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Search Results for "PI-091"

1

抑制剂 & 化合物

47

化合物库

1

TargetMol 试剂盒

1

仪器耗材

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Cat. No. Product Name
L9400 PPI抑制剂库

260 compounds
260种已知活性的PPI相关的抑制剂,可用于高通量、高内涵筛选;
DP2680 Bcl2-Bax PPI抑制剂库

DO1800 螺旋模拟物PPI化合物库

L1610 FDA 上市激酶抑制剂库

280 compounds
TargetMol FDA上市激酶库包含280个具有明确激酶抑制活性的上市药物
L1600 激酶抑制剂库

2230 compounds
2230种激酶抑制剂的独特集合,用于特定靶向激酶,可用于高通量筛选和高内涵筛选;
L1300 PI3K/Akt/mTOR 化合物库

425 compounds
425种与PI3K/Akt/mTOR相关的生物活性小分子化合物的特有集合,用于PI3K/Akt/mTOR相关研究以及高通量、高内涵筛选;
L9830 抗帕金森病化合物库

908 compounds
908种帕金森病相关的化合物集合,可用于高通量和高内涵筛选;
DQ3000 Factor XIa化合物库

6500 compounds
DC1080 特权片段注释化合物库-GPCR Taste family

2675 compounds
DC1120 特权片段注释化合物库-Thrombopoietin receptors

4908 compounds
DC1230 特权片段注释化合物库-Beta amyloid A4 protein

4617 compounds
DC1070 特权片段注释化合物库-GPCR Family C

5071 compounds
DC1020 特权片段注释化合物库-Spiro Library

20563 compounds
DC1050 特权片段注释化合物库-Voltage-gated

17952 compounds
DC1110 特权片段注释化合物库-Proteases

22863 compounds
DC1010 特权片段注释化合物库-GPCR Family A

24763 compounds
DC1000 特权片段注释化合物库

190000 compounds
The database contains 190k small molecules divided into 23 sub libraries each focused at a specific target. According to the recent studies, molecules acting on a particular target or class of targets usually have characteristic moieties (PF) containing key binding points responsible for activity, e.g. hinge-binding fragments. We used this principle for the statistical analysis of the reported active molecules and corresponding targets for the annotation of pre-filtered ChemDiv in house colle...
DC1130 特权片段注释化合物库-Phosphodiesterases

13154 compounds
DC1060 特权片段注释化合物库-Kinases

18350 compounds
DC1220 特权片段注释化合物库-Aminoacyltransferases

3008 compounds
DC1210 特权片段注释化合物库-Phosphatases

15354 compounds
DC1160 特权片段注释化合物库-Toll-like and Il-1 receptors

3536 compounds
DC1090 特权片段注释化合物库-Ligases

11828 compounds
DC1140 特权片段注释化合物库-Ligand-gated

9028 compounds
DC1180 特权片段注释化合物库-Lyases

19530 compounds
DC1150 特权片段注释化合物库-GPCR Family B

9320 compounds
DC1170 特权片段注释化合物库-Oxidoreductases

8812 compounds
DC1190 特权片段注释化合物库-Sigma Opioid receptors

8724 compounds
DC1040 特权片段注释化合物库-Transferases

23001 compounds
DC1030 特权片段注释化合物库-Epigenetics

9196 compounds
DC1100 特权片段注释化合物库-GPCR Frizzled family

3434 compounds
DC1200 特权片段注释化合物库-Isomerases

1206 compounds
L2191 抗乳腺癌化合物库

1965 compounds
1965种与乳腺癌相关的化合物,可以用于抗乳腺癌药物研发和药理研究;
L2620 神经退行性疾病化合物库

1622 compounds
1622种与神经退行性疾病相关的化合物,可用于高通量和高内涵筛选;
DP9200 DGK抑制剂库

12000 compounds
包含12000种类药化合物,源自知名品牌Chemdiv,从160万小分子中百里挑一;
L6210 藏药化合物库

754 compounds
754种藏药来源的天然产物分子集合,可以用于高通量和高内涵筛选;
L1510 核受体化合物库

420 compounds
420个核受体作用化合物的独特集合,可用于高通量筛选和高内涵筛选;
L7800 高溶解性片段库

2731 compounds
2731种片段分子合集,数量适中,是FBDD方法新药筛选的有力工具。
L6130 萜类天然产物库

349 compounds
349种萜类天然产物的独特集合,可用于高通量筛选和高内涵筛选;
L2800 5-羟色胺分子库

275 compounds
275种生物活性小分子化合物,用于高通量、高内涵筛选;
L4100 TGF-β/Smad靶点化合物库

180 compounds
180个TGF-β/Smad靶点相关的小分子化合物的特有集合,用于高通量、高内涵筛选;
L2610 神经递质受体化合物库

1513 compounds
1513种与神经递质受体相关的化合物,用于高通量、高内涵筛选;
L2540 肠道微生物代谢化合物库

352 compounds
352种肠道微生物代谢物的集合,可以用于高通量和高内涵筛选;
L9840 抗阿尔茨海默症化合物库

1040 compounds
1040 种阿尔茨海默症相关的化合物集合,可用于高通量和高内涵筛选;
CL0106 HIF/HIF-PH inhibitor/activator kit

