gabapentin

Gabapentin (Neurontin) 是GABA 类似物，是一种抗癫痫药，可用于缓解神经性疼痛。

Gabapentin hydrochloride (Neurontin HCl) 是GABA 类似物，可用于缓解神经性疼痛。

Gabapentin enacarbil (XP-13512) 是抗惊厥和镇痛药物加巴喷丁的前药。Gabapentin enacarbil 提供持续剂量比例的 Gabapentin 暴露和可预测的生物利用度。

Gabapentin-d4 是 Gabapentin 的氘代化合物。Gabapentin 的 CAS 号为 60142-96-3。Gabapentin 是GABA类似物，是一种抗癫痫药，可用于缓解神经性疼痛。

Gabapentin-d6 Hydrochloride 是 Gabapentin Hydrochloride 的氘代化合物。Gabapentin Hydrochloride 的 CAS 号为 60142-95-2。Gabapentin hydrochloride 是GABA类似物，可用于缓解神经性疼痛。

Gabapentin-d6 是 Gabapentin 的氘代化合物。Gabapentin 的 CAS 号为 60142-96-3。Gabapentin 是GABA类似物，是一种抗癫痫药，可用于缓解神经性疼痛。

1-Carboxycyclohexaneacetic acid may be present as a potential impurity in commercial gabapentin, an antiepileptic drug. Furthermore, it serves as a precursor for synthesizing antagonists targeting the serotonin (5-HT) receptor subtype 5-HT2A.

Atagabalin, also known as PD 0200390, is a gabamimetic agent under development for the treatment for insomnia. Atagabalin is related to gabapentin, which similarly binds to the α2δ calcium channels (1 and 2). It was discontinued following unsatisfactory t

PD-217014 is a GABA analog. It inhibits (3)H-gabapentin binding to alpha(2)delta subunit of voltage-gated calcium channels in a concentration-dependent manner (K(i) = 18 nmol/l). PD-217014 possesses visceral analgesic activity.

H-D-Allo-Ile-OH能够抑制3[H] gabapentin结合电压依赖性L型钙通道，可用于研究神经和精神疾病。

Tiagabine-d6 is intended for use as an internal standard for the quantification of tiagabine by GC- or LC-MS. Tiagabine is an inhibitor of GABA transporter 1. It inhibits seizures induced by DMCM in mice. Tiagabine reduces allodynia in a rodent model of neuropathic pain when used at a dose of 72.8 µmol kg, and it acts synergistically with gabapentin to delay pain responses in mice in the hot plate test. Formulations containing tiagabine have been used as adjunctive therapies in the treatment of partial seizures.