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植物来源化合物库

植物来源化合物库

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产品编号 L4600 Selected Plant-Sourced Compound Library
  库化合物信息   Excel SDF

自然界创造了几乎无穷无尽的分子实体,为药物研发特别是新型药效团的发现创造了无限资源。在全球范围内,天然产物自古以来一直都是传统治疗的支柱。植物作为药物治疗疾病具有悠久的历史,植物来源的化合物具有更好的耐受性和可接受性。迄今为止,已对35,000-70,000种植物进行了药用筛选。半合成纯药物阿司匹林,是基于从白柳中分离出的天然产品水杨苷,由拜耳于1899年推出。此后陆续分离出了多种早期药物,如洋地黄毒苷、奎宁和毛果芸香碱等,其中一些仍在使用中,以及其他一些近期出现的植物衍生化合物,这些化合物经过开发并已作为药物销售,其中包括:来自短叶红豆杉的紫杉醇,用于肺部、卵巢癌和乳腺癌;青蒿素来自中国传统植物青蒿,用于对抗多药耐药性疟疾;水飞蓟素从水飞蓟种子中提取,用于治疗肝脏疾病。 TargetMol 植物来源化合物库精选3076 个植物来源天然产物的独特集合,具有良好的成药潜力,可用于天然产物来源的化合物筛选和新药研发。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
咨询化合物库
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产品描述

  • 3076个植物来源天然产物的独特集合;
  • 可用于高通量筛选和高内涵筛选;
  • 处于临床前研究或临床期实验阶段,是颇具研究潜力的天然产物集合;
  • 包含青蒿素,人参皂苷等热门的天然产物;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L4600)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

