首页工具

登录

搜索结果

Search Results for " besylate "

如果没找到您满意的产品或者您对产品有其他要求，可以联系我们专业顾问为您提供针对性的合理建议。 QQ咨询网站留言咨询

Cat. No.	Product Name	Target	Signaling Pathways
T6177	PF-562271 besylate PF-00562271 Besylate	FAK; PYK2; CDK	Angiogenesis; Cell Cycle/Checkpoint; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors
	PF-562271 besylate (PF-00562271 Besylate) 是一种可逆的，有效的，ATP 竞争性的 FAK(IC50:1.5 nM)和 Pyk2 (IC50:13 nM)激酶抑制剂。
T4284	Levamlodipine besylate 左旋氨氯地平,(S)-Amlodipine Besylate (103129-82-4(free base))	Calcium Channel	Membrane transporter/Ion channel; Metabolism
	Levamlodipine besylate ((S)-Amlodipine Besylate(103129-82-4(free base))) 是一种二氢吡啶钙通道阻滞剂，具有舒张血管的作用，可用于高血压和心绞痛的研究。
T6397	Atracurium besylate Tracrium,51W89,BW-33A,苯磺酸阿曲库铵	AChR	Neuroscience
	Atracurium besylate (51W89) 是一种神经肌肉阻断剂，ED95为0.2 mg/kg。
T1459	Cisatracurium besylate 顺苯磺酸阿曲库铵,顺苯磺阿曲库铵,51W89	Adrenergic Receptor; AChR; Autophagy	Autophagy; GPCR/G Protein; Neuroscience
	Cisatracurium besylate (51W89) 是一种用于静脉内给药的非去极化骨骼肌松弛剂。
T0231	Amlodipine Besylate Amlodipine benzenesulfonate,苯磺酸氨氯地平	Calcium Channel	Membrane transporter/Ion channel; Metabolism
	Amlodipine Besylate (Amlodipine benzenesulfonate) 是可口服的二氢吡啶钙通道阻滞剂，有抗心绞痛作用。它通过阻断电压依赖性的 L 型钙通道，从而抑制钙离子内流，用于高血压和癌症的研究。
T3086	Mesoridazine Besylate Mesoridazine benzenesulfonate,Serentil,苯磺酸美索达嗪	Dopamine Receptor; 5-HT Receptor	GPCR/G Protein; Neuroscience
	Mesoridazine Besylate (Serentil) 是一种哌啶类精神安定药，属于称为吩噻嗪类的药物，用于治疗精神分裂症。它是硫利达嗪的代谢物。
T6174	R406 R-406 besylate	Apoptosis; FLT; Syk	Angiogenesis; Apoptosis; Tyrosine Kinase/Adaptors
	R406 (R-406 besylate) 是一种具有口服活性的 ATP 竞争性 Syk/FLT3抑制剂，Ki 为 30 nM。它有效抑制 Syk 激酶活性，IC50为 41 nM。它还抑制 Lyn 和 Lck，IC50值分别为 63 nM 和 37 nM。它可减轻免疫复合物介导的炎症。
T11472L	Molibresib besylate I-BET 762 besylate,GSK 525762C	CCR	Immunology/Inflammation; Microbiology/Virology
	Molibresib besylate is an inhibitor of BET bromodomain (IC50: 32.5-42.5 nM).
T14357	Spebrutinib besylate CC-292 (besylate),AVL-292 (benzenesulfonate)	BTK	Angiogenesis; Tyrosine Kinase/Adaptors
	Spebrutinib besylate (AVL-292 benzenesulfonate; CC-292 besylate) is a Btk kinase activity inhibitor (IC50<0.5 nM, Kinact/Ki=7.69×104 M-1s-1s).
T68567	AMG-131 besylate
	AMG-131 besylate is a hypoglycemic agent. It is a potent PPARγ partial agonist that displays robust glucose-lowering activity in rodent models of diabetes while exhibiting a reduced side-effects profile compared to marketed TZDs.
T70158	Quilseconazole besylate
	Quilseconazole besylate, also known as VT-1129 besylate, is a potent, orally active fungal Cyp51 (lanosterol 14-α-demethylase) inhibitor.
T31647	Epelsiban besylate GSK-557296B,GSK557296B
	Epelsiban Besylate is an oral drug that is a highly selective anamol oxytocin receptor antagonist.
T11400	Gisadenafil besylate UK 369003-26	Others	Others
	Gisadenafil besylate (UK 369003-26) is a specific, orally active phosphodiesterase 5 (PDE5) inhibitor ,prevents degradation of cyclic guanosine monophosphate (cGMP), with an IC50 of 3.6 nM .
T69399	MK-0359 besylate
	MK-0359 besylate is a Phosphodiesterase-4 (PDE4) inhibitor.
T10589	BPN-15606 besylate (1914989-49-3 free base) BPN-15606 besylate	Others	Others
	BPN-15606 besylate is a highly potent, orally active γ-secretase modulator, attenuates the production of Aβ40 and Aβ42 by SHSY5Y neuroblastoma cells (IC50s: 7 nM and 17nM).
T0231L3	Amlodipine besylate monohydrate
	Amlodipine besylate monohydrate is a medication used to lower blood pressure and prevent chest pain.
T78217	(R)-Azasetron besylate SENS-401	Phosphatase	Metabolism
	(R)-Azasetron besylate (SENS-401)是一种口服活性的钙调神经磷酸酶抑制剂，能够减轻Cisplatin引发的听力损失和耳蜗损害。
T30001	Amlodipine besylate, (R)-
	Amlodipine besylate, (R)- is a medication used to lower blood pressure and prevent chest pain.
T64425	Crenolanib besylate
	Crenolanib besylate 是一种有用的有机化合物，可用于生命科学领域的相关研究，其产品编号为 T64425。
T61434	Mirogabalin besylate
	Mirogabalin besylate is a potent and orally active ligand that selectively targets the α2δ subunit of voltage-gated calcium channels. It displays high affinity (K d ) values, namely 13.5 nM, 22.7 nM, 27 nM, and 47.6 nM, for human α2δ-1, human α2δ-2, rat α2δ-1, and rat α2δ-2, respectively.
T68451	AG-28262 besylate
	AG-28262 besylate is a VEGFR-2 Inhibitorwhich may affect alanine aminotransferase gene expression and enzymatic activity in the liver.
T64081	BPN-15606 besylate
	BPN-15606 besylate 是一种高效的、口服具有活力的 γ-secretase 调节剂 (GSM)，能够减少 SHSY5Y 神经母细胞瘤细胞产生 Aβ42 (IC50: 7 nM) 和 Aβ40 (IC50: 17 nM) 的作用。BPN-15606 besylate 能够减少大鼠和小鼠中枢神经系统中的 Aβ42 和 Aβ40 水平。BPN-15606 besylate 表现出良好的 PK/PD 特性（包括生物利用度，半衰期和清除率）。
T29706	AG28262 free base AG28262,AG-28262,AG 28262,AG-28262 besylate
	AG28262 is a VEFG-2 inhibitor that increases serum ALT, due in part to both gene up-regulation.
T70157	GGTI-297
	GGTI-297 is a potent, cell-permeable, and selective peptidomimetic inhibitor of GGTase I compared to Farnesyl Transferase (FTase).
T69432	Avanafil dibesylate
	Avanafil dibesylate is a PDE5 inhibitor.
T36006	Olmesartan medoxomil impurity C
	Olmesartan medoxomil impurity C is an Olmesartan medoxomil impurity. Olmesartan medoxomil is a potent and selective angiotensin AT1 receptor inhibitor with IC50 of 66.2 μM. [1]. Senda A, et al. Effects of Angiotensin II Receptor Blockers on Metabolism of Arachidonic Acid via CYP2C8. Biol Pharm Bull. 2015;38(12):1975-9. [2]. Shah S, et al. Simultaneous Quantitative Analysis of Olmesartan Medoxomil and Amlodipine Besylate in Plasma by High-performance Liquid Chromatography Technique. J Young Phar...

化合物

PF-562271 besylate

Cat.No: T6177

Synonym: PF-00562271 Besylate

Target: FAK, PYK2, CDK

Levamlodipine besylate

Cat.No: T4284

Synonym: 左旋氨氯地平,(S)-Amlodipine Besylate (103129-82-4(free base))

Target: Calcium Channel

Atracurium besylate

Cat.No: T6397

Synonym: Tracrium,51W89,BW-33A,苯磺酸阿曲库铵

Target: AChR

Cisatracurium besylate

Cat.No: T1459

Synonym: 顺苯磺酸阿曲库铵,顺苯磺阿曲库铵,51W89

Target: Adrenergic Receptor, AChR, Autophagy

Amlodipine Besylate

Cat.No: T0231

Synonym: Amlodipine benzenesulfonate,苯磺酸氨氯地平

Target: Calcium Channel

Mesoridazine Besylate

Cat.No: T3086

Synonym: Mesoridazine benzenesulfonate,Serentil,苯磺酸美索达嗪

Target: Dopamine Receptor, 5-HT Receptor

Cat.No: T6174

Synonym: R-406 besylate

Target: Apoptosis, FLT, Syk

Molibresib besylate

Cat.No: T11472L

Synonym: I-BET 762 besylate,GSK 525762C

Target: CCR

Spebrutinib besylate

Cat.No: T14357

Synonym: CC-292 (besylate),AVL-292 (benzenesulfonate)

Target: BTK

AMG-131 besylate

Cat.No: T68567

Quilseconazole besylate

Cat.No: T70158

Epelsiban besylate

Cat.No: T31647

Synonym: GSK-557296B,GSK557296B

Gisadenafil besylate

Cat.No: T11400

Synonym: UK 369003-26

Target: Others

MK-0359 besylate

Cat.No: T69399

BPN-15606 besylate (1914989-49-3 free base)

Cat.No: T10589

Synonym: BPN-15606 besylate

Target: Others

Amlodipine besylate monohydrate

Cat.No: T0231L3

(R)-Azasetron besylate

Cat.No: T78217

Synonym: SENS-401

Target: Phosphatase

Amlodipine besylate, (R)-

Cat.No: T30001

Crenolanib besylate

Cat.No: T64425

Mirogabalin besylate

Cat.No: T61434

AG-28262 besylate

Cat.No: T68451

BPN-15606 besylate

Cat.No: T64081

AG28262 free base

Cat.No: T29706

Synonym: AG28262,AG-28262,AG 28262,AG-28262 besylate

Cat.No: T70157

Avanafil dibesylate

Cat.No: T69432

Olmesartan medoxomil impurity C

Cat.No: T36006

我们的所有产品和服务仅用于科学研究，不能被用于人体，我们也不向个人提供产品和服务。

Copyright © 2015-2024 TargetMol Chemicals Inc. All rights reserved. 沪ICP备20019793号-4

沪公网安备 31010602006700号

沪公网安备 31010602006700号

TargetMol Loading

联系我们

电话：

400-820-0310

邮箱：

service@tsbiochem.com

QQ：

2881945090（终端用户）

2885109491（经销商）

经销：

终端：

地址：

上海市静安区江场三路238号8楼