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Search Results for "Ac-FLTD-CMK"

1

抑制剂 & 化合物

50

化合物库

1

TargetMol 试剂盒

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Cat. No. Product Name
DC1230 特权片段注释化合物库-Beta amyloid A4 protein

4617 compounds
L6300 药食同源库

1088 compounds
1088个药食同源化合物的独特集合,可用于高通量筛选和高内涵筛选;
L1610 FDA 上市激酶抑制剂库

280 compounds
TargetMol FDA上市激酶库包含280个具有明确激酶抑制活性的上市药物
L3400 临床期小分子药物库

3142 compounds
3142个临床期化合物集合,可用于高通量筛选和高内涵筛选;
L1600 激酶抑制剂库

2230 compounds
2230种激酶抑制剂的独特集合,用于特定靶向激酶,可用于高通量筛选和高内涵筛选;
L9840 抗阿尔茨海默症化合物库

1040 compounds
1040 种阿尔茨海默症相关的化合物集合,可用于高通量和高内涵筛选;
L8100 细胞周期化合物库

695 compounds
695种细胞周期相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
L2610 神经递质受体化合物库

1513 compounds
1513种与神经递质受体相关的化合物,用于高通量、高内涵筛选;
DC1140 特权片段注释化合物库-Ligand-gated

9028 compounds
DC1180 特权片段注释化合物库-Lyases

19530 compounds
DC1150 特权片段注释化合物库-GPCR Family B

9320 compounds
DC1170 特权片段注释化合物库-Oxidoreductases

8812 compounds
DC1190 特权片段注释化合物库-Sigma Opioid receptors

8724 compounds
DC1040 特权片段注释化合物库-Transferases

23001 compounds
DC1030 特权片段注释化合物库-Epigenetics

9196 compounds
DC1100 特权片段注释化合物库-GPCR Frizzled family

3434 compounds
DC1200 特权片段注释化合物库-Isomerases

1206 compounds
DC1050 特权片段注释化合物库-Voltage-gated

17952 compounds
DC1110 特权片段注释化合物库-Proteases

22863 compounds
DC1010 特权片段注释化合物库-GPCR Family A

24763 compounds
DC1000 特权片段注释化合物库

190000 compounds
The database contains 190k small molecules divided into 23 sub libraries each focused at a specific target. According to the recent studies, molecules acting on a particular target or class of targets usually have characteristic moieties (PF) containing key binding points responsible for activity, e.g. hinge-binding fragments. We used this principle for the statistical analysis of the reported active molecules and corresponding targets for the annotation of pre-filtered ChemDiv in house colle...
DC1130 特权片段注释化合物库-Phosphodiesterases

13154 compounds
DC1060 特权片段注释化合物库-Kinases

18350 compounds
DC1220 特权片段注释化合物库-Aminoacyltransferases

3008 compounds
DC1210 特权片段注释化合物库-Phosphatases

15354 compounds
DC1160 特权片段注释化合物库-Toll-like and Il-1 receptors

3536 compounds
DC1090 特权片段注释化合物库-Ligases

11828 compounds
DQ3000 Factor XIa化合物库

6500 compounds
DC1080 特权片段注释化合物库-GPCR Taste family

2675 compounds
DC1120 特权片段注释化合物库-Thrombopoietin receptors

4908 compounds
DC1070 特权片段注释化合物库-GPCR Family C

5071 compounds
DC1020 特权片段注释化合物库-Spiro Library

20563 compounds
L2620 神经退行性疾病化合物库

1622 compounds
1622种与神经退行性疾病相关的化合物,可用于高通量和高内涵筛选;
L6610 抗感染天然产物库

1070 compounds
1070个抗感染相关的天然产物集合,是药物开发、药理研究的有效工具;
L7300 钾通道分子库

160 compounds
160种钾通道相关化合物的独特集合,可用于高通量筛选和高内涵筛选;
L3500 组蛋白修饰化合物库

362 compounds
362个组蛋白修饰相关的小分子化合物的特有集合,用于高通量、高内涵筛选;
L4710 非甾体类抗炎化合物库

530 compounds
530种非甾体类的抗炎相关化合物,可用于高通量和高内涵筛选;
L3600 细胞因子抑制剂库

613 compounds
613个与细胞因子紧密相关的化合物集合,是高通量、高内涵筛选的良好载体;
L6730 抗病毒中药单体化合物库

270 compounds
270种具有抗病毒活性的中药单体集合,是药物开发、药理研究的有效工具;
L1110 微管靶向化合物库

80 compounds
80种靶向微管的分子集合,用于高通量筛选和高内涵筛选;
L5300 线粒体靶向库

447 compounds
447种具有潜在或确定线粒体靶向活性的化合物,以促进针对线粒体的药物研究;
L9830 抗帕金森病化合物库

908 compounds
908种帕金森病相关的化合物集合,可用于高通量和高内涵筛选;
L1310 细胞骨架化合物库

590 compounds
590种细胞骨架相关的化合物,可以用于高通量和高内涵筛选;
L4020 NO PAINS 化合物库

9555 compounds
TargetMol NO PAINS 化合物库包含 9555 个剔除了PAINS的小分子活性化合物,可用于新药研发,信号通路研究,老药新用等研究。
L2170 肿瘤免疫治疗小分子化合物库

