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多肽分子库

多肽分子库

现 货
产品编号 L9600 Peptide Compound Library
  库化合物信息   Excel SDF

自1901年,肽分子首次在诺贝尔化学奖获得者 Emil Fischer 教授的一篇文章中亮相学术界,并于次年获得 Peptide 这一专属名词以来的一百余年,多肽分子一直活跃在药物领域。除了不断开创出索马鲁肽等传统激素类药物之外,多肽在抗感染、抗菌以及抗肿瘤领域都有着极其广阔的探索空间。

多肽是介于大分子蛋白质和小分子药物之间的具有调节细胞生物功能的化合物。由于其主要来源于天然多肽或者天然多肽类似物,通常情况下,其结构清楚、作用机制明确,许多性质往往介于小分子化学药物与大分子抗体药物之间。研究表明多肽具有靶点亲和力高、疗效稳定、免疫原性低、毒副作用小、特异性强等优点。

随着生物技术与多肽合成技术的日臻成熟,越来越多的多肽药物被开发并应用于临床。因适应症广、安全性高且疗效显著,多肽药物目前已被广泛应用于肿瘤、肝炎、糖尿病、艾滋病等领域,具有广阔的开发前景。

为满足进行多肽研究的客户需求,TargetMol 多肽化合物库收集了800 个多肽分子,可用于多肽类药物的开发和相关机制研究。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
咨询化合物库
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产品描述

  • 800种多肽类分子,可用于多肽药物开发及信号转导通路和作用机制研究;
  • 包括免疫活性肽、神经活性肽、激素肽、抗癌多肽、酶调节剂等多种类型多肽分子;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;
  • 严格质检,保证产品结构准确,纯度高,保障实验顺利进行。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L9600)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

Opioid Receptor (37)
Antibacterial (29)
RAAS (21)
Neurokinin receptor (21)
Glucagon Receptor (20)
Neuropeptide Y Receptor (19)
Integrin (16)
Melanocortin Receptor (15)
Endogenous Metabolite (15)
GNRH Receptor (14)
Antibiotic (13)
Beta Amyloid (13)
Bradykinin Receptor (13)
Protease-activated Receptor (12)
HIV Protease (11)
GPR (10)
Somatostatin (8)
Apoptosis (8)
PKC (8)
Autophagy (8)
CRFR (8)
CaMK (8)
cholecystokinin (7)
PKA (7)
Vasopressin Receptor (7)
CXCR (6)
Amino Acids and Derivatives (6)
Neurotensin Receptor (6)
IGF-1R (6)
Apelin receptor (5)
Caspase (5)
Calcium Channel (5)
Melanin-concentrating Hormone Receptor (MCHR) (5)
Gap Junction Protein (5)
GHSR (4)
Complement System (4)
Bombesin Receptor (4)
Endothelin Receptor (4)
Thyroid hormone receptor(THR) (3)
GluR (3)
Proteasome (3)
MMP (3)
Influenza Virus (3)
Serine Protease (3)
Oxytocin Receptor (3)
TLR (3)
AChR (3)
JNK (3)
Phospholipase (3)
Potassium Channel (3)
CGRP Receptor (3)
Microtubule Associated (2)
Cannabinoid Receptor (2)
OX Receptor (2)
Amylin Receptor (2)
HSP (2)
NF-κB (2)
STAT (2)
Ephrin Receptor (2)
Sodium Channel (2)
IL Receptor (2)
Guanylate cyclase (2)
Adrenergic Receptor (2)
Antioxidant (2)
c-Met/HGFR (2)
Antifungal (2)
Cysteine Protease (2)
ERK (2)
Raf (2)
NMDAR (2)
Phosphatase (2)
Adenylyl cyclase (1)
Thrombin (1)
GTPase (1)
LHRH (1)
Glutathione Peroxidase (1)
AMPK (1)
Histamine Receptor (1)
Histone Demethylase (1)
BACE (1)
5-HT Receptor (1)
P450 (1)
Reductase (1)
Kinesin (1)
TNF (1)
PD-1/PD-L1 (1)
Dopamine Receptor (1)
YAP (1)
Proton pump (1)
p38 MAPK (1)
p53 (1)
Galectin (1)
ATPase (1)
Dynamin (1)
DAPK (1)
Syk (1)
NADPH-oxidase (1)
Src (1)
Ras (1)
Piezo Channel (1)
Estrogen/progestogen Receptor (1)
Estrogen Receptor/ERR (1)
Retinoid Receptor (1)
PDE (1)
iGluR (1)
Glucocorticoid Receptor (1)
Annexin A (1)
PTEN (1)
Angiotensin-converting Enzyme (ACE) (1)
Motilin Receptor (1)
Gamma-secretase (1)
TGF-beta/Smad (1)
CDK (1)
CCR (1)
HSV (1)
P2X Receptor (1)
Fatty Acid Synthase (1)
APC (1)
Immunology/Inflammation related (1)
EGFR (1)
CaSR (1)
GPCR19 (1)
BCL (1)
PAI-1 (1)
PPAR (1)
Nrf2 (1)
Wnt/beta-catenin (1)
Sirtuin (1)
Trk receptor (1)
MAPK (1)
SARS-CoV (1)
Parasite (1)
Rho (1)
Antiviral (1)
Serine/threonin kinase (1)
Survivin (1)
NO Synthase (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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