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抗感染化合物库

抗感染化合物库

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产品编号 L1800 Anti-Infection Compound Library
  库化合物信息   Excel SDF

当外来生物进入人体并造成伤害时就会发生感染,这些引起感染的外来生物称为病原体,例如细菌、病毒、真菌和寄生虫等。有些感染是轻微的几乎不可察觉,但有些感染严重甚至危及生命,且对治疗有抵抗力。

针对上述情况,TargetMol 精选了2977 种具有抗菌、抗病毒以及抗寄生虫等抗感染活性的化合物的组成抗感染化合物库,以用于抗感染研究中的药物高通量筛选、确认药物靶点以及其他医药研发和科研领域。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
咨询化合物库
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产品描述

  • 2977种具有抗感染活性的化合物的特有集合,包括抗细菌、抗真菌、抗巨细胞病毒、抗HIV、抗SARS、抗流感等活性;
  • 含有磺胺类,氨基糖苷类,四环素类和大环内酯类等化合物,是筛选新型抗感染药的有效工具;可用于高通量筛选和高内涵筛选;
  • 通过前期临床研究和临床实验,生物活性和安全性已经得到验证;其中一些抗感染化合物已得到FDA批准上市;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L1800)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

Antibacterial (234)
Antibiotic (168)
HIV Protease (88)
Antifungal (79)
Antifection (72)
DNA/RNA Synthesis (69)
Parasite (50)
Autophagy (44)
HCV Protease (44)
Antiviral (42)
Topoisomerase (40)
Endogenous Metabolite (37)
AChR (36)
ribosome (31)
Influenza Virus (29)
COX (27)
NF-κB (27)
P450 (25)
Dehydrogenase (25)
HBV (21)
Apoptosis (21)
Antioxidant (20)
Reverse Transcriptase (18)
ATPase (18)
Histamine Receptor (18)
Microtubule Associated (17)
GABA Receptor (17)
HSV (16)
STAT (15)
PKC (14)
Dopamine Receptor (14)
ROS (14)
Sodium Channel (14)
Tyrosinase (13)
CCR (13)
IL Receptor (13)
TLR (13)
HDAC (12)
Estrogen/progestogen Receptor (12)
Nucleoside Antimetabolite/Analog (12)
TNF (11)
Caspase (11)
Adrenergic Receptor (11)
SARS-CoV (11)
DNA gyrase (11)
5-HT Receptor (10)
Akt (10)
Potassium Channel (10)
Proton pump (9)
MMP (9)
Vitamin (9)
PI3K (9)
p38 MAPK (8)
PARP (8)
mTOR (8)
MAO (8)
BCL (8)
CDK (8)
CXCR (8)
AMPK (8)
Glucocorticoid Receptor (8)
CAT (7)
JAK (7)
DHFR (7)
EGFR (7)
Epigenetic Reader Domain (7)
Phosphatase (7)
Glucokinase (7)
Phospholipase (7)
Adenosine Receptor (7)
TRP/TRPV Channel (6)
DNA Methyltransferase (6)
Cysteine Protease (6)
Retinoid Receptor (6)
P2 Receptor (6)
HSP (6)
NMDAR (6)
PPAR (6)
PDE (6)
DNA Alkylation (6)
PKA (6)
Serine Protease (5)
Sirtuin (5)
Cell wall (5)
Lipoxygenase (5)
Carbonic Anhydrase (5)
Lipid (5)
Calcium Channel (5)
cAMP (4)
DprE1 (4)
NADPH (4)
Reductase (4)
MEK (4)
ERK (4)
NOS (4)
Src (4)
Bcr-Abl (4)
P-gp (4)
PDGFR (4)
Proteasome (4)
S6 Kinase (4)
Anti-infection (4)
p53 (4)
Thyroid hormone receptor(THR) (3)
DNA-PK (3)
Thrombin (3)
JNK (3)
FXR (3)
RSV (3)
IκB/IKK (3)
GSK-3 (3)
Tyrosine Kinases (3)
transporter (3)
NADPH-oxidase (3)
Opioid Receptor (3)
ATM/ATR (3)
Virus Protease (3)
VEGFR (3)
ABC (3)
BACE (3)
Chk (3)
Chloride channel (3)
CRM1 (3)
HIF (2)
PKM (2)
Hedgehog/Smoothened (2)
Histone Demethylase (2)
PAFR (2)
Prostaglandin Receptor (2)
Histone Methyltransferase (2)
Serine/threonin kinase (2)
HMG-CoA Reductase (2)
PLK (2)
RAAS (2)
IAP (2)
Integrase (2)
MPO (2)
Nrf2 (2)
Norepinephrine (2)
NOD (2)
LTR (2)
Raf (2)
Mitochondrial Metabolism (2)
MRP (2)
GPR (2)
Monoamine Transporter (2)
Androgen Receptor (2)
Aminopeptidase (2)
GPCR19 (2)
Ferroptosis (2)
Transferase (2)
Telomerase (2)
Electron transport (2)
Syk (2)
UGT (2)
Estrogen Receptor/ERR (2)
STING (2)
Cannabinoid Receptor (2)
CaMK (2)
Beta Amyloid (2)
Wnt/beta-catenin (2)
TGF-beta/Smad (2)
Fatty Acid Synthase (2)
FAK (2)
Free radical scavengers (2)
AhR (2)
Arginase (2)
Annexin A (2)
GluCls (2)
GluR (2)
PI4K (1)
Deubiquitinase (1)
c-Met/HGFR (1)
Ras (1)
Amino Acids and Derivatives (1)
PERK (1)
c-Kit (1)
cell cycle arrest (1)
Neurokinin receptor (1)
PDK (1)
NO Synthase (1)
Adiponectin receptor (1)
VDA (1)
ASK (1)
Casein Kinase (1)
Acyltransferase (1)
AChE (1)
BMI-1 (1)
PAK (1)
Acetyl-CoA Carboxylase (1)
Xanthine Oxidase (1)
Aurora Kinase (1)
P2X Receptor (1)
Aromatase (1)
Mitophagy (1)
Rho (1)
DUB (1)
Hexokinase (1)
S1P Receptor (1)
FLT (1)
Gap Junction Protein (1)
Histone Acetylation (1)
HIF/HIF Prolyl-Hydroxylase (1)
Somatostatin (1)
HER (1)
Hydroxylase (1)
Glutathione reductase (1)
SGK (1)
Hck (1)
SGLT (1)
GST (1)
GNRH Receptor (1)
Hydrogenase (1)
IDO (1)
MicroRNA (1)
LIM Kinase (1)
Dynamin (1)
Mdm2 (1)
MAPK (1)
gp120/CD4 (1)
TAM Receptor (1)
Lipase (1)
RIP kinase (1)
IFNAR (1)
IRAK (1)
Integrin (1)
ROCK (1)
Immunology & Inflammation related (1)
Factor Xa (1)
IGF-1R (1)
DNA (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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