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Targets Recommended: Epigenetic Reader Domain

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Cat. No. Product Name Target Signaling Pathways
T17249 VZ185

Epigenetic Reader Domain Chromatin/Epigenetic
VZ185 is an effective and selective dual BRD7/9 PROTAC degrader (DC50s: 4.5 and 1.8 nM, respectively).
T41201 cis-VZ 185

cis-VZ 185 is a negative control for VZ 185.
T17697 BRD7-IN-1

Epigenetic Reader Domain Chromatin/Epigenetic
BRD7-IN-1 是一种修饰的 BI7273 衍生物 (BRD7/9 抑制剂)。BRD7-IN-1 通过与 VHL 配体连接形成 PROTAC VZ185VZ185 抑制 BRD7/9 的 DC50分别是 4.5 nM 和1.8 nM。
T17696 BRD7-IN-1 free base

Others Others
BRD7-IN-1 free base, a modified derivative of BI7273 (BRD7/9 inhibitor), interacts with a VHL ligand through a linker, constituting the PROTAC VZ185 (targeting BRD7/9 with DC50 values of 4.5 and 1.8 nM, respectively)[1].

化合物

VZ185
Cat.No: T17249
Synonym:
Target: Epigenetic Reader Domain
cis-VZ 185
Cat.No: T41201
Synonym:
Target:
BRD7-IN-1
Cat.No: T17697
Synonym:
Target: Epigenetic Reader Domain
BRD7-IN-1 free base
Cat.No: T17696
Synonym:
Target: Others
TargetMol Loading
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