15)
IκB/IKK (15)
MMP (15)
Prostaglandin Receptor (14)
STAT (14)
GSK-3 (14)
Monoamine Oxidase (14)
DNA Alkylator/Crosslinker (14)
Virus Protease (14)
Akt (14)
Gamma-secretase (13)
ROR (13)
ATPase (13)
ERK (13)
Sirtuin (13)
NMDAR (12)
Phosphatase (12)
Aurora Kinase (12)
c-RET (12)
P2 Receptor (12)
CXCR (12)
HSV (12)
NADPH (12)
HSP (12)
DNA Alkylation (12)
Interleukin (12)
Trk receptor (11)
S1P Receptor (11)
PKA (11)
iGluR (11)
Glucokinase (11)
HIF/HIF Prolyl-Hydroxylase (11)
Serine Protease (11)
Lipoxygenase (11)
MEK (11)
ribosome (11)
Caspase (11)
Nucleoside Antimetabolite/Analog (11)
DUB (10)
DNA Methyltransferase (10)
Chk (10)
Casein Kinase (10)
JNK (10)
Glucocorticoid Receptor (10)
PARP (10)
Indoleamine 2,3-Dioxygenase (IDO) (10)
ROCK (10)
Hedgehog/Smoothened (10)
Phospholipase (9)
AMPK (9)
P-gp (9)
LPL Receptor (9)
Norepinephrine (9)
Reverse Transcriptase (9)
SGLT (9)
ATM/ATR (9)
Serine/threonin kinase (9)
Cannabinoid Receptor (9)
Serotonin Transporter (9)
CaMK (9)
CFTR (8)
AChE (8)
PLK (8)
p53 (8)
Syk (8)
Cysteine Protease (8)
DNA-PK (8)
Drug Metabolite (8)
Ras (8)
Endothelin Receptor (8)
TLR (8)
c-Fms (8)
S6 Kinase (8)
Transferase (8)
HIF (8)
HBV (8)
HER (8)
Aryl Hydrocarbon Receptor (7)
Monocarboxylate transporter (7)
Proton pump (7)
CCR (7)
Reductase (7)
Thyroid hormone receptor(THR) (7)
TAM Receptor (7)
HMG-CoA Reductase (7)
NOS (7)
Tyrosine Kinases (6)
AhR (6)
NOD (6)
Mdm2 (6)
Mitochondrial Metabolism (6)
Histone Acetyltransferase (6)
ROS (6)
OX Receptor (6)
FAK (6)
Rho (6)
Acyltransferase (6)
Chloride channel (6)
Smo (6)
Sigma receptor (6)
Lipase (6)
PDK (6)
PKM (6)
BTK (6)
Aromatase (6)
PAK (5)
PD-1/PD-L1 (5)
DNA gyrase (5)
DNA (5)
PERK (5)
DPP-4 (5)
NAMPT (5)
DHFR (5)
Telomerase (5)
Histone Demethylase (5)
Phosphorylase (5)
IDO (5)
Androgen Receptor (5)
MAPK (5)
MRP (5)
Factor Xa (5)
LRRK2 (5)
FAAH (5)
Kinesin (5)
FXR (5)
ATP Citrate Lyase (5)
IGF-1R (5)
Glutathione Peroxidase (5)
BACE (4)
Acetyl-CoA Carboxylase (4)
GPCR19 (4)
RIP kinase (4)
PAI-1 (4)
transporter (4)
ABC (4)
BMI-1 (4)
PGE Synthase (4)
Tie-2 (4)
Lipid (4)
Xanthine Oxidase (4)
IRE1 (4)
p97 (4)
Porcupine (4)
CAT (4)
NO Synthase (4)
Monoamine Transporter (4)
Ephrin Receptor (4)
Annexin A (4)
Progesterone Receptor (4)
Fatty Acid Synthase (4)
Tyrosinase (4)
Melatonin Receptor (4)
NOD-like Receptor (NLR) (4)
cAMP (4)
CaSR (4)
LTR (4)
CSF-1R (4)
MNK (4)
UGT (3)
Survivin (3)
RSV (3)
PTEN (3)
STING (3)
IRAK (3)
Pim (3)
Na+/Ca2+ Exchanger (3)
ACK (3)
advanced glycation end products (3)
Cell wall (3)
CETP (3)
c-Myc (3)
DprE1 (3)
Free radical scavengers (3)
Hydroxylase (3)
Leukotriene Receptor (3)
LIM Kinase (3)
Liver X Receptor (3)
GNRH Receptor (3)
Neurokinin receptor (3)
P2X Receptor (3)
Neprilysin (3)
Pyroptosis (2)
Carboxypeptidase(CPG2) (2)
Gap Junction Protein (2)
DYRK (2)
Myosin (2)
CRISPR/Cas9 (2)
Thrombin (2)
BCRP (2)
Beta-Secretase (2)
GlyT (2)
Antiviral (2)
Antioxidant (2)
Antifolate (2)
Antifection (2)
Vasopressin Receptor (2)
Wee1 (2)
PAFR (2)
GluCls (2)
Stearoyl-CoA Desaturase (SCD) (2)
PI4K (2)
Protease-activated Receptor (2)
MTH1 (2)
MT Receptor (2)
MLK (2)
LPA Receptor (2)
NADPH-oxidase (2)
LDL (2)
Integrin (2)
IFNAR (2)
YAP (2)
GRK (2)
OCT (1)
lysosomal autophagy (1)
SGK (1)
Adenosine deaminase (1)
GPX (1)
Adenylyl cyclase (1)
PAD (1)
VDA (1)
Amino Acids and Derivatives (1)
Aminopeptidase (1)
GST (1)
Nrf2 (1)
Anti-infection (1)
Hck (1)
Na-K-Cl cotransporter (1)
Arginase (1)
Glutathione reductase (1)
Neuropeptide Y Receptor (1)
Discoidin Domain Receptor (DDR) (1)
Hippo pathway (1)
IAP (1)
ASK (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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