首页 工具
登录
购物车
血管生成库

血管生成库

现 货
产品编号 L4800 Angiogenesis related Compound Library
  库化合物信息   Excel SDF

血管生成是正常生长和发育过程以及伤口愈合和肉芽组织形成过程中的基本事件,然而异常的血管生成将导致各种疾病,例如肿瘤、糖尿病、免疫病、先兆子痫、肢体缺血等。因此,血管生成已成为治疗这些疾病的药物靶点。例如,血管生成与癌症发生密切相关,肿瘤通过分泌各种生长因子(例如VEGF)和蛋白质诱导毛细血管生成进入肿瘤,为癌细胞提供氧气和其他必需的营养物质,并及时运走代谢废物,血管生成也是肿瘤扩散或转移所必需的。因此血管生成抑制剂用于治疗癌症。此外,诱导血管生成,建立新的侧支循环是治疗缺血性心脑血管疾病(冠心病、脑卒中等)的极佳治疗方式。有效新生血管靶分子的筛选为相关疾病研究带来了广阔前景。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
咨询化合物库
点击图片重新获取验证码
获取报价
点击图片重新获取验证码

产品描述

  • 1370个高潜力的抑制或促进血管生成的小分子集合,可用于药物靶点开发、血管生成机理研究的高通量筛选,高内涵筛选;
  • 包含了目前研究较多潜力的血管生成通路以及S1P、VEGFR、PDGF等相关靶点的热门产品;
  • 包含了Sunitinib Malate、Lenalidomide、sorafenib、Erlotinib等研究成熟的上市药物,以及Vatalanib、Orantinib、2-Methoxyestradiol(Panzem)、Celecoxib等临床药物;
  • 是研究血管生成机理以及药物靶向研究的有效工具;
  • 产品经过临床验证和临床实验,具有生物安全保障和一定的生物活性;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR和HPLC检测技术保证产品高纯度和高质量;
  • 所有化合物现货供应。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L4800)
点击图片重新获取验证码

