AChR

An acetylcholine receptor (abbreviated AChR) is an integral membrane protein that responds to the binding of acetylcholine, a neurotransmitter.

Cat. No.	Product Name	CAS No.	Purity
T16563	Pozanicline 化合物 T16563	161417-03-4	98%
T16563	Pozanicline reverses nicotine withdrawal-induced cognitive deficits, may be an effective component of novel therapeutic strategies for nicotine addiction. Pozani...
TN1790	Isopteropodine 钩藤碱 E	5171-37-9	98%
TN1790	Isopteropodine (Uncarine E) 是从 Hamelia patens micropropagated 分离得到的一种异育亨宾型辛吲哚生物碱.具有抗菌活性，可刺激机体免疫系统。Isopteropodine 是 M1 型毒蕈碱乙酰胆碱 (muscarinic M1) 受体及 5-HT2 受体的正向调节剂...
TN3875	Dipterocarpol 化合物 TN3875	471-69-2	98%
TN3875	Dipterocarpol is a dammarane-type triterpenoid, as are the major bioactive compounds of ginseng. Dipterocarpol A shows moderate acetylcholinesterase inhibitory a...
TN2067	Picfeltarraegenin X 苦玄参苷X	1391826-61-1	98%
TN2067	Picfeltarraenin X shows stronger AChE inhibition than the known AChE inhibitor Tacrine.
T12525	Pozanicline dihydrochloride 化合物Pozanicline dihydrochloride	161416-61-1	98%
T12525	Pozanicline dihydrochloride (ABT-089 dihydrochloride) 是口服有效的烟碱型乙酰胆碱受体激动剂，与 [3H] 胱氨酸位点结合，Ki 为 16.7 nM，对 α4β2 nAChR 的选择性高于α7nAChR。
T12191	NBTGR 化合物 T12191	13153-27-0	98%
T12191	NBTGR is a potent nucleoside transport inhibitor(adenosine uptake ,Ki of 70 nM).
T19623	α-Muricholic acid 化合物 T19623	2393-58-0	98%
T19623	α-Muricholic acid is the most abundant primary bile acid in rodents.
TN2504	1,5-Dihydroxyxanthone 化合物 TN2504	14686-65-8	98%
TN2504	1,5-Dihydroxyxanthone exhibits the epidermal growth factor receptor (EGFR) -tyrosine kinase inhibitory activity, with the IC50 value of 90.34 nM. It may have ant...
TN4812	Pluviatolide 化合物 TN4812	28115-68-6	98%
TN4812	(-)-Pluviatolide can inhibit electrically-induced and acetylcholine-induced contraction in the isolated guinea-pig ileum.
T16417	Oxitropium Bromide 氧托溴铵	30286-75-0	98%
T16417	Oxitropium bromide is a mAChR antagonist. It is used as an anticholinergic bronchodilator drug for the treatment of asthma and chronic obstructive pulmonary dise...
T13256	UP202-56 化合物 T13256	163838-04-8	98%
T13256	UP202-56 is an adenosinergic agonist and is an adenosine analog.
TN4456	Lucidadiol 化合物 TN4456	252351-95-4	98%
TN4456	Lucidadiol exhibits butyrylcholinesterase-inhibitory activity at concentrations up to 200 uM, it also possesses inhibitory activity against acetylcholinesterase ...
T12868	Sch412348 化合物 T12868	377727-26-9	98%
T12868	Sch412348 is a potent competitive the human adenosine A2A receptor antagonist with Ki of 0.6 nM and has >1000-fold selectivity over all other adenosine receptors...
TN1409	Asimilobine 巴婆碱	6871-21-2	98%
TN1409	(-)-Asimilobine shows antioxidative, anti-acetylcholinesterase (AChE), anti-α±-glucosidase, anti-leishmanial and anti-fungal activities; it displays weak inhibit...
T10731	CDD0102 化合物 T10731	146422-58-4	98%
T10731	CDD0102 is a potent agonist of M1 Muscarinic receptor.
T12446	Phenserine 化合物 T12446	101246-66-6	98%
T12446	Phenserine is a derivative of Physostigmine and is annoncompetitive, long-acting and selective inhibitor of AChE.
T5476	MAChr-in-1 化合物mAChr-in-1	119391-56-9	98%
T5476	mAChR-IN-1 是一种毒蕈碱胆碱能受体拮抗剂，IC50为17 nM。
T13772	MHP 133 化合物 T13772	147340-43-0	98%
T13772	MHP 133 is a drug with multiple CNS targets(AChE with Ki of 69 μM).
T8868	4BP-TQS 化合物4BP-TQS	360791-49-7	99.99%
T8868	4BP-TQS 是 α7nAChR 变构激动剂。它利用变构跨膜位点激活 nAChRs。
T8552	PSEM 89S TFA 化合物PSEM 89S TFA	1336913-03-1	99.98%
T8552	PSEM 89S TFA 是一种脑渗透性和选择性离子通道激动剂，分别对 Q79G 和 L141F 具有正交选择性。