t 1001

T1001 is an antagonist of hypoxia-inducible factor-2α subunit (HIF-2α) which displaces residue M252 from inside the HIF-2α PAS-B pocket toward the ARNT subunit to weaken heterodimerization.

Dicloxacillin Sodium hydrate 是一种青霉素类窄谱β内酰胺抗生素，可研究革兰氏阳性菌感染。

1-Acetyl-3-o-toluyl-5-fluorouracil is a potent antineoplastic agent.

1-Deazaadenosine is a potent Adenosine deaminase inhibitor (Ki: 0.66 μM). It exhibits anti-cancer activities in vitro and has the potential to be a chemotherapy agent for lymphoproliferative disorders.

P7C3-OMe 是促神经原性化合物，其 R-对映体活性远高于 S-对映体。可以用于研究神经精神疾病和神经退行性疾病。

1-(2-Quinoxalinyl)-1,2,3,4-butanetetrol是一种喹喔啉衍生物和内源性代谢物，可用于生物化学实验和药物合成研究。

1,3,5-Tricaffeoylquinic acid is a derivative of tricaffeoylquinic acid isolated from *Helichrysum populifolium* and exhibits anti-HIV activity.

(1α,1'S,4β)-Lanabecestat is a Beta site APP Cleaving Enzymel (BACE1) inhibitor, and has IC50s of 2.2 nM (TR-FRET assay) and 0.28 nM (sAPPp release assay), respectively.

Hydrocarbon chain derivative 1 has inhibitory activities against lipid synthesis.

1-Linoleoyl Glycerol (Monolinolein) 是脂肪酸甘油。

GL-1001 disodium tetrahydrate is an ACE2 inhibitor.

AT-1001 (Larazotide) 是一种具有口服活性的紧密连接调节剂及连蛋白 (Zonulin) 拮抗剂。它通过阻断 Zonulin 受体信号通路维持肠道上皮细胞间紧密连接的完整性，能有效降低乳糜泻及炎症性肠病模型中的肠道通透性。

Kahweol oleate is emi-syntetic derivative of kahweol, a natural product found in coffee beans. It exhibits a wide variety of biological activities, including inhibiting RANKL-induced osteoclast generation, inducing cell cycle arrest and apoptosis in oral squamous cell carcinoma cells, preventing aflatoxin B1 induced DNA adduct formation, and suppressing H2O2-induced DNA damage and oxidative stress.

BMS-1001 hydrochloride 是一种人 PD-L1/PD-1免疫检查点的抑制剂，具有口服活性且细胞毒性低。