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抑制剂&激动剂
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TargetMol产品目录中 "radioligand"的结果
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TargetMol产品目录中 "

radioligand

"的结果
  • 抑制剂&激动剂
    60
    TargetMol | Inhibitors_Agonists
  • 多肽产品
    1
    TargetMol | Peptide_Products
  • 染料试剂
    1
    TargetMol | Dye_Reagents
  • 天然产物
    2
    TargetMol | Natural_Products
  • 同位素
    4
    TargetMol | Isotope_Products
  • FAUC-365
    T21667474432-66-1
    FAUC-365 是一种高度选择性的多巴胺D3受体拮抗剂,能够作用于 D3 受体(Ki:0.5 nM)、D4.4 受体(Ki:340 nM)、D2short 受体(Ki:2600 nM)和 D2Long 受体(Ki:3600 nM)。它可用于研究帕金森病、精神分裂症等疾病。
    • ¥ 461
    In stock
    规格
    数量
  • Sigma-2 Radioligand 2
    T2009742860554-31-8
    Sigma-2 Radioligand 2 (compound 4) 展现对σ2受体的高度亲和性(Ki=2.30 nM)以及显著的亚型选择性(Ki(σ1) Ki(σ2) > 1500)。
    • ¥ 12800
    10-14周
    规格
    数量
  • CB2 PET Radioligand 1
    T79577
    CB2PET Radioligand 1 (compound [18F]9) 作为hCB2靶向的PET Radioligand (Ki=7.7 nM),采用Cu介导的18F-氟化方法制备,并在小鼠神经炎症模型中展现了高脑摄取率。
    • 待询
    规格
    数量
  • Sigma-2 Radioligand 1
    T873922860554-32-9
    Sigma-2 Radioligand 1(compound 1)是一种针对Sigma-2的选择性配体。在生物分布性方面,该化合物在小鼠体内表现出色,且在大鼠中展现了良好的体内活性。经[18F]标记后的Sigma-2 Radioligand 1,在微型PET CT成像中能有效可视化肿瘤,显示出高肿瘤摄取率和优秀的肿瘤与背景比例。此外,研究表明,Sigma-2 Radioligand 1在U87MG胶质瘤异种移植模型中表现出高度的特异性结合。
    • 待询
    10-14周
    规格
    数量
  • Lusaperidone
    芦沙哌酮, R107474
    T11894214548-46-6In house
    Lusaperidone (R107474) 是一种有效的α2肾上腺素受体 (adrenergic receptor) 拮抗剂,是 α (2)-肾上腺素受体的潜在放射性配体,对 α2A和α2C 具有抑制作用, Ki 值分别为0.13和0.15 nM。
    • ¥ 1260
    In stock
    规格
    数量
    TargetMol | Inhibitor Sale
  • MRS 1754
    T16140264622-58-4In house
    MRS 1754 是A2B 腺苷受体选择性拮抗剂,对人和大鼠的 A1和 A3受体的亲和力非常低。
    • ¥ 373
    In stock
    规格
    数量
  • (S)-Desmethyl-NNC112
    (+)-Desmethyl-NNC112
    T29261221132-62-3In house
    (S)-Desmethyl-NNC112 ((+)-Desmethyl-NNC112) 是一种选择性 PET 放射性配体,可与 D-多巴胺受体结合。
    • ¥ 1980
    In stock
    规格
    数量
  • Arotinolol hydrochloride
    Arotinolol HCl, 阿罗洛尔盐酸盐
    T3014068377-91-3
    Arotinolol hydrochloride(Arotinolol HCl) 是一种非选择性的 α β-肾上腺素受体 (α β-adrenergic receptor ) 阻滞剂。Arotinolol hydrochloride 对放射性配体 125I-ICYP 与 5HT1B-羟色胺受体能结合有抑制作用。Arotinolol hydrochloride 是一种抗高血压和抗肥胖试剂,可改善大鼠主动脉僵硬,研究肥胖相关疾病。
    • ¥ 343
    In stock
    规格
    数量
  • 3-Aminopropylphosphonic Acid
    3-氨基丙烷磷酸
    T3820513138-33-5
    3-Aminopropylphosphonic Acid 是与膦酸的磷相连的氢被3-氨基丙基取代的膦酸,是 GABAB 受体(GABABR)的部分激动剂和基础催乳素分泌拮抗剂。
    • ¥ 148
    In stock
    规格
    数量
    TargetMol | Inhibitor Sale
  • Arotinolol
    阿罗洛尔
    T1037168377-92-4
    Arotinolol is a nonselective α β-adrenergic receptor blocker and a vasodilating β-blocker. Arotinolol also shows potency for inhibiting the binding of the radioligand 125I-ICYP to 5HT1B-serotonergic receptor sites. It is an antihypertensive agent.
    • ¥ 565
    5日内发货
    规格
    数量
  • MLi-2
    T161151627091-47-7
    MLi-2 是一种结构新颖、高效、选择性的 LRRK2 激酶抑制剂,具有中枢神经系统活性,IC50为 0.76 nM,有潜力用于帕金森氏病。
    • ¥ 529
    In stock
    规格
    数量
  • PCS1055 dihydrochloride
    T16443361979-40-0
    PCS1055 dihydrochloride is an effective, selective, and competitive muscarinic M4 receptor antagonist (IC50: 18.1 nM and a Kd: 5.72 nM). PCS1055 dihydrochloride is also a potent AChE inhibitor (IC50 s: 22 nM and 120 nM for electric eel and human AChE, res
    • ¥ 10600
    6-8周
    规格
    数量
  • PK14105
    T16547107257-28-3
    PK14105 has been evaluated biologically as a potential radioligand for positron emission tomography (PET) studies targeting peripheral benzodiazepine binding sites (PBBS) receptors. When administered to rats with unilaterally lesioned striata, PK14105 was observed to quickly cross the blood-brain barrier, displaying significant radioactivity retention in the lesioned striatum, in contrast to the unlesioned striatum or cerebellar vermis. Additionally, PK14105 has the capability to inhibit receptor ligands, calcium channel ligands, and co-transporters in all salivary glands.
    • ¥ 1090
    5日内发货
    规格
    数量
  • SB 224289
    SB-224289, SB224289
    T19690180083-23-2
    SB 224289 is a selective antagonist of 5-HT1B receptor with pKi of 8.2. It is a centrally active following oral administration in vivo. SB 224289 displays 60-fold selectivity over 5-HT1D, 5-HT1A, 5-HT1E, 5-HT1F, 5-HT2A and 5-HT2C receptors in radioligand
    • ¥ 17200
    3-6月
    规格
    数量
  • SDM-8
    T2016112242777-37-1
    SDM-8, 作为一种 PET 放射剂,与 SV2A 结合力较高,具体的 Ki 值为 0.58 nM。此化合物主要应用于阿尔茨海默病的研究。
    • 待询
    10-14周
    规格
    数量
  • A-317920
    T26478360551-59-3
    A-317920 is an inverse agonist radioligand.
    • ¥ 10600
    6-8周
    规格
    数量
  • GSK-215083
    GSK215083
    T27455607742-80-3
    GSK-215083 is a PET radioligand for the 5-HT6 receptor. GSK 215083 is a quinoline based compounds and acts by antagonising the 5-HT6 receptor. GSK-215083 binds to receptors 5-hydroxytrypamine-6 (5HT6) in the striatum and 5-hydroxytryptamine-2A (5HT2A) in
    • ¥ 10600
    6-8周
    规格
    数量
  • GSK931145
    GSK 931145,GSK-931145
    T27494896117-64-9
    GSK931145 is a positron emission tomography (PET) radioligand, it is suitable for quantifying glycine transporter (GlyT1) availability in the living brain.
    • ¥ 10600
    6-8周
    规格
    数量
  • PD 140376
    PD-140376,PD140376
    T28335149027-97-4
    PD 140376 is a highly selective antagonist radioligand for the cholecystokinin(B)-gastrin receptor in guinea pig gastric mucosa & cerebral cortex in the peripheral and central nervous systems.
    • ¥ 23800
    10-14周
    规格
    数量
  • AH-9700 free base
    T29742184638-09-3
    AH-9700 free base 用于治疗急迫性尿失禁和尿毒症。在一项放射性配体结合研究中,AH-9700 free base 对 sigma 受体表现出较高的亲和力,对膀胱功能正常的实验动物的排尿反射(即膀胱容量增加作用)有明显的抑制作用。
    • ¥ 10600
    待询
    规格
    数量
  • Altanserin
    R-53200, R53200, R 53200
    T2991376330-71-7
    Altanserin can binds to the 5-HT2A receptor. Labeled with the isotope fluorine-18 it is used as a radioligand in positron emission tomography (PET) studies of the brain.
    • ¥ 447
    5日内发货
    规格
    数量
  • Altanserin tartrate
    R-53,200
    T29913L79449-96-0
    Altanserin tartrate is a compound that binds to the 5-HT2A receptor. Labeled with the isotope fluorine-18 it is used as a radioligand in positron emission tomography (PET) studies of the brain.
    • ¥ 10600
    6-8周
    规格
    数量
  • AZD-2184
    J2.698.897G,AZD2184
    T30253945400-24-8
    AZD-2184 is a radioligand for detecting beta-amyloid deposits.
    • ¥ 10600
    6-8周
    规格
    数量
  • AZD4694
    NAV-4694, NAV4694, NAV 4694, Flutafuranol, AZD-4694, AZD 4694
    T318281054629-49-0
    Flutafuranol, also known as AZD 4694 and NAV4694, is a bio-active chemical. AZD4694 shows high affinity for beta-amyloid fibrils in vitro (K(d) = 2.3 + - 0.3 nM). The fluorine-18 labeled AZD4694 may have potential for PET-visualization of cerebral beta-am
    • ¥ 9890
    5日内发货
    规格
    数量