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Search Results for "Prostaglandin E3"

2

抑制剂 & 化合物

52

化合物库

1

仪器耗材

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Cat. No. Product Name
L8600 泛素化化合物库

214 compounds
214种泛素化相关的小分子,用于高通量和高内涵筛选;
L8500 HIF-1化合物库

1352 compounds
1352个HIF-1相关小分子的独特集合,可用于缺血性疾病、癌症等相关领域的药物开发和药理研究;
L4710 非甾体类抗炎化合物库

530 compounds
530种非甾体类的抗炎相关化合物,可用于高通量和高内涵筛选;
L9700 内质网应激化合物库

193 compounds
193个内质网应激相关的化合物集合,可用于高通量和高内涵筛选;
L2191 抗乳腺癌化合物库

1965 compounds
1965种与乳腺癌相关的化合物,可以用于抗乳腺癌药物研发和药理研究;
DC1140 特权片段注释化合物库-Ligand-gated

9028 compounds
DC1180 特权片段注释化合物库-Lyases

19530 compounds
DC1150 特权片段注释化合物库-GPCR Family B

9320 compounds
DC1170 特权片段注释化合物库-Oxidoreductases

8812 compounds
DC1190 特权片段注释化合物库-Sigma Opioid receptors

8724 compounds
DC1040 特权片段注释化合物库-Transferases

23001 compounds
DC1030 特权片段注释化合物库-Epigenetics

9196 compounds
DC1100 特权片段注释化合物库-GPCR Frizzled family

3434 compounds
DC1200 特权片段注释化合物库-Isomerases

1206 compounds
DC1050 特权片段注释化合物库-Voltage-gated

17952 compounds
DC1110 特权片段注释化合物库-Proteases

22863 compounds
DC1010 特权片段注释化合物库-GPCR Family A

24763 compounds
DC1000 特权片段注释化合物库

190000 compounds
The database contains 190k small molecules divided into 23 sub libraries each focused at a specific target. According to the recent studies, molecules acting on a particular target or class of targets usually have characteristic moieties (PF) containing key binding points responsible for activity, e.g. hinge-binding fragments. We used this principle for the statistical analysis of the reported active molecules and corresponding targets for the annotation of pre-filtered ChemDiv in house colle...
DC1130 特权片段注释化合物库-Phosphodiesterases

13154 compounds
DC1060 特权片段注释化合物库-Kinases

18350 compounds
DC1220 特权片段注释化合物库-Aminoacyltransferases

3008 compounds
DC1210 特权片段注释化合物库-Phosphatases

15354 compounds
DC1160 特权片段注释化合物库-Toll-like and Il-1 receptors

3536 compounds
DC1090 特权片段注释化合物库-Ligases

11828 compounds
DQ3000 Factor XIa化合物库

6500 compounds
DC1080 特权片段注释化合物库-GPCR Taste family

2675 compounds
DC1120 特权片段注释化合物库-Thrombopoietin receptors

4908 compounds
DC1230 特权片段注释化合物库-Beta amyloid A4 protein

4617 compounds
DC1070 特权片段注释化合物库-GPCR Family C

5071 compounds
DC1020 特权片段注释化合物库-Spiro Library

20563 compounds
L1380 转录因子库

704 compounds
704种转录因子靶向、结构新颖的化合物;
L6900 稀有天然产物库

284 compounds
284种稀有天然产物的集合,可以用于高通量和高内涵筛选;
L6020 天然产物单体化合物库

19377 compounds
19377 种精选天然产物集合,结构多样,遍布多种动植物与微生物;
L6600 胃肠炎天然产物库

223 compounds
223种胃肠炎相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
L6700 抗癌天然产物库

1471 compounds
1471种已知活性天然产物的独特集合,是肿瘤药物开发、抗癌先导化合物筛选等领域的有力工具,可用于HTS和HCS。
DF4500 多样性核心库Part1

50000 compounds
绝大部分分子量<500,主要集中于250-450之间,方便后续的改造优化;
NY1000 天然产物衍生物库

4000 compounds
22个天然产物骨架,4000个天然产物衍生物;
VM1400 多样性核心库Part2

25920 compounds
分子量<500,主要集中于250-450之间,方便后续的改造优化;
L6120 黄酮类天然产物库

477 compounds
477种黄酮类天然产物的独特集合,可用于高通量筛选和高内涵筛选;
L6030 天然产物衍生物虚筛化合物库

135000 compounds
13.5万种天然产物衍生物,并且在持续增加中;
CL0097 Prostaglandin Receptor antagonist/agonist kit

CL0137 E1/E2/E3 Enzyme inhibitor kit

CL0113 ER stress pathway inhibitor/inducer kit

CL0067 Sodium Channel inhibitor kit

CL0066 P450 inhibitor kit

CL0103 mGluR agonist/antagonist/modulator kit

CL0126 Androgen Receptor antagonist kit

CL0139 ROS inhibitor kit

CL0132 DHFR inhibitor kit

L8710 铜死亡化合物库

411 compounds
TargetMol 铜死亡化合物库集合了 411 种与铜死亡相关的化合物,可以用于铜死亡机制及相关疾病研究
L1010 FDA上市及药典收录分子库

