DC1230
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特权片段注释化合物库-Beta amyloid A4 protein
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4617 compounds
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L6300
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药食同源库
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1088 compounds
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1088个药食同源化合物的独特集合,可用于高通量筛选和高内涵筛选;
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L7700
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神经再生化合物库
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529 compounds
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529种神经再生相关化合物的独特集合,可用于高通量筛选和高内涵筛选;
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L9840
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抗阿尔茨海默症化合物库
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1040 compounds
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1040 种阿尔茨海默症相关的化合物集合,可用于高通量和高内涵筛选;
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L6620
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抗寄生虫天然产物库
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233 compounds
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233个抗寄生虫相关的天然产物集合,是药物开发、药理研究的有效工具;
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L6210
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藏药化合物库
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754 compounds
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754种藏药来源的天然产物分子集合,可以用于高通量和高内涵筛选;
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L4020
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NO PAINS 化合物库
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9555 compounds
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TargetMol NO PAINS 化合物库包含 9555 个剔除了PAINS的小分子活性化合物,可用于新药研发,信号通路研究,老药新用等研究。
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DC1140
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特权片段注释化合物库-Ligand-gated
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9028 compounds
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DC1180
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特权片段注释化合物库-Lyases
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19530 compounds
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DC1150
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特权片段注释化合物库-GPCR Family B
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9320 compounds
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DC1170
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特权片段注释化合物库-Oxidoreductases
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8812 compounds
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DC1190
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特权片段注释化合物库-Sigma Opioid receptors
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8724 compounds
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DC1040
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特权片段注释化合物库-Transferases
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23001 compounds
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DC1030
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特权片段注释化合物库-Epigenetics
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9196 compounds
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DC1100
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特权片段注释化合物库-GPCR Frizzled family
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3434 compounds
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DC1200
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特权片段注释化合物库-Isomerases
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1206 compounds
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DC1050
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特权片段注释化合物库-Voltage-gated
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17952 compounds
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DC1110
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特权片段注释化合物库-Proteases
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22863 compounds
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DC1010
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特权片段注释化合物库-GPCR Family A
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24763 compounds
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|
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DC1000
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特权片段注释化合物库
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190000 compounds
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The database contains 190k small molecules divided into 23 sub libraries each focused at a specific target.
According to the recent studies, molecules acting on a particular target or class of targets usually have characteristic moieties (PF) containing key binding points responsible for activity, e.g. hinge-binding fragments. We used this principle for the statistical analysis of the reported active molecules and corresponding targets for the annotation of pre-filtered ChemDiv in house colle...
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DC1130
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特权片段注释化合物库-Phosphodiesterases
|
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13154 compounds
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|
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DC1060
|
特权片段注释化合物库-Kinases
|
|
18350 compounds
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|
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DC1220
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特权片段注释化合物库-Aminoacyltransferases
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3008 compounds
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DC1210
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特权片段注释化合物库-Phosphatases
|
|
15354 compounds
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DC1160
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特权片段注释化合物库-Toll-like and Il-1 receptors
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|
3536 compounds
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DC1090
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特权片段注释化合物库-Ligases
|
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11828 compounds
|
|
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DQ3000
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Factor XIa化合物库
|
|
6500 compounds
|
|
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DC1080
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特权片段注释化合物库-GPCR Taste family
|
|
2675 compounds
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|
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DC1120
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特权片段注释化合物库-Thrombopoietin receptors
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4908 compounds
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|
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DC1070
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特权片段注释化合物库-GPCR Family C
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5071 compounds
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|
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DC1020
|
特权片段注释化合物库-Spiro Library
|
|
20563 compounds
|
|
|
L6130
|
萜类天然产物库
|
|
349 compounds
|
|
349种萜类天然产物的独特集合,可用于高通量筛选和高内涵筛选;
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L9210
|
儿童药物库
|
|
1015 compounds
|
|
1015种儿童药物的独特集合,可用于高通量筛选和高内涵筛选
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L2620
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神经退行性疾病化合物库
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|
1622 compounds
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|
1622种与神经退行性疾病相关的化合物,可用于高通量和高内涵筛选;
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L6610
|
抗感染天然产物库
|
|
1070 compounds
|
|
1070个抗感染相关的天然产物集合,是药物开发、药理研究的有效工具;
|
L4100
|
TGF-β/Smad靶点化合物库
|
|
180 compounds
|
|
180个TGF-β/Smad靶点相关的小分子化合物的特有集合,用于高通量、高内涵筛选;
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L7300
|
钾通道分子库
|
|
160 compounds
|
|
160种钾通道相关化合物的独特集合,可用于高通量筛选和高内涵筛选;
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L3500
|
组蛋白修饰化合物库
|
|
362 compounds
|
|
362个组蛋白修饰相关的小分子化合物的特有集合,用于高通量、高内涵筛选;
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L1600
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激酶抑制剂库
|
|
2230 compounds
|
|
2230种激酶抑制剂的独特集合,用于特定靶向激酶,可用于高通量筛选和高内涵筛选;
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L4710
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非甾体类抗炎化合物库
|
|
530 compounds
|
|
530种非甾体类的抗炎相关化合物,可用于高通量和高内涵筛选;
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NY1000
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天然产物衍生物库
|
|
4000 compounds
|
|
22个天然产物骨架,4000个天然产物衍生物;
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L3600
|
细胞因子抑制剂库
|
|
613 compounds
|
|
613个与细胞因子紧密相关的化合物集合,是高通量、高内涵筛选的良好载体;
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L1610
|
FDA 上市激酶抑制剂库
|
|
280 compounds
|
|
TargetMol FDA上市激酶库包含280个具有明确激酶抑制活性的上市药物
|
L6730
|
抗病毒中药单体化合物库
|
|
270 compounds
|
|
270种具有抗病毒活性的中药单体集合,是药物开发、药理研究的有效工具;
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L1110
|
微管靶向化合物库
|
|
80 compounds
|
|
80种靶向微管的分子集合,用于高通量筛选和高内涵筛选;
|
L5300
|
线粒体靶向库
|
|
447 compounds
|
|
447种具有潜在或确定线粒体靶向活性的化合物,以促进针对线粒体的药物研究;
|
L9830
|
抗帕金森病化合物库
|
|
908 compounds
|
|
908种帕金森病相关的化合物集合,可用于高通量和高内涵筛选;
|
L1310
|
细胞骨架化合物库
|
|
590 compounds
|
|
590种细胞骨架相关的化合物,可以用于高通量和高内涵筛选;
|
L2610
|
神经递质受体化合物库
|
|
1513 compounds
|
|
1513种与神经递质受体相关的化合物,用于高通量、高内涵筛选;
|
L2170
|
肿瘤免疫治疗小分子化合物库
|
|
454 compounds
|
|
454种靶向肿瘤免疫治疗靶点的小分子,可用于高通量和高内涵筛选,是研究肿瘤免疫治疗的有力工具;
|
CL0122
|
ACE inhibitor kit
|
|
|
|
|
CL0135
|
ROCK inhibitor kit
|
|
|
|
|
L9860
|
抗抑郁症化合物库
|
|
1181 compounds
|
|
1181种与抑郁症相关的化合物,可以用于高通量和高内涵筛选
|
L8710
|
铜死亡化合物库
|
|
411 compounds
|
|
TargetMol 铜死亡化合物库集合了 411 种与铜死亡相关的化合物,可以用于铜死亡机制及相关疾病研究
|