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Search Results for "a-7 hydrochloride"
Targets Recommended: CaMK

34

抑制剂 & 化合物

2

天然产物

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Cat. No. Product Name Target Signaling Pathways
T22538 A-7 hydrochloride

CaMK Neuroscience
A-7 hydrochloride 是一种钙调蛋白拮抗剂,会引起 MDA-MB-231细胞中 CD44+CD24-亚群的改变。
T20792 W-7 hydrochloride

N-(6-氨基己基)-5-氯-1-萘磺胺盐酸盐,W-7 HCl,W 7 HCl,W7 HCl

CaMK; Apoptosis; Myosin; PDE Apoptosis; Cytoskeletal Signaling; Metabolism; Neuroscience
W-7 hydrochloride 是一种选择性的钙调蛋白拮抗剂。它抑制Ca2+-钙调蛋白依赖性磷酸二酯酶和肌球蛋白轻链激酶,IC50值分别为 28 μM 和 51 μM。它可诱导细胞凋亡,具有抗癌活性。
T28531 Facinicline hydrochloride

RG3487

AChR; 5-HT Receptor GPCR/G Protein; Neuroscience
Facinicline hydrochloride 是一种口服有效的烟碱α7 receptor 部分激动剂,对人 nAChR 的 Ki 值为 6 nM。它可改善啮齿类动物的认知和感觉运动门控。它与5-HT3受体结合的 Ki 为 1.2 nM。
T10883L CRA-026440 hydrochloride

CRA-026440 hydrochloride(847460-34-8 Free base)

HDAC Chromatin/Epigenetic; DNA Damage/DNA Repair
CRA-026440 hydrochloride 是有效的、广谱的 HDAC 抑制剂。CRA-026440 hydrochloride 作用于 HDAC1,HDAC2,HDAC3,HDAC6,HDAC8 和 HDAC10, Ki 值分别为 4 nM,14 nM,11 nM,15 nM,7 nM 和 20 nM。CRA-026440 hydrochloride 具有抗血管生成和抗肿瘤活性。
T1400 Demeclocycline hydrochloride

Detravis,Clortetrin,地美环素,盐酸地美环素,Demeclocycline HCl,Declomycin

Antibiotic; ribosome; Antibacterial Microbiology/Virology
Demeclocycline hydrochloride 是四环素类抗生素,可治疗粉刺,莱姆病和支气管炎。
T6010 Idarubicin hydrochloride

盐酸伊达比星,伊达比星盐酸盐,Zavedos,Idarubicin HCl,4-demethoxydaunorubicin (NSC256439, 4-DMDR) HCl,Idamycin,4-Demethoxydaunorubicin hydrochloride

Autophagy; Antibacterial; Topoisomerase; Antifungal Autophagy; DNA Damage/DNA Repair; Microbiology/Virology
Idarubicin HCl 是一种蒽环类抗白血病药物,能抑制细菌和酵母菌生长,还抑制拓扑异构酶 II,干扰 DNA 复制和 RNA 转录。
T0486L Irinotecan Hydrochloride

盐酸伊立替康,伊立替康盐酸盐,Camptothecin 11 hydrochloride,CPT-11 hydrochloride

Topoisomerase; Autophagy Autophagy; DNA Damage/DNA Repair
Irinotecan Hydrochloride 是喜树碱半合成衍生物的盐酸盐,是一种拓扑异构酶 I 抑制剂,可研究结肠癌和直肠癌。
T4261 BPR1J-097 hydrochloride (1327167-19-0(free base))

FLT Angiogenesis; Tyrosine Kinase/Adaptors
BPR1J-097 hydrochloride (1327167-19-0(free base)) 是一种新型小分子 FLT-3抑制剂(IC50=11±7 nM),具有很好的体内抗肿瘤活性。
T5164 Cabozantinib hydrochloride

