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TargetMol产品目录中 "

dgat-1-in-1

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  • 抑制剂&激动剂
    6
    TargetMol | Inhibitors_Agonists
  • 天然产物
    1
    TargetMol | Natural_Products
  • 分子与细胞研究
    1
    TargetMol | Inhibitors_Agonists
  • DGAT1-IN-1
    T151091449779-49-0
    DGAT1-IN-1是 DGAT1的高效抑制剂,在 Hep3B 细胞过表达 DGAT1裂解物中,测得IC50低于10nM。
    • ¥ 448
    In stock
    规格
    数量
  • ABT-046
    ABT046
    T140851031336-60-3
    ABT-046 是一种具有口服活性、选择性和高效性的二酰基甘油酰基转移酶 1 (DGAT-1) 抑制剂,可用于研究代谢疾病。
    • ¥ 1280
    In stock
    规格
    数量
  • Phenylpyropene A
    T37690189564-20-3
    Phenylpyropene A is a fungal metabolite originally isolated from P. griseofulvum that has enzyme inhibitory and insecticidal activities.1,2,3 It inhibits acyl-coenzyme A:cholesterol acyltransferase (ACAT; IC50 = 0.8 μM).1 Phenylpyropene A inhibits diacylglycerol acyltransferase (DGAT) in rat liver microsomes (IC50 = 78.7 μM). It induces mortality in 100% of M. persicae when used at a concentration of 5 ppm.3 |1. Kwon, O.E., Rho, M.C., Song, H.Y., et al. Phenylpyropene A and B, new inhibitors of acyl-CoA: Cholesterol acyltransferase produced by Penicillium griseofulvum F1959. J. Antibiot. (Tokyo) 55(11), 1004-1008 (2002).|2. Lee, S.W., Rho, M.C., Choi, J.H., et al. Inhibition of diacylglycerol acyltransferase by phenylpyropenes produced by Penicillium griseofulvum F1959. J. Microbiol. Biotechnol. 18(11), 1785-1788 (2008).|3. Horikoshi, R., Goto, K., Mitomi, M., et al. Identification of pyripyropene A as a promising insecticidal compound in a microbial metabolite screening. J. Antibiot. (Tokyo) 70(3), 272-276 (2017).
    • ¥ 3029
    待询
    规格
    数量
  • T863
    DGAT-3, DGAT-1 inhibitor
    T4681701232-20-4
    T863 (DGAT-3) 是口服有效的二酰基甘油酰基转移酶1 选择性抑制剂。T863结合DGAT1的酰基辅酶A 结合位点,抑制三酰甘油在细胞内的合成。
    • ¥ 322
    In stock
    规格
    数量
  • DGAT1-IN-3
    T62220939375-07-2
    DGAT1-IN-3 是一种选择性的、有效的,口服具有活力的 DGAT-1 抑制剂,能够抑制人类 DGAT-1 (IC50: 38 nM) 和大鼠 DGAT-1 (IC50: 120 nM)。DGAT1-IN-3 能够用于肥胖、血脂异常和代谢综合征的研究。
    • ¥ 2990
    5日内发货
    规格
    数量
  • ALN29882
    T7188624529-88-2
    ALN29882 is a glycerolipid, that is located at the plasma membrane. It is made up of two fatty acid chains that are covalently attached to a single glycerol molecule with the help of an ester linkage. 18:1 DG has been used as a diacyl-glycerol source in diacylglycerol O-acyltransferase 1 (DGAT1) assay. It has also been used as substrate to assess compounds as potential inhibitors of DGAT-1 in DGAT-1 enzyme assay. It is suitable to use in lipid-protein overlay screen assay with the recombinant protein His-AtROP6.
    • 待估
    35日内发货
    规格
    数量