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神经信号分子库

神经信号分子库

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产品编号 L2600 Neuronal Signaling Compound Library
  库化合物信息   Excel SDF

神经元之间和神经元内部的通信对于神经系统的所有功能至关重要,无论是从发育到衰老,还是从健康到疾病。在过去十年中,我们对神经系统内分子、细胞和系统信号通路的认识取得了巨大进步,在信号通路研究方面取得了重大突破,这些神经信号通路是神经发生、成瘾、自闭症以及情绪障碍的病理生理学和治疗基础。例如:G 蛋白偶联受体(GPCR),包括5-HT 受体、组胺受体、阿片受体等,是研究较多的神经元信号传导途径,GPCR 功能障碍会引起多种神经疾病;Notch 信号途径调节神经干细胞增殖、存活、自我更新和分化,Notch 信号传导异常参与中风、阿尔茨海默病和CNS 肿瘤等疾病中发生的病理过程。因此靶向神经元信号传导,可以用来治疗多种不同CNS 疾病。

TargetMol 神经信号分子库包含2540 种与中枢神经系统信号传导有关的小分子化合物,主要用于神经系统类疾病的药物研发,可用于高通量、高内涵筛选。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
咨询化合物库
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产品描述

  • 2540种CNS相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 靶点包括5-HT receptor、AChR、Histamine receptor、dopamine receptor、Opiod receptor等;?
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L2600)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

5-HT Receptor (334)
AChR (292)
COX (263)
Adrenergic Receptor (228)
Dopamine Receptor (220)
Calcium Channel (170)
Histamine Receptor (157)
GABA Receptor (131)
GluR (121)
Autophagy (118)
TRP/TRPV Channel (114)
Apoptosis (104)
Endogenous Metabolite (101)
iGluR (88)
AChE (86)
Adenosine Receptor (79)
Opioid Receptor (75)
NMDAR (73)
MAO (62)
Beta Amyloid (57)
Antibacterial (53)
NF-κB (45)
Monoamine Oxidase (43)
P-gp (42)
Potassium Channel (39)
Cannabinoid Receptor (38)
Serotonin Transporter (38)
Parasite (37)
P2X Receptor (36)
Gamma-secretase (36)
Norepinephrine (34)
Sodium Channel (34)
CaMK (31)
P450 (30)
FAAH (27)
Sigma receptor (23)
NO Synthase (22)
Reactive Oxygen Species (22)
Neurokinin receptor (22)
P2Y Receptor (20)
GPR (19)
Lipoxygenase (18)
PDE (18)
Antibiotic (18)
TNF (17)
HIV Protease (17)
OX Receptor (17)
Influenza Virus (17)
PPAR (17)
Neuropeptide Y Receptor (16)
Mitophagy (14)
Ferroptosis (14)
BACE (14)
Antifungal (13)
Beta-Secretase (12)
NOS (12)
Prostaglandin Receptor (12)
ERK (11)
IL Receptor (11)
Melanocortin Receptor (11)
Antioxidant (10)
Imidazoline Receptor (10)
Melatonin Receptor (10)
Phospholipase (10)
Drug Metabolite (9)
Caspase (9)
Virus Protease (9)
PGE Synthase (8)
MT Receptor (8)
HDAC (8)
ROS (8)
p38 MAPK (8)
DNA/RNA Synthesis (8)
HSV (7)
Akt (7)
GlyT (7)
SARS-CoV (7)
Interleukin (7)
AMPK (7)
Adenylyl cyclase (7)
Chloride channel (7)
HER (7)
Transferase (7)
BCL (6)
Estrogen/progestogen Receptor (6)
Glucocorticoid Receptor (6)
EGFR (6)
PKA (6)
MRP (6)
PKC (6)
HCV Protease (5)
IκB/IKK (5)
MMP (5)
STAT (5)
Carbonic Anhydrase (5)
Tyrosinase (5)
Dehydrogenase (5)
Microtubule Associated (5)
Glutathione Peroxidase (5)
Monoamine Transporter (4)
PI3K (4)
GSK-3 (4)
TLR (4)
CGRP Receptor (4)
NADPH (4)
Histone Demethylase (4)
PARP (4)
TGF-beta/Smad (4)
Histone Methyltransferase (4)
HIF/HIF Prolyl-Hydroxylase (4)
cholecystokinin (4)
AAK1 (AP2 associated kinase 1) (4)
Antifection (3)
ABC (3)
RAAS (3)
JNK (3)
Topoisomerase (3)
ATPase (3)
Phosphatase (3)
Immunology/Inflammation related (3)
Na+/Ca2+ Exchanger (3)
VEGFR (3)
PAFR (3)
Mitochondrial Metabolism (3)
Melanin-concentrating Hormone Receptor (MCHR) (3)
CCR (3)
Wnt/beta-catenin (3)
GST (3)
MEK (3)
Src (3)
transporter (3)
Anti-infection (3)
Neurotensin Receptor (3)
Serine/threonin kinase (3)
GluCls (2)
RSV (2)
Lipase (2)
advanced glycation end products (2)
BCRP (2)
Reductase (2)
Nrf2 (2)
DYRK (2)
IFNAR (2)
Acyltransferase (2)
Free radical scavengers (2)
Transaminase (2)
Amino Acids and Derivatives (2)
Hydroxylase (2)
cAMP (2)
mTOR (2)
PAK (2)
IAP (2)
ROCK (2)
UGT (2)
LDL (2)
Leukotriene Receptor (2)
CDK (2)
DNA Methyltransferase (2)
FAK (2)
NOD (2)
Guanylate cyclase (2)
Estrogen Receptor/ERR (2)
HBV (2)
Androgen Receptor (2)
JAK (2)
Aurora Kinase (2)
Progesterone Receptor (2)
Gap Junction Protein (2)
CaSR (2)
DNA (2)
IGF-1R (2)
Epoxide Hydrolase (2)
Epigenetic Reader Domain (2)
Thrombin (1)
NOD-like Receptor (NLR) (1)
CFTR (1)
S6 Kinase (1)
HMG-CoA Reductase (1)
ROS Kinase (1)
lysosomal autophagy (1)
FGFR (1)
AhR (1)
NMU2R (1)
Platelet aggregation (1)
NADPH-oxidase (1)
Syk (1)
Adenosine deaminase (1)
p53 (1)
FLT (1)
Protease-activated Receptor (1)
Bombesin Receptor (1)
CRISPR/Cas9 (1)
cell cycle arrest (1)
Bcr-Abl (1)
Adiponectin receptor (1)
FLAP (1)
Annexin A (1)
Myosin (1)
Aryl Hydrocarbon Receptor (1)
FXR (1)
Cysteine Protease (1)
Antifolate (1)
GRK (1)
N-Acetylglucosaminyltransferase (1)
OCT (1)
GTPase (1)
Neuropeptide W (1)
LPL Receptor (1)
Integrin (1)
ROR (1)
Monocarboxylate transporter (1)
CAT (1)
Raf (1)
Glucagon Receptor (1)
Retinoid Receptor (1)
Antiviral (1)
Reverse Transcriptase (1)
Casein Kinase (1)
Histone Acetyltransferase (1)
Sirtuin (1)
GPCR19 (1)
Aminopeptidase (1)
Trk receptor (1)
STING (1)
HSP (1)
MAPK (1)
Glucosidase (1)
Indoleamine 2,3-Dioxygenase (IDO) (1)
ACK (1)
PAD (1)
Somatostatin (1)
Stearoyl-CoA Desaturase (SCD) (1)
Proteasome (1)
Fatty Acid Synthase (1)
MAGL (1)
Anion Exchanger (1)
S1P Receptor (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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