Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T11381 |
Pictilisib dimethanesulfonate
GDC-0941 2 MeSO3H salt,GDC-0941 dimethanesulfonate |
Apoptosis; DNA-PK; PI3K; mTOR; Autophagy | Apoptosis; Autophagy; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling |
Pictilisib dimethanesulfonate 是一种 PI3Kα/δ抑制剂,IC50值为 3 nM。对 p110β 和 p110γ的选择性分别为11倍和25倍。 |