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k-111

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  • 抑制剂&激动剂
    9
    TargetMol | Inhibitors_Agonists
  • 多肽产品
    1
    TargetMol | Peptide_Products
  • PROTAC
    1
    TargetMol | PROTAC
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    1
    TargetMol | Natural_Products
  • K-111
    K111, K 111, BM-170744, BM170744, BM 170744
    T27706221564-97-2In house
    K-111 (BM-170744) 是一种可口服的过氧化物酶体增殖物激活受体 (PPAR)-α 激动剂和胰岛素增强剂,可用于研究肥胖型糖尿病和代谢综合征。
    • ¥ 1980 TargetMol
    In stock
    规格
    数量
  • PK 11195
    RP 52028
    T1654685532-75-8
    PK 11195 (RP 52028) 是一种用于神经成像的 TSPO 配体,对 CoCl2 诱导的改变表现出显着的保护能力,可用于研究利什曼病。
    • ¥ 272
    In stock
    规格
    数量
  • (R)-N-Desmethyl PK11195
    (R)-N-Desmethyl PK 11195,(R)-N-Desmethyl PK-11195,(R)-N Desmethyl PK11195,(R) N-Desmethyl PK11195
    T29258157809-85-3
    (R)-N-Desmethyl PK11195 is a precursor for (R)-[N-Methyl-11C-]PK11195.
    • ¥ 10600
    待询
    规格
    数量
  • serabelisib
    TAK-117, MLN1117, INK1117
    T31531268454-23-4
    Serabelisib (INK1117) 是选择性的 p110α 抑制剂,其 IC50=15 nM。
    • ¥ 292
    In stock
    规格
    数量
    TargetMol | Inhibitor Sale
  • AMPK-α1β1γ1 activator 1
    T831251943510-86-8
    AMPK-α1β1γ1激活剂1 (M1) 是一个衍生于Indole-3-carcinoma的酰基葡萄糖醛酸代谢AMPK激活剂,专一性地针对人类β1亚型,表现出38.1nM的EC50值。该化合物能够直接结合至人AMPK α1β1γ1亚型,适用于糖尿病肾病的相关研究。
    • 待询
    8-10周
    规格
    数量
  • (rel)-Asperparaline A
    T37609195966-93-9
    Aspergillimide is a fungal metabolite originally isolated from A. japonicus.1 It reduces nicotinic acetylcholine receptor (nAChR) peak and slowly-desensitizing amplitudes induced by acetylcholine in silkworm (B. mori) larval neurons (IC50s = 20.2 and 39.6 nM, respectively) but has no effect on chicken α3β4-, α4β2-, and α7-containing nAChRs.2 Dietary administration of aspergillimide A (10 μg/g of diet) induces paralysis in silkworm fourth instar larvae.1 Aspergillimide A (10 and 20 mg/kg) reduces T. colubriformis fecal egg count in gerbils.3References1. Hayashi, H., Nishimoto, Y., Akiyama, K., et al. New paralytic alkaloids, asperparalines A, B and C, from Aspergillus japonicus JV-23. Biosci. Biotechnol. Biochem. 64(1), 111-115 (2000).2. Hirata, K., Kataoka, S., Furutani, S., et al. A fungal metabolite asperparaline a strongly and selectively blocks insect nicotinic acetylcholine receptors: The first report on the mode of action. PLoS One 6(4), e18354 (2011).3. Banks, R.M., Blanchflower, S.E., Everett, J.R., et al. Novel anthelmintic metabolites from an Aspergillus species; the aspergillimides. J. Antibiot. (Tokyo) 50(10), 840-846 (1997). Aspergillimide is a fungal metabolite originally isolated from A. japonicus.1 It reduces nicotinic acetylcholine receptor (nAChR) peak and slowly-desensitizing amplitudes induced by acetylcholine in silkworm (B. mori) larval neurons (IC50s = 20.2 and 39.6 nM, respectively) but has no effect on chicken α3β4-, α4β2-, and α7-containing nAChRs.2 Dietary administration of aspergillimide A (10 μg/g of diet) induces paralysis in silkworm fourth instar larvae.1 Aspergillimide A (10 and 20 mg/kg) reduces T. colubriformis fecal egg count in gerbils.3 References1. Hayashi, H., Nishimoto, Y., Akiyama, K., et al. New paralytic alkaloids, asperparalines A, B and C, from Aspergillus japonicus JV-23. Biosci. Biotechnol. Biochem. 64(1), 111-115 (2000).2. Hirata, K., Kataoka, S., Furutani, S., et al. A fungal metabolite asperparaline a strongly and selectively blocks insect nicotinic acetylcholine receptors: The first report on the mode of action. PLoS One 6(4), e18354 (2011).3. Banks, R.M., Blanchflower, S.E., Everett, J.R., et al. Novel anthelmintic metabolites from an Aspergillus species; the aspergillimides. J. Antibiot. (Tokyo) 50(10), 840-846 (1997).
    • ¥ 1850
    35日内发货
    规格
    数量
  • Brain-Derived Acidic Fibroblast Growth Factor (102-111) (bovine) (trifluoroacetate salt)
    T37819
    Brain-derived acidic fibroblast growth factor (102-111) is a peptide fragment of brain-derived acidic fibroblast growth factor (aFGF). aFGF is an angiogenic vascular endothelial cell mitogen produced in bovine brain that has sequence homology to interleukin-1. It also shares sequence homology with the known neuropeptides neuromedin C , bombesin , neuromedin K , substance K , substance P , physalaemin, and eledoisin. aFGF (102-111) corresponds to amino acid residues 102-111 of the fulllength peptide.
    • 待估
    35日内发货
    规格
    数量
  • Antibacterial agent 111
    T611232448358-84-5
    Antibacterial agent 111 (Compound 3) exhibits potent antibacterial activity against B. cereus and K. pneumonia, with MIC values of 3.90 μg mL and 0.49 μg mL, respectively. It achieves this antibacterial effect by strongly binding to specific residues of tyrosyl-tRNA synthetase [1].
    • ¥ 10600
    6-8周
    规格
    数量
  • GXF-111
    T79034
    GXF-111是一种PROTAC分子,能够选择性促进BRD3与BRD4-L在细胞内的降解。该分子与BRD3BD1和BRD3BD2的结合亲和力显著,Ki值分别为11.97 nM和2.35 nM。GXF-111主要用于癌症研究领域。
    • 待询
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