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激酶抑制剂库

激酶抑制剂库

产品编号 L1600 Kinase Inhibitor Library
  库化合物信息   Excel SDF

在生物化学中,激酶是一类从高能供体分子(如 ATP)转移磷酸基团到特定靶分子的酶;这一过程谓之磷酸化。比较常见的激酶族群是蛋白激酶,蛋白激酶作用于特定的蛋白质,使其磷酸化而改变其活性。这些激酶在细胞的信号转导及其复杂的生命活动中起了广泛的作用。其他不同的激酶作用于小分子物质(脂质、糖、氨基酸、核苷等),或者为了发出信号,或者使它们为代谢中各种生化反应作好准备。

TargetMol 激酶抑制剂库含有 2230 种具有明确激酶抑制活性的小分子化合物,这些抑制剂作用的激酶包括:Insulin/IGF Receptors、PI 3-Kinase、CaM Kinase II、JAKPKACDKJNKPKC、CKI II、MAPKRAFEGFRMEK、SAPK、GSK、MLCK、Src-family、IKK、PDGFRVEGFR 等。该库是化学基因组学和药理学研究的理想工具。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
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产品描述

  • 2230种激酶抑制剂的独特集合,用于特定靶向激酶,可用于高通量筛选和高内涵筛选;
  • 其中一些激酶抑制剂已得到FDA批准上市;
  • 大部分为ATP竞争性抑制剂;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR和HPLC检测技术保证产品高纯度;
  • 所有化合物现货供应。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L1600)
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化合物库组成

Apoptosis (382)
Autophagy (284)
CDK (166)
PI3K (156)
EGFR (145)
VEGFR (142)
Reactive Oxygen Species (140)
JAK (94)
FLT (89)
Akt (85)
PDGFR (85)
ERK (84)
mTOR (84)
Src (81)
p38 MAPK (78)
Endogenous Metabolite (72)
NF-κB (72)
FGFR (72)
PKC (68)
c-Kit (67)
Raf (66)
c-Met/HGFR (60)
Antibacterial (58)
Ras (57)
GSK-3 (54)
Bcr-Abl (51)
AMPK (50)
Aurora Kinase (49)
ALK (49)
ROS (48)
JNK (45)
Tyrosine Kinases (42)
MEK (42)
TGF-beta/Smad (40)
MAPK (40)
BTK (39)
Serine/threonin kinase (36)
Casein Kinase (36)
DNA-PK (35)
ROCK (33)
TAM Receptor (33)
PKA (33)
IGF-1R (32)
IκB/IKK (32)
CaMK (32)
c-RET (31)
S6 Kinase (30)
HER (30)
PLK (27)
Parasite (27)
Trk receptor (27)
FAK (26)
COX (26)
Ferroptosis (25)
RIP kinase (25)
Influenza Virus (24)
TNF (24)
STAT (24)
Epigenetic Reader Domain (23)
Glucosidase (23)
Antibiotic (22)
ATM/ATR (22)
c-Fms (22)
Syk (21)
HIV Protease (21)
Chk (20)
Antifungal (20)
LRRK2 (19)
Caspase (18)
Mitophagy (17)
Aryl Hydrocarbon Receptor (17)
Potassium Channel (17)
Pim (16)
Antioxidant (16)
PDK (16)
IRAK (16)
DNA/RNA Synthesis (15)
Tyrosinase (15)
Calcium Channel (15)
Glucokinase (15)
PAK (15)
P450 (15)
IL Receptor (15)
DYRK (14)
IRE1 (14)
PERK (13)
PPAR (13)
5-HT Receptor (13)
PI4K (12)
Mitochondrial Metabolism (12)
CSF-1R (12)
Dehydrogenase (12)
ROR (11)
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MMP (11)
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SGK (8)
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SGLT (1)
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Fer/FerT kinase (1)
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Na+/Ca2+ Exchanger (1)
RSV (1)
Cysteine Protease (1)
MRP (1)
Phosphorylase (1)
Monoamine Transporter (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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