TargetMol Library Books客户使用化合物库发表的文献

收起

化合物库组成

5-HT Receptor (248)
Apoptosis (202)
Autophagy (158)
PI3K (152)
EGFR (141)
VEGFR (136)
JAK (90)
FLT (81)
Src (81)
PDGFR (80)
Dopamine Receptor (76)
Akt (72)
FGFR (71)
TNF (63)
COX (60)
c-Kit (58)
MMP (54)
Bcr-Abl (51)
ALK (49)
RAAS (48)
mTOR (45)
Adrenergic Receptor (40)
TGF-beta/Smad (38)
Endogenous Metabolite (38)
HER (37)
NF-κB (37)
BTK (36)
Histamine Receptor (33)
Tyrosine Kinases (31)
c-Met/HGFR (30)
HIF (30)
Antibacterial (30)
IL Receptor (29)
AChR (26)
FAK (26)
DNA-PK (24)
CDK (24)
ERK (23)
HIF/HIF Prolyl-Hydroxylase (22)
Reactive Oxygen Species (22)
Serotonin Transporter (21)
c-RET (21)
Syk (20)
STAT (20)
p38 MAPK (19)
Aurora Kinase (19)
IGF-1R (18)
PKC (17)
Norepinephrine (17)
Potassium Channel (17)
Raf (16)
c-Fms (14)
Influenza Virus (14)
Parasite (14)
TAM Receptor (14)
PKA (13)
AMPK (12)
Trk receptor (12)
HIV Protease (11)
JNK (11)
ROS (11)
NO Synthase (11)
HDAC (11)
S6 Kinase (10)
MEK (10)
Drug Metabolite (9)
Virus Protease (9)
Caspase (9)
Antibiotic (8)
CSF-1R (8)
Interleukin (8)
P450 (8)
Mitophagy (8)
Tyrosinase (8)
Casein Kinase (7)
Ferroptosis (7)
Lipoxygenase (7)
ROS Kinase (7)
DNA/RNA Synthesis (7)
Sodium Channel (7)
Ephrin Receptor (6)
Prostaglandin Receptor (6)
MLK (6)
ATM/ATR (6)
GSK-3 (6)
Antifungal (6)
PDE (6)
PI4K (6)
Integrin (6)
ROCK (5)
Nrf2 (5)
Antioxidant (5)
Microtubule Associated (5)
SARS-CoV (5)
PDK (5)
PYK2 (5)
Ligand for E3 Ligase (5)
P-gp (5)
PLK (5)
PPAR (5)
Sigma receptor (5)
TLR (5)
HCV Protease (5)
Chk (5)
Carbonic Anhydrase (4)
Dehydrogenase (4)
MAPK (4)
Topoisomerase (4)
Transferase (4)
BCL (4)
Adenosine Receptor (4)
Serine/threonin kinase (4)
Histone Methyltransferase (4)
NOS (4)
IκB/IKK (4)
Tie-2 (4)
ACK (4)
HSP (4)
HSV (4)
Opioid Receptor (4)
IFNAR (4)
PARP (3)
TRP/TRPV Channel (3)
NOD (3)
Reverse Transcriptase (3)
Beta Amyloid (3)
MRP (3)
Anti-infection (3)
Glucosidase (3)
PGE Synthase (3)
Discoidin Domain Receptor (DDR) (3)
CaMK (3)
Molecular Glues (3)
Serine Protease (3)
CCR (3)
AChE (3)
Ligands for Target Protein for PROTAC (3)
Estrogen/progestogen Receptor (3)
Survivin (3)
DYRK (3)
Sirtuin (3)
Hck (3)
Proton pump (2)
PTEN (2)
Wnt/beta-catenin (2)
p53 (2)
GABA Receptor (2)
GluR (2)
ribosome (2)
VDA (2)
Calcium Channel (2)
IRAK (2)
IRE1 (2)
Leukotriene Receptor (2)
transporter (2)
SGK (2)
MAO (2)
Guanylate cyclase (2)
SGLT (2)
iGluR (2)
RIP kinase (2)
BCRP (2)
NOD-like Receptor (NLR) (2)
BACE (2)
Epigenetic Reader Domain (2)
ROR (1)
STING (1)
Stearoyl-CoA Desaturase (SCD) (1)
RSV (1)
S1P Receptor (1)
PROTACs (1)
Pyroptosis (1)
PROTAC Linker (1)
LDL (1)
PKM (1)
DNA Alkylator/Crosslinker (1)
Gap Junction Protein (1)
Gamma-secretase (1)
FXR (1)
Free radical scavengers (1)
FAAH (1)
Estrogen Receptor/ERR (1)
Epoxide Hydrolase (1)
Endothelin Receptor (1)
E1/E2/E3 Enzyme (1)
DUB (1)
DNA Alkylation (1)
GST (1)
CXCR (1)
CRISPR/Cas9 (1)
Chloride channel (1)
CFTR (1)
cell cycle arrest (1)
Beta-Secretase (1)
ATPase (1)
ATP Citrate Lyase (1)
Antifection (1)
Acyltransferase (1)
GRK (1)
HBV (1)
Pim (1)
Na+/Ca2+ Exchanger (1)
Phospholipase (1)
Phosphatase (1)
PERK (1)
PAD (1)
p97 (1)
P2X Receptor (1)
NMDAR (1)
Neprilysin (1)
NADPH-oxidase (1)
NADPH (1)
Myosin (1)
Hedgehog/Smoothened (1)
Monoamine Transporter (1)
MNK (1)
Melatonin Receptor (1)
Melanin-concentrating Hormone Receptor (MCHR) (1)
LTR (1)
LRRK2 (1)
Immunology/Inflammation related (1)
Histone Demethylase (1)
Histone Acetyltransferase (1)
Hippo pathway (1)
YAP (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
TargetMol Loading
陶术
生物
TargetMol®中国区唯一合作伙伴
点击进入陶术生物官网陶术生物
联系我们
400-820-0310

上海市静安区江场三路238号8楼