(±)-verapamil

Verapamil hydrochloride (Verapamil HCl) 是一种钙通道阻滞剂，是一种可口服的 P 糖蛋白 (P-gp) 抑制剂，可抑制CYP3A4，用于高血压、心律不齐和心绞痛的研究。

Verapamil (CP-16533-1) 是一种非二氢吡啶类钙通道阻滞剂，一种 P-gp 抑制剂，也是一种 CYP3A4 抑制剂，具有口服活性。Verapamil 可以用于治疗高血压、心绞痛、心肌梗塞等。

R-Verapamil-d7 HCL 是 R-Verapamil HCL 的氘代化合物。R-Verapamil HCL 的 CAS 号为 1188265-55-5。

NSC-609249 hydrochloride, an impurity of Verapamil, is a calcium channel blocker with potent orally active properties. It also functions as a first-generation P-glycoprotein (P-gp) inhibitor.

S-Verapamil-d7 HCL 是 S-Verapamil HCL 的氘代化合物。S-Verapamil HCL 的 CAS 号为 1188265-55-5。

(+ -)-Verapamil hydrochloride-d7 是 (+ -)-Verapamil hydrochloride 的氘代化合物。(+ -)-Verapamil hydrochloride 的 CAS 号为 152-11-4。Verapamil hydrochloride 是一种钙通道阻滞剂，是一种可口服的 P 糖蛋白 (P-gp) 抑制剂，可抑制CYP3A4，用于高血压、心律不齐和心绞痛的研究。

(S)-Verapamil hydrochloride is an inhibitor of leukotriene C4 (LTC4) and calcein transport by MRP1,and leads to the death of potentially resistant tumor cells.

Verapamil-d7 Hydrochloride 是 Verapamil Hydrochloride 的氘代化合物。Verapamil Hydrochloride 的 CAS 号为 152-11-4。Verapamil hydrochloride 是一种钙通道阻滞剂，是一种可口服的 P 糖蛋白 (P-gp) 抑制剂，可抑制CYP3A4，用于高血压、心律不齐和心绞痛的研究。

(R)-Verapamil hydrochloride ((R)-(+)-Verapamil hydrochloride) is a inhibitor of P-Glycoprotein.

Gallopamil hydrochloride (Methoxyverapamil hydrochloride) 是苯烷基胺钙的拮抗剂。Gallopamil hydrochloride 可用于抗心律失常和血管扩张剂研究。

Gallopamil (Methoxyverapamil) 是一种苯烷基胺钙拮抗剂，以浓度依赖性方式抑制酸分泌 (IC50 = 10.9 μM)。Gallopamil 显示出抗心律失常和血管扩张剂的功效。

Norverapamil hydrochloride (D591 hydrochloride) 是 Verapamil 的 N-去甲基代谢物，是 L 型钙通道阻滞剂和 P-糖蛋白 (P-gp) 功能抑制剂。

Dexverapamil is the R-enantiomer of the calcium channel blocker verapamil. Dexverapamil competitively inhibits the multidrug resistance efflux pump P-glycoprotein (MDR-1), thereby potentially increasing the effectiveness of a wide range of antineoplastic drugs which are inactivated by MDR-1 mechanisms.

Arverapamil is a chiral metabolite of Verapamil.

Norverapamil-d7 HCl (D591-d7 HCl) 是一种 2H 标记的 Norverapamil HCl。Norverapamil 是一种钙通道阻滞剂和 P-糖蛋白 (P-gp)抑制剂,也是冠脉扩张剂，可用于研究心血管疾病和神经系统疾病。

Norverapamil is a blocker of L-type calcium channel and an inhibitor of P-glycoprotein (P-gp) function .

Norverapamil D7 is a deuterium labeled Norverapamil . Norverapamil is a blocker of L-type calcium channel and an inhibitor of P-glycoprotein (P-gp) function .

Homoveratronitrile 是Verapamil 的杂质。它也是制备肌肉松弛剂罂粟碱的中间体。

Pulegone ((+)-Pulegone) 是 Calamintha nepeta (L.) Savi 的精油的主要化学成分，也是禽类驱虫剂之一。它在禽类物种中驱避作用的分子靶点是伤害感受性 TRP 锚蛋 1。它刺激鸡感觉神经元中的 TRPM8 和 TRPA1 通道，并在高浓度下抑制前者但不抑制后者。

Jatrophane 5 demonstrates the most powerful inhibition of P-gp, higher than R(+)-verapamil and tariquidar in colorectal multi-drug resistant (MDR) cells (DLD1-TxR).

2,5,7,8,9,14-Hexaacetoxy-3-benzoyloxy-15-hydroxyjatropha-6(17),11E-diene (Jatrophane 2 ) exhibits significant antifeedant activity against a generalist plant-feeding insect, the cotton bollworm (Helicoverpa armigera). Jatrophane 2 also demonstrates the mo

LU 49888 is a photoaffinity analog of verapamil that has been used to identify specific binding sites for phenylalkylamines of calcium channels present in rabbit skeletal muscle microsomes.

Ronipamil is an analogue of verapamil that used as a calcium entry blocker.

Butoprozine 具有多重心脏电生理效应：它延长了动作电位时长，类似于 amiodarone 的效果；抑制了平台期，与 verapamil 的作用相似；并降低了振幅与最大去极化速率。