CL0083 Dehydrogenase inhibitor kit

CL0122 ACE inhibitor kit

化合物库

PPI抑制剂库
L9400
Compounds: 260
Bcl2-Bax PPI抑制剂库
DP2680
Compounds: 0
螺旋模拟物PPI化合物库
DO1800
Compounds: 0
FDA 上市激酶抑制剂库
L1610
Compounds: 280
激酶抑制剂库
L1600
Compounds: 2230
PI3K/Akt/mTOR 化合物库
L1300
Compounds: 425
抗帕金森病化合物库
L9830
Compounds: 908
Factor XIa化合物库
DQ3000
Compounds: 6500
特权片段注释化合物库-GPCR Taste family
DC1080
Compounds: 2675
特权片段注释化合物库-Thrombopoietin receptors
DC1120
Compounds: 4908
特权片段注释化合物库-Beta amyloid A4 protein
DC1230
Compounds: 4617
特权片段注释化合物库-GPCR Family C
DC1070
Compounds: 5071
特权片段注释化合物库-Spiro Library
DC1020
Compounds: 20563
特权片段注释化合物库-Voltage-gated
DC1050
Compounds: 17952
特权片段注释化合物库-Proteases
DC1110
Compounds: 22863
特权片段注释化合物库-GPCR Family A
DC1010
Compounds: 24763
特权片段注释化合物库
DC1000
Compounds: 190000
特权片段注释化合物库-Phosphodiesterases
DC1130
Compounds: 13154
特权片段注释化合物库-Kinases
DC1060
Compounds: 18350
特权片段注释化合物库-Aminoacyltransferases
DC1220
Compounds: 3008
特权片段注释化合物库-Phosphatases
DC1210
Compounds: 15354
特权片段注释化合物库-Toll-like and Il-1 receptors
DC1160
Compounds: 3536
特权片段注释化合物库-Ligases
DC1090
Compounds: 11828
特权片段注释化合物库-Ligand-gated
DC1140
Compounds: 9028
特权片段注释化合物库-Lyases
DC1180
Compounds: 19530
特权片段注释化合物库-GPCR Family B
DC1150
Compounds: 9320
特权片段注释化合物库-Oxidoreductases
DC1170
Compounds: 8812
特权片段注释化合物库-Sigma Opioid receptors
DC1190
Compounds: 8724
特权片段注释化合物库-Transferases
DC1040
Compounds: 23001
特权片段注释化合物库-Epigenetics
DC1030
Compounds: 9196
特权片段注释化合物库-GPCR Frizzled family
DC1100
Compounds: 3434
特权片段注释化合物库-Isomerases
DC1200
Compounds: 1206
抗乳腺癌化合物库
L2191
Compounds: 1965
神经退行性疾病化合物库
L2620
Compounds: 1622
DGK抑制剂库
DP9200
Compounds: 12000
藏药化合物库
L6210
Compounds: 754
核受体化合物库
L1510
Compounds: 420
高溶解性片段库
L7800
Compounds: 2731
萜类天然产物库
L6130
Compounds: 349
5-羟色胺分子库
L2800
Compounds: 275
TGF-β/Smad靶点化合物库
L4100
Compounds: 180
神经递质受体化合物库
L2610
Compounds: 1513
肠道微生物代谢化合物库
L2540
Compounds: 352
抗阿尔茨海默症化合物库
L9840
Compounds: 1040
HIF/HIF-PH inhibitor/activator kit
CL0106
Compounds: 0
Dehydrogenase inhibitor kit
CL0083
Compounds: 0
ACE inhibitor kit
CL0122
Compounds: 0
Cat. No. Product Name Form Specificity Of Inhibition
C0003 Phosphatase Inhibitor Cocktail II (100× DMSO)

磷酸酶抑制剂 Cocktail II

Solution (100× in DMSO) Alkaline phosphatases, Ser/Thr phosphatases, Acid and PP1 and PP2A

TargetMol 试剂盒

磷酸酶抑制剂 Cocktail II
C0003
Cat. No. Product Name
P-0.4-96U Agen 96孔 0.4mL圆孔微孔板,U型底

仪器耗材

Agen 96孔 0.4mL圆孔微孔板,U型底
P-0.4-96U
Cat. No. Product Name Target Signaling Pathways
T28412 PI-091

PI-091 inhibits platelet aggregation.

化合物

PI-091
T28412
synonym:
Target: