win

WIN site inhibitor 1 is a WIN site of chromatin-associated WD repeat-containing protein 5 (WDR5) inhibitor (Kd: 0.1 nM), with anti-cancer activity.

WIN 51,708 是一种神经激肽受体（NK1）拮抗剂。

WIN 54954 是一种可口服的抗病毒剂，抑制柯萨奇病毒，抑制病毒翻译或转录。WIN 54954 可用于研究小核糖核酸病毒感染。

WIN 55,212-2 Mesylate ((R)-(+)-WIN 55212) 是 cannabinoid receptor 激动剂，对人重组 CB1 受体(Ki:62.3 nM) 和 CB2 受体 (Ki:3.3 nM)。

WIN 68577 是一种天然化合物，可作为天然产物对照品，其 CAS 号为 151928-33-5。

WIN-64821 是一种天然化合物，可作为天然产物对照品，其 CAS 号为 150881-27-9。

Win-62005 is an inhibitor of cyclic AMP phosphodiesterase III (PDE III)(Kis: 25 and 26 nM for rat heart and canine aorta).

Win 58237 is an inhibitor of cyclic nucleotide phosphodiesterase (PDE) (Ki: 170 nM for PDE V), with vasorelaxant activity.

WIN site inhibitor 1 TFA is a WIN site of chromatin-associated WD repeat-containing protein 5 (WDR5) inhibitor (Kd: 0.1 nM).

WIN 5063-3 is the enantiomeric analog of the antimicrobial Thiamphenicol.

WIN 62,577 is a allosteric antagonist of mAChR.

WIN-68056 is a wetting agent in x-ray contrast compositions.

(±)-WIN 55,212-2 is a potent aminoalkylindole cannabinoid (CB) receptor agonist with a Ki value of 62.3 and 3.3 nM for human recombinant central cannabinoid (CB1) and peripheral cannabinoid (CB2) receptors, respectively. In contrast, the enantiomer (-)-WIN 55,212-3 acts a partial inverse agonist at CB1 (pIC50 = 5.5) and as a competitive neutral antagonist of CB2, reversing the inverse agonism evoked by SR 144528 (pEC50 = 5.3). (+)-WIN 55,212 (mesylate) is a mixture of the two enantiomers, (+)-WIN 55,212-2 and (-)-WIN 55,212-3.

WIN 66306 is a cyclic heptapeptide antagonist of neurokinin-1 (NK1) and NK2 receptors originally isolated from A. flavipes. It binds to NK1 and NK2 receptors and inhibits contractions induced by substance P in isolated guinea pig ileum in a concentration-dependent manner.

(-)-WIN 55,212-3 mesylate 是 WIN 55,212-2 mesylate的低活性对映异构体，无神经保护活性和减少肠道运输的作用。(-)-WIN 55,212-3 mesylate是一种大麻素受体激动剂， 可用于研究神经系统疾病。

Win 18446 是口服有效的睾丸特异性的ALDH1a2的抑制剂，IC50为 0.3 μM。Win 18446 抑制睾丸内视黄醇合成视黄酸，可逆的抑制多个物种的精子形成，。

Milrinone (Win 47203) 是一种 PDE3抑制剂，也是一种强心药、血管舒张药。

Hycanthone (Etrenol(mesylate)) 是 Lucanthone 的生物活性代谢产物，是一种抗血吸虫病药。它是一个噻吨酮类 DNA 嵌入剂，可抑制 RNA 合成以及 DNA 拓扑异构酶 I 和 II。它通过直接蛋白质结合来抑制核酸生物合成并抑制嘌呤内切核酸酶1，KD 为 10 nM。

Disoxaril (BRN 3626820, WIN 51711) is an anti-picornavirus agent that inhibits enterovirus replication by binding to a hydrophobic bag within the VP1 coat protein, thereby stabilizing virions and preventing their uncoating. When used in combination with A

Octenidine saccharin is a Dental Plaque Inhibitor

Oxarbazole is an antagonist of slow-reacting substance of anaphylaxis.

Cyclindole is an antipsychotic with a tricyclic structure that was never marketed. It displaces spiperone binding in vitro and elevates dopamine levels in the striatum, indicating it acts as a D₂ receptor antagonist.

Bitolterol is a new beta 2-adrenergic agonist and classified as a pro-drug.

Scytonemin is a biological pigment synthesized by many strains of cyanobacteria, including Calothrix sp., Lyngbya aestuarii, and others. Scytonemin is also a potent PKL1 inhibitor, which inhibits cell proliferation and arrests cell cycle through downregulating Plk1 activity in many cancel cells. Scytonemin was able to inhibit the proliferation of three myeloma cells in a dose-dependent manner, while U266 was the most sensitive one to scytonemin. Scytonemin , representing a novel Plk1 inhibitor, induced the inhibition of cell growth and cell cycle arrest in multiple myeloma cells by specifically decreasing Plk1 activity.