Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T15817 |
Eglumegad
Eglumetad,LY354740 |
Others | Others |
Eglumegad is a highly effective and selective agonist of group II (mGlu2/3) receptor (IC50s: 5 and 24 nM on transfected human mGlu2 and mGlu3 receptors, respectively). | |||
T78094 |
Eglumegad hydrochloride
LY354740 hydrochloride,Eglumetad hydrochloride |
Others | Others |
Eglumegad (LY354740) hydrochloride是一种高效且选择性的group II (mGlu2/3) receptor激动剂,其对人mGlu2和mGlu3受体的IC50值分别是5和24 nM。该化合物能够保护神经元不受NMDA毒性影响,并表现出抗焦虑及抗精神病样作用。 | |||
T60611 |
Talaglumetad hydrochloride
|
Others | Others |
Talaglumetad (hydrochloride) 是Eglumegad 的前药,Eglumegad 是II 型代谢型谷氨酸受体(mGluR2/3)有效选择性的激动剂,用于治疗焦虑等精神疾病。 |