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Targets Recommended: Others

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Cat. No. Product Name Target Signaling Pathways
T23055 NAS181

NAS-181

Others Others
rat 5-HT1B receptor antagonist
T69958 Tofacitinib maleate

Tofacitinib, also known as tasocitinib, CP-690550, is a Janus kinase (JAK) inhibitor. Tofacitinib modulates the signaling pathway at the point of JAKs, preventing the phosphorylation and activation of STATs. JAK enzymes transmit cytokine signaling through pairing of JAKs (e.g., JAK1/JAK3, JAK1/JAK2, JAK1/TyK2, JAK2/JAK2). Tofacitinib inhibited the in vitro activities of JAK1/JAK2, JAK1/JAK3, and JAK2/JAK2 combinations with IC50 of 406, 56, and 1377 nM, respectively.

化合物

NAS181
T23055
synonym: NAS-181
Target: Others
Tofacitinib maleate
T69958
synonym:
Target:
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