454 compounds
454种靶向肿瘤免疫治疗靶点的小分子,可用于高通量和高内涵筛选,是研究肿瘤免疫治疗的有力工具;
CL0094 FLT3 inhibitor kit

CL0056 CDK inhibitor kit

CL0122 ACE inhibitor kit

CL0148 LPL Receptor antagonist/agonist kit

L8710 铜死亡化合物库

411 compounds
TargetMol 铜死亡化合物库集合了 411 种与铜死亡相关的化合物,可以用于铜死亡机制及相关疾病研究

化合物库

特权片段注释化合物库-Beta amyloid A4 protein
DC1230
Compounds: 4617
药食同源库
L6300
Compounds: 1088
FDA 上市激酶抑制剂库
L1610
Compounds: 280
临床期小分子药物库
L3400
Compounds: 3142
激酶抑制剂库
L1600
Compounds: 2230
抗阿尔茨海默症化合物库
L9840
Compounds: 1040
细胞周期化合物库
L8100
Compounds: 695
神经递质受体化合物库
L2610
Compounds: 1513
特权片段注释化合物库-Ligand-gated
DC1140
Compounds: 9028
特权片段注释化合物库-Lyases
DC1180
Compounds: 19530
特权片段注释化合物库-GPCR Family B
DC1150
Compounds: 9320
特权片段注释化合物库-Oxidoreductases
DC1170
Compounds: 8812
特权片段注释化合物库-Sigma Opioid receptors
DC1190
Compounds: 8724
特权片段注释化合物库-Transferases
DC1040
Compounds: 23001
特权片段注释化合物库-Epigenetics
DC1030
Compounds: 9196
特权片段注释化合物库-GPCR Frizzled family
DC1100
Compounds: 3434
特权片段注释化合物库-Isomerases
DC1200
Compounds: 1206
特权片段注释化合物库-Voltage-gated
DC1050
Compounds: 17952
特权片段注释化合物库-Proteases
DC1110
Compounds: 22863
特权片段注释化合物库-GPCR Family A
DC1010
Compounds: 24763
特权片段注释化合物库
DC1000
Compounds: 190000
特权片段注释化合物库-Phosphodiesterases
DC1130
Compounds: 13154
特权片段注释化合物库-Kinases
DC1060
Compounds: 18350
特权片段注释化合物库-Aminoacyltransferases
DC1220
Compounds: 3008
特权片段注释化合物库-Phosphatases
DC1210
Compounds: 15354
特权片段注释化合物库-Toll-like and Il-1 receptors
DC1160
Compounds: 3536
特权片段注释化合物库-Ligases
DC1090
Compounds: 11828
Factor XIa化合物库
DQ3000
Compounds: 6500
特权片段注释化合物库-GPCR Taste family
DC1080
Compounds: 2675
特权片段注释化合物库-Thrombopoietin receptors
DC1120
Compounds: 4908
特权片段注释化合物库-GPCR Family C
DC1070
Compounds: 5071
特权片段注释化合物库-Spiro Library
DC1020
Compounds: 20563
神经退行性疾病化合物库
L2620
Compounds: 1622
抗感染天然产物库
L6610
Compounds: 1070
钾通道分子库
L7300
Compounds: 160
组蛋白修饰化合物库
L3500
Compounds: 362
非甾体类抗炎化合物库
L4710
Compounds: 530
细胞因子抑制剂库
L3600
Compounds: 613
抗病毒中药单体化合物库
L6730
Compounds: 270
微管靶向化合物库
L1110
Compounds: 80
线粒体靶向库
L5300
Compounds: 447
抗帕金森病化合物库
L9830
Compounds: 908
细胞骨架化合物库
L1310
Compounds: 590
NO PAINS 化合物库
L4020
Compounds: 9555
肿瘤免疫治疗小分子化合物库
L2170
Compounds: 454
FLT3 inhibitor kit
CL0094
Compounds: 0
CDK inhibitor kit
CL0056
Compounds: 0
ACE inhibitor kit
CL0122
Compounds: 0
LPL Receptor antagonist/agonist kit
CL0148
Compounds: 0
铜死亡化合物库
L8710
Compounds: 411
Cat. No. Product Name Form Specificity Of Inhibition
C0005 Cell Counting Kit-8 (CCK-8)

Cell Counting Kit-8 (CCK-8)

Solution in bottle

TargetMol 试剂盒

Cell Counting Kit-8 (CCK-8)
C0005
Cat. No. Product Name Target Signaling Pathways
T36819 Ac-FLTD-CMK

Ac-FLTD-CMK, a gasdermin D (GSDMD)-derived inhibitor, is a specific inflammatory caspases inhibitor. Ac-FLTD-CMK is potent against caspases-1 (IC50 of 46.7 nM), caspases-4 (IC50 of 1.49 μM), caspases-5 (IC50 of 329 nM), and caspases-11 , but not the apoptotic caspases such as caspase-3[1]. Ac-FLTD-CMK, inhibits GSDMD cleavage by caspases-1, -4, -5, and -11 in vitro, suppresses pyroptosis downstream of both canonical and noncanonical inflammasomes, as well as reduces IL-1β release following activ...

化合物

Ac-FLTD-CMK
T36819
synonym:
Target: