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天然产物库

天然产物库

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产品编号 L6010 Natural Product Library
  库化合物信息   Excel SDF

天然产物在化学结构和生物活性多样性方面的优势,使其在新药研发中具有不可替代的重要地位。近年来提取分离和结构鉴定技术的快速发展, 大大提高了从天然产物中开发新药的效率和成功率。据统计,1981年至 2019年所有上市的药物中,有近2/3的药物在不同程度上都与天然产物相关。我国近50年自研成功的新药90%以上与天然产物有关。

然而,长期困扰天然产物药物筛选的问题之一是,得到天然产物苗头化合物进行后继的药理实验时,天然产物的成本太高。为了一定程度上帮助研发人员避免这个问题,TargetMol 推出L6010天然产物库,收集 3720 种天然产物单体,广泛涉及1800种植物来源。在筛得阳性化合物以后,您从自然界或者天然产物全合成中得到此产品大包装的难度更小,更能满足您对于苗头化合物进行深入研究时成本控制的需求。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
咨询化合物库
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产品描述

  • 3720种天然产物的独特集合,可用于高通量筛选和高内涵筛选;
  • 提供产品的生物学信息和药物学信息,为筛选提供理论方向和研究基础;
  • 来源清晰:精选来自动物、植物、微生物的已知活性天然产物;更具体到植物种属,并标注准确英文名与拉丁名,方便您的后期研究确证;
  • 结构多样性好:含黄酮类、生物碱类在内的多种化合物类型,拥有详细的分类信息;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L6010)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

Endogenous Metabolite (954)
Apoptosis (373)
Antibacterial (331)
Autophagy (243)
NF-κB (176)
Antibiotic (154)
Antifungal (117)
Reactive Oxygen Species (103)
Antioxidant (97)
COX (90)
Parasite (77)
Influenza Virus (66)
P450 (66)
DNA/RNA Synthesis (59)
TNF (57)
AChR (50)
Anti-infection (48)
HIV Protease (47)
AChE (46)
NO Synthase (44)
ERK (43)
p38 MAPK (43)
Akt (42)
IL Receptor (41)
Caspase (41)
Calcium Channel (41)
STAT (40)
PPAR (40)
GABA Receptor (37)
Tyrosinase (36)
AMPK (34)
Ferroptosis (34)
Virus Protease (33)
MMP (32)
Topoisomerase (32)
Estrogen/progestogen Receptor (31)
Microtubule Associated (29)
PKC (29)
BCL (29)
ROS (29)
PI3K (29)
5-HT Receptor (29)
JNK (26)
Estrogen Receptor/ERR (26)
Dehydrogenase (26)
Potassium Channel (26)
Nrf2 (25)
Adrenergic Receptor (25)
HSV (24)
Lipoxygenase (24)
Mitophagy (24)
ribosome (23)
Prostaglandin Receptor (22)
NOS (22)
Beta Amyloid (21)
TRP/TRPV Channel (20)
ATPase (20)
Glucosidase (20)
Antifection (20)
PARP (19)
PDE (19)
Sodium Channel (19)
P-gp (19)
Antiviral (18)
Immunology/Inflammation related (17)
Nucleoside Antimetabolite/Analog (16)
Dopamine Receptor (16)
Wnt/beta-catenin (16)
Interleukin (15)
Mitochondrial Metabolism (15)
EGFR (15)
HIF/HIF Prolyl-Hydroxylase (15)
HBV (14)
Adenosine Receptor (14)
JAK (14)
iGluR (14)
Phosphatase (14)
HDAC (14)
VEGFR (13)
TLR (13)
SARS-CoV (13)
Drug Metabolite (13)
Histamine Receptor (12)
MAO (12)
NMDAR (12)
mTOR (12)
Opioid Receptor (11)
HCV Protease (11)
Reductase (11)
TGF-beta/Smad (11)
Phospholipase (11)
Androgen Receptor (11)
Cannabinoid Receptor (11)
Sirtuin (10)
HSP (9)
HMG-CoA Reductase (9)
NOD (9)
GluR (9)
Amino Acids and Derivatives (9)
Glucocorticoid Receptor (9)
MAPK (9)
transporter (8)
p53 (8)
CDK (8)
RAAS (8)
PKA (8)
HIF (8)
Fatty Acid Synthase (8)
FXR (7)
IκB/IKK (7)
GPR (7)
MEK (7)
UGT (7)
Monoamine Oxidase (7)
Progesterone Receptor (7)
Transferase (6)
Carbonic Anhydrase (6)
CaMK (6)
Reverse Transcriptase (6)
BACE (6)
Indoleamine 2,3-Dioxygenase (IDO) (6)
Xanthine Oxidase (6)
Aryl Hydrocarbon Receptor (6)
Proteasome (5)
NOD-like Receptor (NLR) (5)
HER (5)
Gamma-secretase (5)
Epigenetic Reader Domain (5)
MRP (5)
IGF-1R (5)
PTEN (5)
c-Met/HGFR (5)
LDL (5)
PAFR (5)
Retinoid Receptor (5)
FAAH (5)
Aromatase (5)
Chloride channel (5)
CXCR (4)
FGFR (4)
Lipid (4)
Beta-Secretase (4)
PGE Synthase (4)
cAMP (4)
FAK (4)
ATP Citrate Lyase (4)
Proton pump (4)
Tyrosine Kinases (4)
AhR (4)
Serine Protease (4)
ABC (4)
Arginase (4)
NADPH (4)
Platelet aggregation (4)
IAP (4)
E1/E2/E3 Enzyme (4)
Cysteine Protease (4)
GST (4)
DNA Methyltransferase (4)
Serine/threonin kinase (4)
Histone Acetyltransferase (4)
Thyroid hormone receptor(THR) (4)
Antifolate (4)
S6 Kinase (4)
Integrin (4)
Src (4)
GSK-3 (4)
ROR (4)
Hedgehog/Smoothened (4)
DHFR (4)
Trk receptor (3)
Acyltransferase (3)
Free radical scavengers (3)
GPCR19 (3)
PDK (3)
Syk (3)
Aminopeptidase (3)
Bombesin Receptor (3)
Telomerase (3)
CCR (3)
LTR (3)
Glutathione Peroxidase (3)
Serotonin Transporter (3)
Liver X Receptor (3)
Phosphorylase (3)
P2X Receptor (3)
DNA gyrase (3)
PDGFR (3)
cell cycle arrest (3)
S1P Receptor (2)
Aurora Kinase (2)
Thrombin (2)
Bcr-Abl (2)
Adiponectin receptor (2)
Ras (2)
Amylase (2)
RANKL/RANK (2)
Glucokinase (2)
Leukotriene Receptor (2)
SGLT (2)
Casein Kinase (2)
IRAK (2)
Pim (2)
DNA Alkylator/Crosslinker (2)
P2Y Receptor (2)
Hydroxylase (2)
DNA (2)
Lipase (2)
Neurokinin receptor (2)
Cell wall (2)
Amylin Receptor (2)
DYRK (2)
Pyroptosis (2)
Decarboxylase (2)
DPP-4 (2)
CAT (2)
Imidazoline Receptor (2)
PKM (2)
PAK (2)
Smo (2)
Monoamine Transporter (2)
hCE (2)
OAT (2)
Glutathione reductase (2)
PAI-1 (2)
aconitase (1)
NMU2R (1)
IFNAR (1)
Mdm2 (1)
advanced glycation end products (1)
NADPH-oxidase (1)
LPL Receptor (1)
FLT (1)
PD-1/PD-L1 (1)
Adenylyl cyclase (1)
Hydrogenase (1)
MyD88 (1)
CFTR (1)
Transaminase (1)
Dynamin (1)
ROS Kinase (1)
cholecystokinin (1)
Histone Methyltransferase (1)
NPC1L1 (1)
ATTECs (1)
Monocarboxylate transporter (1)
stilbene oxidase (1)
CYP19A1 (1)
Bradykinin Receptor (1)
RAR/RXR  (1)
BCRP (1)
RSV (1)
ALK (1)
GluCls (1)
Raf (1)
MT Receptor (1)
Glucagon Receptor (1)
Epoxide Hydrolase (1)
MTH1 (1)
PAD (1)
GlyT (1)
Hexokinase (1)
Somatostatin (1)
DNA Alkylation (1)
Stearoyl-CoA Desaturase (SCD) (1)
Fas/FasL (1)
ATM/ATR (1)
Histone Demethylase (1)
Survivin (1)
PERK (1)
Norepinephrine (1)
Adenosine deaminase (1)
Factor Xa (1)
Melatonin Receptor (1)
OCT (1)
Oxytocin Receptor (1)
Carboxypeptidase (1)
CaSR (1)
Thrombopoietin Receptor (1)
CRISPR/Cas9 (1)
IDO (1)
Prolyl Endopeptidase (PREP) (1)
IRE1 (1)
c-Myc (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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