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Search Results for " isoproterenol "

19

抑制剂 & 化合物

1

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T21411	Isoproterenol Norisodrine,Isoprenaline,Novodrin,Isuprel,Medihaler-Iso	Endogenous Metabolite; Adrenergic Receptor	GPCR/G Protein; Metabolism; Neuroscience
	Isoproterenol (Norisodrine) 是一种非选择性且具有口服活性的 β-肾上腺素受体激动剂。Isoproterenol 是有效的外周血管扩张剂和支气管扩张剂。Isoproterenol 可用于研究心动过缓和支气管哮喘，用于治疗心脏传导阻滞、心动过缓。
T25546	Isoproterenol tartrate, (-)- L-Isoproterenol D-bitartrate,Isoproterenol D-bitartrate, L-,Isolevin
	Isoproterenol tartrate, (-)- is a beta-Adrenoceptor agonist agent that increases cytosolic cAMP.
T29262	(S)-Isoproterenol bitartrate EINECS 238-683-4,d-Isoproterenol bitartrate,L-(+)-Isoproterenol bitartrate,d-N-Isopropylnorepinephrine bitartrate
	(S)-Isoproterenol bitartrate is a bioactive chemical.
T20122	Isoproterenol sulfate anhydrous Norisodrine,Novodrine,Novodrin,dl-Isoproterenol sulfate,Isoprenaline sulphate,Aleudrin
	Isoproterenol sulfate anhydrous is a useful alkaloid. It is used for biological research.
T21411L	Isoproterenol bitartrate
	Isoproterenol bitartrate is a beta-sympathomimetic and an isopropyl analog of Epinephrine, which acts on the heart, bronchi, skeletal muscle, and alimentary tract. It is used mainly as a bronchodilator and heart stimulant.
T69598	Isoproterenol-d7 HCl
	Isoproterenol-d7 is intended for use as an internal standard for the quantification of isoproterenol by GC- or LC-MS. Isoproterenol is an agonist of β1- and β2-adrenergic receptors (β1- and β2-ARs; Kis = 224 and 458 nM, respectively). It is selective for β1- and β2-ARs over β3-ARs (Ki = 1,570 nM). Isoproterenol inhibits contractions in isolated field-stimulated rat vas deferens (EC50 = 45.6 nM). In vivo, isoproterenol (0.33 mg/kg) decreases blood pressure and increases water intake in nephrectom...
T1056	Isoprenaline hydrochloride NCI-c55630,Isoproterenol hydrochloride,Isoprenaline HCl,盐酸异丙肾上腺素	PI3K; Endogenous Metabolite; Adrenergic Receptor; PDE	GPCR/G Protein; Metabolism; Neuroscience; PI3K/Akt/mTOR signaling
	Isoprenaline hydrochloride (NCI-c55630) 是非选择性的β-肾上腺素能受体激动剂，有支气管扩张剂，外周血管扩张剂和心脏刺激活性。
T23312	SB 204741	5-HT Receptor	GPCR/G Protein; Neuroscience
	SB 204741 是一种选择性的5-HT2B 拮抗剂，具有高亲和性，pKi 值为7.1。
T69040	Dichloroisoproterenol
	Dichloroisoproterenol is also known as Dichloroisoprenaline (DCI), was the first beta blocker ever to be developed. It is non-selective for the β1-adrenergic and β2-adrenergic receptors. DCI has low potency and acts as a partial agonist/antagonist at these receptors. Dichloroisoprenaline is a racemic mixture of enantiomers.
T31435	Dichloroisoproterenol hydrochloride DCI hydrochloride,Dichloroisoprenaline hydrochloride,Dichloroisoproterenol HCl
	Dichloroisoproterenol hydrochloride is a biochemical. It may be used for cardiac arrhythmia.
T26822	Bisaramil hydrochloride RGH-2957,NK 1556,NK1556,Bisaramil,NK-1556,RGH 2957	Potassium Channel; Adrenergic Receptor	GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
	Bisaramil hydrochloride (Bisaramil) 是一种新型二氮双环壬烷抗心律失常化合物，抑制自由基生成。Bisaramil hydrochloride 可阻断钠电流，抑制异丙肾上腺素在 K（+）去极化肌上诱导的缓慢 Ca（2+）动作电位。
T34329	Rimiterol
	Rimiterol, a beta 2 stimulant, therefore affects the cardiovascular system less than isoproterenol.
T70854	Protokylol hydrochloride
	Protokylol hydrochloride is the salt form of Protokylol (free base) (Asmetil, Caytine, Palison, Ventaire), a β-adrenergic receptor agonist used as a bronchodilator in Europe and the United States. It is methylenedioxyphenyl-isoproterenol.
T69126	Clofeverine (free base)
	Clofeverine (free base) is a highly selective relaxant for gastrointestinal smooth muscles with a beta-receptor stimulative nature. On isolated ileum, the inhibitory effect of clofeverine for spontaneous motility was comparable to that of isoproterenol and 100 times higher than that of papaverine.
T69324	Clofeverine hydrochloride
	Clofeverine hydrochloride is the salt form of Clofeverine (free base), a highly selective relaxant for gastrointestinal smooth muscles with a beta-receptor stimulative nature. On isolated ileum, the inhibitory effect of clofeverine for spontaneous motility was comparable to that of isoproterenol and 100 times higher than that of papaverine.
T37896	AZ 1729
	FFA2 allosteric agonist. Inhibits forskolin-induced cAMP increase and stimulates 35SGTPγS binding in biochemical assays (pEC50 values are 6.9 and 7.23, respectively). Binds at allosteric binding site. In functional assays, displays positive allosteric modulation of FFA-induced Gi signaling and negative allosteric modulation of FFA-induced Gq/G11 signaling. Inhibits lipolytic effect of isoproterenol (pEC50 = 5.03) and induces migration of human neutrophils in vitro. Bolognini et al (2016) A novel...
T71141	Fenspiride-d5
	Fenspiride-d5 is intended for use as an internal standard for the quantification of fenspiride by GC- or LC-MS. Fenspiride is an antagonist of histamine H1 receptors and a non-steroidal anti-inflammatory drug (NSAID). It inhibits histamine-induced contraction of isolated guinea pig trachea but not histamine-induced inotropy of isolated guinea pig heart. It also inhibits phosphodiesterase 4 (PDE4), PDE5, and PDE3 (IC50s = 69, ~158, and 363 µM, respectively, in isolated human bronchi derived from ...
T37475	Cyclic ADP-Ribose (ammonium salt) cADP-Ribose,cADPR,Cyclic ADP-Ribose (ammonium salt)
	Cyclic ADP-ribose (cADP-ribose) is an endogenous metabolite of NAD+ that mobilizes the release of stored Ca2+ in the endoplasmic reticulum via ryanodine receptors in various cell types.[1],[2],[3],[4],[5] This second messenger is generated via the cADP-ribose synthases CD38 and CD157.[6],[5],[7] cADP-Ribose may also trigger the cell surface Ca2+ influx channel TRPM2 in a temperature-dependent manner.[8] In vitro, cADP-ribose modulates Ca2+ signaling in rat and mouse cardiomyocytes treated with i...
T36679	Rp-cAMPS sodium salt
	Rp-cAMPS sodium salt, a cAMP analog, is a potent, competitive cAMP-induced activation of cAMP-dependent PKA I and II (Kis of 12.5 μM and 4.5 μM, respectively) antagonist. Rp-cAMPS sodium salt is resistant to hydrolysis by phosphodiesterases[1][2][3][4][5][6]. A membrane-permeable competitive cAMP antagonist (Rp-cAMPS) that blocks PKA activation by binding to the regulatory subunits without dissociating the kinase holoenzyme also inhibits synaptic plasticity but has no effect on normal synaptic t...