Endogenous Metabolite (441)
Apoptosis (346)
Antibacterial (228)
Autophagy (207)
NF-κB (180)
Antifungal (109)
Antioxidant (106)
COX (89)
Reactive Oxygen Species (88)
Parasite (74)
P450 (69)
Influenza Virus (61)
TNF (58)
AChR (56)
AChE (51)
Antibiotic (48)
NO Synthase (46)
HIV Protease (46)
p38 MAPK (45)
IL Receptor (45)
Anti-infection (45)
ERK (45)
Akt (42)
STAT (39)
Caspase (39)
Calcium Channel (38)
PPAR (38)
GABA Receptor (37)
Tyrosinase (37)
DNA/RNA Synthesis (36)
AMPK (33)
Nrf2 (31)
BCL (31)
MMP (29)
Virus Protease (29)
PI3K (27)
JNK (27)
Topoisomerase (26)
Lipoxygenase (26)
Microtubule Associated (25)
5-HT Receptor (25)
ROS (25)
PKC (24)
Ferroptosis (24)
TRP/TRPV Channel (23)
NOS (23)
Estrogen Receptor/ERR (23)
Dehydrogenase (22)
Antifection (22)
ATPase (21)
HSV (21)
Immunology/Inflammation related (21)
Estrogen/progestogen Receptor (21)
P-gp (21)
Potassium Channel (20)
PDE (20)
Adrenergic Receptor (20)
Prostaglandin Receptor (20)
PARP (19)
Beta Amyloid (19)
Sodium Channel (18)
Antiviral (18)
Glucosidase (17)
Mitophagy (17)
Wnt/beta-catenin (16)
Mitochondrial Metabolism (15)
EGFR (15)
MAO (14)
JAK (14)
HBV (14)
Interleukin (14)
HDAC (13)
TLR (13)
Adenosine Receptor (13)
SARS-CoV (12)
HIF/HIF Prolyl-Hydroxylase (12)
TGF-beta/Smad (12)
MAPK (11)
Dopamine Receptor (11)
VEGFR (11)
Drug Metabolite (11)
mTOR (11)
Sirtuin (10)
Reductase (10)
HCV Protease (10)
p53 (9)
Phosphatase (9)
Fatty Acid Synthase (9)
Androgen Receptor (9)
Opioid Receptor (9)
transporter (8)
CDK (8)
HSP (8)
Cannabinoid Receptor (8)
Phospholipase (8)
Monoamine Oxidase (8)
RAAS (8)
BACE (7)
NOD (7)
MEK (7)
PKA (7)
IκB/IKK (7)
Nucleoside Antimetabolite/Analog (7)
LDL (7)
UGT (7)
HIF (7)
Xanthine Oxidase (6)
Histamine Receptor (6)
Platelet aggregation (6)
Indoleamine 2,3-Dioxygenase (IDO) (6)
CaMK (6)
GSK-3 (6)
GluR (6)
Chloride channel (6)
NMDAR (5)
Epigenetic Reader Domain (5)
HMG-CoA Reductase (5)
Proteasome (5)
Aryl Hydrocarbon Receptor (5)
Reverse Transcriptase (5)
Free radical scavengers (5)
IAP (5)
iGluR (5)
Gamma-secretase (5)
HER (5)
PAFR (5)
Carbonic Anhydrase (5)
PTEN (4)
GPR (4)
Aromatase (4)
IGF-1R (4)
Transferase (4)
FGFR (4)
c-Met/HGFR (4)
Amylase (4)
GST (4)
ATP Citrate Lyase (4)
PGE Synthase (4)
Beta-Secretase (4)
NOD-like Receptor (NLR) (4)
FAK (4)
S6 Kinase (4)
CXCR (4)
FAAH (4)
E1/E2/E3 Enzyme (4)
cell cycle arrest (4)
MRP (4)
Hedgehog/Smoothened (4)
Integrin (3)
Serine/threonin kinase (3)
NADPH (3)
Syk (3)
FXR (3)
Acyltransferase (3)
Src (3)
Retinoid Receptor (3)
Telomerase (3)
Liver X Receptor (3)
Antifolate (3)
Proton pump (3)
CCR (3)
Serine Protease (3)
DNA Methyltransferase (3)
ROR (3)
Histone Acetyltransferase (3)
DNA (3)
Tyrosine Kinases (3)
PDK (3)
PDGFR (3)
Progesterone Receptor (3)
cAMP (3)
LTR (3)
Decarboxylase (2)
hCE (2)
Bcr-Abl (2)
PAI-1 (2)
Pyroptosis (2)
Casein Kinase (2)
Leukotriene Receptor (2)
Adiponectin receptor (2)
OCT (2)
NADPH-oxidase (2)
RANKL/RANK (2)
Glucocorticoid Receptor (2)
Aminopeptidase (2)
Aurora Kinase (2)
Trk receptor (2)
Monoamine Transporter (2)
Lipase (2)
SGLT (2)
Serotonin Transporter (2)
Glutathione Peroxidase (2)
Lipid (2)
DPP-4 (2)
Pim (2)
Bombesin Receptor (2)
PERK (2)
Smo (2)
DYRK (2)
Thrombin (2)
Cysteine Protease (2)
OAT (2)
IRAK (2)
Arginase (2)
P2X Receptor (2)
ABC (2)
AhR (2)
Hydroxylase (1)
PKM (1)
TAM Receptor (1)
Ras (1)
PD-1/PD-L1 (1)
NMU2R (1)
FLT (1)
Imidazoline Receptor (1)
PLK (1)
Adenosine deaminase (1)
ROS Kinase (1)
ATTECs (1)
Thyroid hormone receptor(THR) (1)
Oxytocin Receptor (1)
MyD88 (1)
Factor Xa (1)
gp120/CD4 (1)
Histone Demethylase (1)
RAR/RXR  (1)
aconitase (1)
IFNAR (1)
P2Y Receptor (1)
Amino Acids and Derivatives (1)
Dynamin (1)
c-Myc (1)
Histone Methyltransferase (1)
CYP19A1 (1)
DHFR (1)
stilbene oxidase (1)
NPC1L1 (1)
Transaminase (1)
Adenylyl cyclase (1)
Mdm2 (1)
advanced glycation end products (1)
Melatonin Receptor (1)
CaSR (1)
CRISPR/Cas9 (1)
Epoxide Hydrolase (1)
Carboxypeptidase (1)
ATM/ATR (1)
RSV (1)
ALK (1)
Survivin (1)
Glutathione reductase (1)
Norepinephrine (1)
Thrombopoietin Receptor (1)
PAD (1)
Glucokinase (1)
Stearoyl-CoA Desaturase (SCD) (1)
DNA gyrase (1)
Phosphorylase (1)
Glucagon Receptor (1)
Raf (1)
Fas/FasL (1)
MTH1 (1)
Prolyl Endopeptidase (PREP) (1)
IDO (1)
S1P Receptor (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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