L8600
|
泛素化化合物库
|
|
214 compounds
|
|
214种泛素化相关的小分子,用于高通量和高内涵筛选;
|
L8500
|
HIF-1化合物库
|
|
1352 compounds
|
|
1352个HIF-1相关小分子的独特集合,可用于缺血性疾病、癌症等相关领域的药物开发和药理研究;
|
L4710
|
非甾体类抗炎化合物库
|
|
530 compounds
|
|
530种非甾体类的抗炎相关化合物,可用于高通量和高内涵筛选;
|
L9700
|
内质网应激化合物库
|
|
193 compounds
|
|
193个内质网应激相关的化合物集合,可用于高通量和高内涵筛选;
|
L2191
|
抗乳腺癌化合物库
|
|
1965 compounds
|
|
1965种与乳腺癌相关的化合物,可以用于抗乳腺癌药物研发和药理研究;
|
DC1140
|
特权片段注释化合物库-Ligand-gated
|
|
9028 compounds
|
|
|
DC1180
|
特权片段注释化合物库-Lyases
|
|
19530 compounds
|
|
|
DC1150
|
特权片段注释化合物库-GPCR Family B
|
|
9320 compounds
|
|
|
DC1170
|
特权片段注释化合物库-Oxidoreductases
|
|
8812 compounds
|
|
|
DC1190
|
特权片段注释化合物库-Sigma Opioid receptors
|
|
8724 compounds
|
|
|
DC1040
|
特权片段注释化合物库-Transferases
|
|
23001 compounds
|
|
|
DC1030
|
特权片段注释化合物库-Epigenetics
|
|
9196 compounds
|
|
|
DC1100
|
特权片段注释化合物库-GPCR Frizzled family
|
|
3434 compounds
|
|
|
DC1200
|
特权片段注释化合物库-Isomerases
|
|
1206 compounds
|
|
|
DC1050
|
特权片段注释化合物库-Voltage-gated
|
|
17952 compounds
|
|
|
DC1110
|
特权片段注释化合物库-Proteases
|
|
22863 compounds
|
|
|
DC1010
|
特权片段注释化合物库-GPCR Family A
|
|
24763 compounds
|
|
|
DC1000
|
特权片段注释化合物库
|
|
190000 compounds
|
|
The database contains 190k small molecules divided into 23 sub libraries each focused at a specific target.
According to the recent studies, molecules acting on a particular target or class of targets usually have characteristic moieties (PF) containing key binding points responsible for activity, e.g. hinge-binding fragments. We used this principle for the statistical analysis of the reported active molecules and corresponding targets for the annotation of pre-filtered ChemDiv in house colle...
|
DC1130
|
特权片段注释化合物库-Phosphodiesterases
|
|
13154 compounds
|
|
|
DC1060
|
特权片段注释化合物库-Kinases
|
|
18350 compounds
|
|
|
DC1220
|
特权片段注释化合物库-Aminoacyltransferases
|
|
3008 compounds
|
|
|
DC1210
|
特权片段注释化合物库-Phosphatases
|
|
15354 compounds
|
|
|
DC1160
|
特权片段注释化合物库-Toll-like and Il-1 receptors
|
|
3536 compounds
|
|
|
DC1090
|
特权片段注释化合物库-Ligases
|
|
11828 compounds
|
|
|
DQ3000
|
Factor XIa化合物库
|
|
6500 compounds
|
|
|
DC1080
|
特权片段注释化合物库-GPCR Taste family
|
|
2675 compounds
|
|
|
DC1120
|
特权片段注释化合物库-Thrombopoietin receptors
|
|
4908 compounds
|
|
|
DC1230
|
特权片段注释化合物库-Beta amyloid A4 protein
|
|
4617 compounds
|
|
|
DC1070
|
特权片段注释化合物库-GPCR Family C
|
|
5071 compounds
|
|
|
DC1020
|
特权片段注释化合物库-Spiro Library
|
|
20563 compounds
|
|
|
L1380
|
转录因子库
|
|
704 compounds
|
|
704种转录因子靶向、结构新颖的化合物;
|
L6900
|
稀有天然产物库
|
|
284 compounds
|
|
284种稀有天然产物的集合,可以用于高通量和高内涵筛选;
|
L6020
|
天然产物单体化合物库
|
|
19377 compounds
|
|
19377 种精选天然产物集合,结构多样,遍布多种动植物与微生物;
|
L6600
|
胃肠炎天然产物库
|
|
223 compounds
|
|
223种胃肠炎相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
|
L6700
|
抗癌天然产物库
|
|
1471 compounds
|
|
1471种已知活性天然产物的独特集合,是肿瘤药物开发、抗癌先导化合物筛选等领域的有力工具,可用于HTS和HCS。
|
DF4500
|
多样性核心库Part1
|
|
50000 compounds
|
|
绝大部分分子量<500,主要集中于250-450之间,方便后续的改造优化;
|
NY1000
|
天然产物衍生物库
|
|
4000 compounds
|
|
22个天然产物骨架,4000个天然产物衍生物;
|
VM1400
|
多样性核心库Part2
|
|
25920 compounds
|
|
分子量<500,主要集中于250-450之间,方便后续的改造优化;
|
L6120
|
黄酮类天然产物库
|
|
477 compounds
|
|
477种黄酮类天然产物的独特集合,可用于高通量筛选和高内涵筛选;
|
L6030
|
天然产物衍生物虚筛化合物库
|
|
135000 compounds
|
|
13.5万种天然产物衍生物,并且在持续增加中;
|
CL0097
|
Prostaglandin Receptor antagonist/agonist kit
|
|
|
|
|
CL0137
|
E1/E2/E3 Enzyme inhibitor kit
|
|
|
|
|
CL0113
|
ER stress pathway inhibitor/inducer kit
|
|
|
|
|
CL0067
|
Sodium Channel inhibitor kit
|
|
|
|
|
CL0066
|
P450 inhibitor kit
|
|
|
|
|
CL0103
|
mGluR agonist/antagonist/modulator kit
|
|
|
|
|
CL0126
|
Androgen Receptor antagonist kit
|
|
|
|
|
CL0139
|
ROS inhibitor kit
|
|
|
|
|
CL0132
|
DHFR inhibitor kit
|
|
|
|
|
L8710
|
铜死亡化合物库
|
|
411 compounds
|
|
TargetMol 铜死亡化合物库集合了 411 种与铜死亡相关的化合物,可以用于铜死亡机制及相关疾病研究
|
L1010
|
FDA上市及药典收录分子库
|
|
3158 compounds
|
|
3158个上市及药典分子集合,可用于高通量筛选和高内涵筛选;
|
CL0092
|
GSK-3 inhibitor kit
|
|
|
|
|