化合物

Isoproterenol

Cat.No: T21411

Synonym: Norisodrine,Isoprenaline,Novodrin,Isuprel,Medihaler-Iso

Target: Endogenous Metabolite, Adrenergic Receptor

Isoproterenol tartrate, (-)-

Cat.No: T25546

Synonym: L-Isoproterenol D-bitartrate,Isoproterenol D-bitartrate, L-,Isolevin

(S)-Isoproterenol bitartrate

Cat.No: T29262

Synonym: EINECS 238-683-4,d-Isoproterenol bitartrate,L-(+)-Isoproterenol bitartrate,d-N-Isopropylnorepinephrine bitartrate

Isoproterenol sulfate anhydrous

Cat.No: T20122

Synonym: Norisodrine,Novodrine,Novodrin,dl-Isoproterenol sulfate,Isoprenaline sulphate,Aleudrin

Isoproterenol bitartrate

Cat.No: T21411L

Isoproterenol-d7 HCl

Cat.No: T69598

Isoprenaline hydrochloride

Cat.No: T1056

Synonym: NCI-c55630,Isoproterenol hydrochloride,Isoprenaline HCl,盐酸异丙肾上腺素

Target: PI3K, Endogenous Metabolite, Adrenergic Receptor, PDE

Cat.No: T23312

Target: 5-HT Receptor

Dichloroisoproterenol

Cat.No: T69040

Dichloroisoproterenol hydrochloride

Cat.No: T31435

Synonym: DCI hydrochloride,Dichloroisoprenaline hydrochloride,Dichloroisoproterenol HCl

Bisaramil hydrochloride

Cat.No: T26822

Synonym: RGH-2957,NK 1556,NK1556,Bisaramil,NK-1556,RGH 2957

Target: Potassium Channel, Adrenergic Receptor

Cat.No: T34329

Protokylol hydrochloride

Cat.No: T70854

Clofeverine (free base)

Cat.No: T69126

Clofeverine hydrochloride

Cat.No: T69324

Cat.No: T37896

Cat.No: T71141

Cyclic ADP-Ribose (ammonium salt)

Cat.No: T37475

Synonym: cADP-Ribose,cADPR,Cyclic ADP-Ribose (ammonium salt)

Rp-cAMPS sodium salt

Cat.No: T36679

Cat. No.	Product Name	Target	Signaling Pathways
T3753	Sinapinic Acid Sinapic acid,芥子酸,Synapoic acid	Apoptosis; RAAS; Reactive Oxygen Species; HDAC	Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; Endocrinology/Hormones; Immunology/Inflammation; Metabolism; NF-κB
	Sinapinic Acid (Synapoic acid) 是从 Hydnophytum formicarumJack. 根中分离到的酚类，是HDAC 抑制剂，对ACE-I 的活性也有抑制作用。它有抗肿瘤活性，诱导肿瘤细胞凋亡，具有抗氧化、抗糖尿病的作用。

天然产物

Cat.No: T3753

Synonym: Sinapic acid,芥子酸,Synapoic acid

Target: Apoptosis, RAAS, Reactive Oxygen Species, HDAC

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