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Cat. No. Product Name Target Signaling Pathways
T39561 Orexin 2 Receptor Agonist 2

Orexin 2 Receptor Agonist 2 (ORA-2) is a specific agonist for the orexin 2 receptor, obtained from patent WO2017135306A1 (example 16).
T3177 Orexin 2 Receptor Agonist

OX2R

OX Receptor GPCR/G Protein; Neuroscience
Orexin 2 Receptor Agonist 是一种选择性有效的OX2R 激动剂, EC50为23 nM。
T39229 YNT-185

OX Receptor GPCR/G Protein; Neuroscience
YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R, respectively. Furthermore, YNT-185 effectively alleviates symptoms of narcolepsy-cataplexy in mouse models.
T39808 Firazorexton

Firazorexton is a potent orexin type 2 receptor (OX2R) agonist (patent WO2019027058A1, example 395).
TP1975L [Ala11,D-Leu15]-Orexin B acetate

[Ala11,D-Leu15]-Orexin B acetate (532932-99-3 Free base)

OX Receptor GPCR/G Protein; Neuroscience
[Ala11,D-Leu15]-Orexin B acetate 是一种特异性 orexin-2 受体 (OX2) 激动剂,EC50 为 0.13 nM,比 OX1 (52 nM) 特异性高 400 倍。
T75921 [Ala11,D-Leu15]-Orexin B(human) TFA

[Ala11,D-Leu15]-Orexin B(human) TFA 是一种有效的,选择性的orexin-2 receptor (OX2)的激动剂。[Ala11,D-Leu15]-Orexin B(human) TFA 对 OX2 (EC50=0.13 nM) 比对 OX1 (52 nM) 高出 400 倍的选择性。
T75925 Orexin B, rat, mouse TFA

Orexin B, rat, mouse (Rat orexin B) TFA 是一种内源性增食欲素受体 (Orexin receptor) 激动剂。Orexin B, rat, mouse TFA 结合并激活两个密切相关的孤儿 G 蛋白偶联受体 OX1-R 和 OX2-R。Orexin B, rat, mouse TFA 刺激食物摄入和能量消耗,并在睡眠-觉醒调节中发挥重要作用。
T37112 YNT-185 dihydrochloride

Potent and selective orexin OX2 receptor agonist (EC50 = 28 nM at human OX2 expressed in CHO cells). Displays approximately 100-fold selectivity for OX2 over OX1 (EC50 = 2.75 μM at human OX1 expressed in CHO cells). Depolarizes OX2-expressing histaminergic neurons in mouse brain slices. Increases wake time in wild type mice. Suppresses cataplexy-like symptoms in OX knockout mice. Nagahara et al (2015) Design and synthesis of non-peptide, selective orexin receptor 2 agonists. J.Med.Chem. 58 7931 ...

化合物

Orexin 2 Receptor Agonist 2
T39561
synonym:
Target:
Orexin 2 Receptor Agonist
T3177
synonym: OX2R
Target: OX Receptor
YNT-185
T39229
synonym:
Target: OX Receptor
Firazorexton
T39808
synonym:
Target:
[Ala11,D-Leu15]-Orexin B acetate
TP1975L
synonym: [Ala11,D-Leu15]-Orexin B acetate (532932-99-3 Free base)
Target: OX Receptor
[Ala11,D-Leu15]-Orexin B(human) TFA
T75921
synonym:
Target:
Orexin B, rat, mouse TFA
T75925
synonym:
Target:
YNT-185 dihydrochloride
T37112
synonym:
Target:
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