Cabozantinib hydrochloride (849217-68-1(free base)),BMS-907351,XL184,盐酸卡博替尼

c-Met/HGFR; TAM Receptor; ROR; VEGFR; FLT; c-Kit Angiogenesis; Metabolism; Tyrosine Kinase/Adaptors
Cabozantinib hydrochloride 是一种有效的泛酪氨酸激酶抑制剂,可抑制 VEGFR2、c-Met、Kit、Axl 和 Flt4(IC50:0.035、1.3、4.6、7 和 6 nM)。
T11719 JMV 2959 hydrochloride (925238-89-7 free base)

JMV 2959 hydrochloride

GHSR GPCR/G Protein
JMV 2959 hydrochloride (925238-89-7 free base) 是一种生长激素促分泌素受体 1a 型 (GHS-R1a) 拮抗剂,在 LLC-PK1 细胞中的 IC50 为 32±3 nM。
T8402 Regorafenib Hydrochloride

瑞戈非尼盐酸盐,BAY73-4506 hydrochloride

c-RET; PDGFR; VEGFR; Autophagy; Raf Angiogenesis; Apoptosis; Autophagy; MAPK; Tyrosine Kinase/Adaptors
Regorafenib Hydrochloride 是一种新型口服多激酶抑制剂,可抑制血管生成、基质和致癌受体酪氨酸激酶,具有强大的临床前抗肿瘤活性。它靶向作用于 VEGFR1/2/3、PDGFRβ、Kit、RET 和 Raf-1,IC50值分别为 13/4.2/46、22、7、1.5 和 2.5 nM。
T3050 ML-7 hydrochloride

ML-7盐酸盐,ML-7 HCl

PKC; Serine/threonin kinase; PKA; YAP; Myosin Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; Metabolism; Stem Cells; Tyrosine Kinase/Adaptors
ML-7 hydrochloride 是一种可渗透细胞的、可逆的、有效的、ATP 竞争性的肌球蛋白轻链激酶 (MLCK) 特异性抑制剂,IC50为300 nM。它还抑制平滑肌肌球蛋白轻链激酶、PKA 和 PKC。
T4690 Betrixaban hydrochloride(330942-05-7(free base))

PRT054021 hydrochloride,盐酸贝曲西班

Factor Xa Metabolism
Betrixaban hydrochloride(330942-05-7(free base)) 是一种有效的、选择性的、口服有效的 Xa 因子 (fXa) 抑制剂 (IC50: 1.5 nM)。
T11638 Ilorasertib hydrochloride

ABT-348 hydrochloride

Aurora Kinase Cell Cycle/Checkpoint; Chromatin/Epigenetic
Ilorasertib hydrochloride (ABT-348 hydrochloride) is an ATP-competitive multitargeted kinase inhibitor, which inhibits Aurora C, Aurora B, and Aurora A (IC50s: 1 nM, 7 nM, 120 nM). It also suppresses RET tyrosine kinase, PDGFRβ, and Flt1 (IC50s: 7 nM, 3 n
T12025 MFZ 10-7 hydrochloride

GluR Neuroscience
MFZ 10-7 hydrochloride is a highly potent and selective negative allosteric modulator of mGluR5 NAM
T34836 Theophylline, 7-(2-(diethylamino)ethyl)-6-thio-, hydrochloride

Theophylline, 7-(2-(diethylamino)ethyl)-6-thio-, hydrochloride is a bioactive chemical.
T63095 GNE 220 hydrochloride

GNE 220 (hydrochloride) 是一种有效的、选择性的 MAP4K4 抑制剂 (IC50: 7 nM)。
T34838 Theophylline, 7-(2-oxo-4-piperidinobutyl)-6-thio-, hydrochloride

Theophylline, 7-(2-oxo-4-piperidinobutyl)-6-thio-, hydrochloride is a bioactive chemical.
T61724 SB 258741 hydrochloride

SB 258741 hydrochloride is a potent antagonist of the 5-HT 7 receptor, designed specifically for studying schizophrenia [1].
T62102 Elimusertib hydrochloride

Elimusertib (BAY 1895344) hydrochloride 是一种有效的、选择性的、口服具有活力的 ATR 抑制剂 (IC50: 7 nM),表现出抗肿瘤作用。Elimusertib hydrochloride 能够用于研究实体瘤和淋巴瘤。
T39641 SHP2-IN-6 hydrochloride

SHP2-IN-6 hydrochloride

SHP2-IN-6 hydrochloride, derived from compound 7 of patent WO2017211303A1, is a highly potent inhibitor of SHP2 with an IC50 of 25.8 nM.
T63622 RF9 hydrochloride

RF9 hydrochloride 是有效的、选择性的神经肽 FF 受体 (Neuropeptide FF receptor) 拮抗剂,能够作用于 hNPFF1R (Ki: 58 nM) 和 hNPFF2R (Ki: 7 nM)。
T11548L HCV-IN-7 hydrochloride

Others Others
HCV-IN-7 hydrochloride is an orally active and potent pan-genotypic HCV NS5A inhibitor (IC50s: 3-47 pM). It shows a superior pan-genotypic profile and a good pharmacokinetic profile coupled with a favorable liver uptake.
T19243 CMP-5 hydrochloride

Others Others
CMP-5 hydrochloride is a potent and selective PRMT5 inhibitor, while displays no activity against PRMT1/4/7 enzymes. It selectively blocks S2Me-H4R3 by inhibiting PRMT5 methyltransferase activity on histone preparations.
T22091 Imiquimod hydrochloride

Imiquimod hydrochloride (R 837 hydrochloride)是一种免疫反应调节剂,是一种选择性的 toll 样受体 7 (TLR7) 激动剂。Imiquimod hydrochloride 在体内表现出抗病毒和抗肿瘤作用。Imiquimod hydrochloride 可用于外生殖器、肛周疣、癌症和 COVID-19 的研究。
T11443L GNE 220 Hydrochloride (1199590-75-4 free base)

GNE 220 Hydrochloride

Others Others
GNE 220 Hydrochloride is a potent and selective inhibitor of MAP4K4 (IC50: 7 nM).
T13157L TG 100801 Hydrochloride

VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
TG 100801 Hydrochloride is a prodrug to treat age-related macular degeneration. TG 100572 is a inhibitor of multi-targeted kinase(IC50s of 2, 7, 2, 16, 13, 5, 0.5, 6, 0.1, 0.4, 1, 0.2 for VEGFR1, VEGFR2, FGFR1, FGFR2, PDGFRβ, Fgr, Fyn, Hck, Lck, Lyn, Src,
T71764 YM 298198 Hydrochloride

YM 298198 Hydrochloride is a non-competitive antagonist with high affinity and selectivity for mGlu1 receptors (Ki = 19 nM). YM 298198 Hydrochloride is inactive at other mGlu receptor subtypes (mGlu2-7), ionotropic receptors and glutamate transporters (IC50 > 10 μM). It inhibits glutamate-induced IP production more potently than CPCCOEt (IC50 values are 16 nM and 6.3 μM respectively).
T36231 Rac-7-hydroxy Propranolol (hydrochloride)

rac-7-hydroxy Propranolol (hydrochloride) is a ring-hydroxylated isomer and metabolite of propranolol that is an antagonist at β-adrenergic receptors (0.95 potency relative to propranolol). It also demonstrates potent vasodilator activity (0.20 potency relative to propranolol; pA2 = 7.58).
T13156L TG 100572 Hydrochloride

VEGFR; FGFR; PDGFR; Src Angiogenesis; Tyrosine Kinase/Adaptors
TG 100572 Hydrochloride 是一种多靶点激酶抑制剂,能够抑制受体酪氨酸激酶和Src 激酶。
T68262 AEG40826

AEG40826 (HGS1029) is the hydrochloride salt of a small-molecule inhibitor of IAP (Inhibitor of Apoptosis Protein) family proteins with potential antineoplastic activity. IAP inhibitor HGS1029 selectively inhibits the biological activity of IAP proteins, which may restore apoptotic signaling pathways; this agent may work synergistically with cytotoxic drugs to overcome tumor cell resistance to apoptosis. IAPs are overexpressed by many cancer cell types, suppressing apoptosis by binding and inhib...
T70235 Cemadotin hydrochloride

Cemadotin hydrochloride is the salt from of Cemadotin (free base), also known as, LU103793, a mitosis inhibitor potentially for the treatment of solid tumours. Cemadotin is also a synthetic derivative of Dolastatin 15, an antiproliferative compound which was isolated from the mollusk Dolabella auricularia. Like Dolastatin 15, LU103793 is highly cytotoxic in vitro (IC50 = 0.1 nM). LU103793 inhibits microtubule polymerization in a concentration-dependent manner (IC50 = 7 microM). Treatment with ...
T35875 CCG258208 hydrochloride

GRKs-IN-1 hydrochloride, Compound 14as, has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50=130 nM) and GRK5 (IC50=7.1 μM).GRKs-IN-1 hydrochloride is a derivative 14as of paroxetine, shows a 100-fold improvement in cardiomyocyte contractility assays over paroxetine[1]. [1]. Waldschmidt HV, et al. Structure-Based Design of Highly Selective and Potent G Protein-Coupled Receptor Kinase 2Inhibitors Based on Paroxetine. J Med Chem. 2017 Apr 13;60(7):305...
T37114 SB 242084 dihydrochloride

SB 242084 hydrochloride is a 5-HT2C receptor antagonist(pKi=9.0) that displays 158- and 100-fold selectivity over 5-HT2A and 5-HT2B receptors respectively.IC50 value: 9.0(pKi) [1]Target: 5-HT2C antagonistin vitro: SB 242084 had over 100-fold selectivity over a range of other 5-HT, dopamine and adrenergic receptors. In studies of 5-HT-stimulated phosphatidylinositol hydrolysis using SH-SY5Y cells stably expressing the cloned human 5-HT2C receptor, SB 242084 acted as an antagonist with a pKb of 9....

化合物

A-7 hydrochloride
T22538
synonym:
Target: CaMK
W-7 hydrochloride
T20792
synonym: N-(6-氨基己基)-5-氯-1-萘磺胺盐酸盐,W-7 HCl,W 7 HCl,W7 HCl
Target: CaMK, Apoptosis, Myosin, PDE
Facinicline hydrochloride
T28531
synonym: RG3487
Target: AChR, 5-HT Receptor
CRA-026440 hydrochloride
T10883L
synonym: CRA-026440 hydrochloride(847460-34-8 Free base)
Target: HDAC
Demeclocycline hydrochloride
T1400
synonym: Detravis,Clortetrin,地美环素,盐酸地美环素,Demeclocycline HCl,Declomycin
Target: Antibiotic, ribosome, Antibacterial
Idarubicin hydrochloride
T6010
synonym: 盐酸伊达比星,伊达比星盐酸盐,Zavedos,Idarubicin HCl,4-demethoxydaunorubicin (NSC256439, 4-DMDR) HCl,Idamycin,4-Demethoxydaunorubicin hydrochloride
Target: Autophagy, Antibacterial, Topoisomerase, Antifungal
Irinotecan Hydrochloride
T0486L
synonym: 盐酸伊立替康,伊立替康盐酸盐,Camptothecin 11 hydrochloride,CPT-11 hydrochloride
Target: Topoisomerase, Autophagy
BPR1J-097 hydrochloride (1327167-19-0(free base))
T4261
synonym:
Target: FLT
Cabozantinib hydrochloride
T5164
synonym: Cabozantinib hydrochloride (849217-68-1(free base)),BMS-907351,XL184,盐酸卡博替尼
Target: c-Met/HGFR, TAM Receptor, ROR, VEGFR, FLT, c-Kit
JMV 2959 hydrochloride (925238-89-7 free base)
T11719
synonym: JMV 2959 hydrochloride
Target: GHSR
Regorafenib Hydrochloride
T8402
synonym: 瑞戈非尼盐酸盐,BAY73-4506 hydrochloride
Target: c-RET, PDGFR, VEGFR, Autophagy, Raf
ML-7 hydrochloride
T3050
synonym: ML-7盐酸盐,ML-7 HCl
Target: PKC, Serine/threonin kinase, PKA, YAP, Myosin
Betrixaban hydrochloride(330942-05-7(free base))
T4690
synonym: PRT054021 hydrochloride,盐酸贝曲西班
Target: Factor Xa
Ilorasertib hydrochloride
T11638
synonym: ABT-348 hydrochloride
Target: Aurora Kinase
MFZ 10-7 hydrochloride
T12025
synonym:
Target: GluR
Theophylline, 7-(2-(diethylamino)ethyl)-6-thio-, hydrochloride
T34836
synonym:
Target:
GNE 220 hydrochloride
T63095
synonym:
Target:
Theophylline, 7-(2-oxo-4-piperidinobutyl)-6-thio-, hydrochloride
T34838
synonym:
Target:
SB 258741 hydrochloride
T61724
synonym:
Target:
Elimusertib hydrochloride
T62102
synonym:
Target:
SHP2-IN-6 hydrochloride
T39641
synonym: SHP2-IN-6 hydrochloride
Target:
RF9 hydrochloride
T63622
synonym:
Target:
HCV-IN-7 hydrochloride
T11548L
synonym:
Target: Others
CMP-5 hydrochloride
T19243
synonym:
Target: Others
Imiquimod hydrochloride
T22091
synonym:
Target:
GNE 220 Hydrochloride (1199590-75-4 free base)
T11443L
synonym: GNE 220 Hydrochloride
Target: Others
TG 100801 Hydrochloride
T13157L
synonym:
Target: VEGFR
YM 298198 Hydrochloride
T71764
synonym:
Target:
rac-7-hydroxy Propranolol (hydrochloride)
T36231
synonym:
Target:
TG 100572 Hydrochloride
T13156L
synonym:
Target: VEGFR, FGFR, PDGFR, Src
AEG40826
T68262
synonym:
Target:
Cemadotin hydrochloride
T70235
synonym:
Target:
CCG258208 hydrochloride
T35875
synonym:
Target:
SB 242084 dihydrochloride
T37114
synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T1400 Demeclocycline hydrochloride

Detravis,Clortetrin,地美环素,盐酸地美环素,Demeclocycline HCl,Declomycin

Antibiotic; ribosome; Antibacterial Microbiology/Virology
Demeclocycline hydrochloride 是四环素类抗生素,可治疗粉刺,莱姆病和支气管炎。
T0486L Irinotecan Hydrochloride

盐酸伊立替康,伊立替康盐酸盐,Camptothecin 11 hydrochloride,CPT-11 hydrochloride

Topoisomerase; Autophagy Autophagy; DNA Damage/DNA Repair
Irinotecan Hydrochloride 是喜树碱半合成衍生物的盐酸盐,是一种拓扑异构酶 I 抑制剂,可研究结肠癌和直肠癌。

天然产物

Demeclocycline hydrochloride
T1400
synonym: Detravis,Clortetrin,地美环素,盐酸地美环素,Demeclocycline HCl,Declomycin
Target: Antibiotic, ribosome, Antibacterial
Irinotecan Hydrochloride
T0486L
synonym: 盐酸伊立替康,伊立替康盐酸盐,Camptothecin 11 hydrochloride,CPT-11 hydrochloride
Target: Topoisomerase, Autophagy
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