3158 compounds
3158个上市及药典分子集合,可用于高通量筛选和高内涵筛选;
CL0092 GSK-3 inhibitor kit

化合物库

泛素化化合物库
L8600
Compounds: 214
HIF-1化合物库
L8500
Compounds: 1352
非甾体类抗炎化合物库
L4710
Compounds: 530
内质网应激化合物库
L9700
Compounds: 193
抗乳腺癌化合物库
L2191
Compounds: 1965
特权片段注释化合物库-Ligand-gated
DC1140
Compounds: 9028
特权片段注释化合物库-Lyases
DC1180
Compounds: 19530
特权片段注释化合物库-GPCR Family B
DC1150
Compounds: 9320
特权片段注释化合物库-Oxidoreductases
DC1170
Compounds: 8812
特权片段注释化合物库-Sigma Opioid receptors
DC1190
Compounds: 8724
特权片段注释化合物库-Transferases
DC1040
Compounds: 23001
特权片段注释化合物库-Epigenetics
DC1030
Compounds: 9196
特权片段注释化合物库-GPCR Frizzled family
DC1100
Compounds: 3434
特权片段注释化合物库-Isomerases
DC1200
Compounds: 1206
特权片段注释化合物库-Voltage-gated
DC1050
Compounds: 17952
特权片段注释化合物库-Proteases
DC1110
Compounds: 22863
特权片段注释化合物库-GPCR Family A
DC1010
Compounds: 24763
特权片段注释化合物库
DC1000
Compounds: 190000
特权片段注释化合物库-Phosphodiesterases
DC1130
Compounds: 13154
特权片段注释化合物库-Kinases
DC1060
Compounds: 18350
特权片段注释化合物库-Aminoacyltransferases
DC1220
Compounds: 3008
特权片段注释化合物库-Phosphatases
DC1210
Compounds: 15354
特权片段注释化合物库-Toll-like and Il-1 receptors
DC1160
Compounds: 3536
特权片段注释化合物库-Ligases
DC1090
Compounds: 11828
Factor XIa化合物库
DQ3000
Compounds: 6500
特权片段注释化合物库-GPCR Taste family
DC1080
Compounds: 2675
特权片段注释化合物库-Thrombopoietin receptors
DC1120
Compounds: 4908
特权片段注释化合物库-Beta amyloid A4 protein
DC1230
Compounds: 4617
特权片段注释化合物库-GPCR Family C
DC1070
Compounds: 5071
特权片段注释化合物库-Spiro Library
DC1020
Compounds: 20563
转录因子库
L1380
Compounds: 704
稀有天然产物库
L6900
Compounds: 284
天然产物单体化合物库
L6020
Compounds: 19377
胃肠炎天然产物库
L6600
Compounds: 223
抗癌天然产物库
L6700
Compounds: 1471
多样性核心库Part1
DF4500
Compounds: 50000
天然产物衍生物库
NY1000
Compounds: 4000
多样性核心库Part2
VM1400
Compounds: 25920
黄酮类天然产物库
L6120
Compounds: 477
天然产物衍生物虚筛化合物库
L6030
Compounds: 135000
Prostaglandin Receptor antagonist/agonist kit
CL0097
Compounds: 0
E1/E2/E3 Enzyme inhibitor kit
CL0137
Compounds: 0
ER stress pathway inhibitor/inducer kit
CL0113
Compounds: 0
Sodium Channel inhibitor kit
CL0067
Compounds: 0
P450 inhibitor kit
CL0066
Compounds: 0
mGluR agonist/antagonist/modulator kit
CL0103
Compounds: 0
Androgen Receptor antagonist kit
CL0126
Compounds: 0
ROS inhibitor kit
CL0139
Compounds: 0
DHFR inhibitor kit
CL0132
Compounds: 0
铜死亡化合物库
L8710
Compounds: 411
FDA上市及药典收录分子库
L1010
Compounds: 3158
GSK-3 inhibitor kit
CL0092
Compounds: 0
Cat. No. Product Name
EC6000 EP管低温冰浴盒

EP管低温冰浴盒,可简单替代冰浴槽;适用于实验室批量快速预冷生物样品,如蛋白、抗体、组织等。兼容0.2ml、1.5ml及2mlEP管和PCR八联排管。

仪器耗材

EP管低温冰浴盒
EC6000
Cat. No. Product Name Target Signaling Pathways
T38194 Prostaglandin E3

PGE3

Prostaglandin E3 (PGE3) is formed via the cyclooxygenase (COX) metabolism of eicosapentaenoic acid. [1] In human ocular tissue, it comprises 2.4% of the COX products formed. [1] When applied to the eyes of a rabbit, a 1 µg dose of PGE3 decreases intraocular pressure from 21 mmHg to about 17 mmHg.[2]
T41267 PROTAC(H-PGDS)-7

PROTAC(H-PGDS)-7 是一种有效的造血前列腺素 D 合酶 (H-PGDS)PROTAC 降解剂( DC50: 17.3 pM)。PROTAC(H-PGDS)-7由H-PGDS抑制剂(TFC-007)和小脑(CRBN) E3连接酶配体(pomalidomide)组成,具有很强的H-PGDS降解活性。

化合物

Prostaglandin E3
T38194
synonym: PGE3
Target:
PROTAC(H-PGDS)-7
T41267
synonym:
Target: