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Search Results for " azoline "

35

抑制剂 & 化合物

3

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T25982	Pramiconazole R-126638,R126638,R 126638,Azoline	Antifungal	Microbiology/Virology
	Pramiconazole (R126638) 是一种可口服的抗真菌化合物。Pramiconazole 是治疗皮肤癣菌和皮肤酵母菌感染的候选化合物，可用于治疗脂溢性皮炎。
T7477	Antazoline	Others	Others
	Antazoline 具有抗组胺和抗胆碱能作用。它用于治疗各种心律失常。
T21447	Tolazoline Priscol,妥拉苏林,Priscoline,Pridazole,Divascol,Vasimid,Benzalolin	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Tolazoline (Benzalolin) 是一种竞争性的α-肾上腺素受体拮抗剂。
T50083	12-oxo-N-[1-(propan-2-yl)piperidin-4-yl]-6H,7H,8H,9H,10H,12H-azepino[2,1-b]quinazoline-3-carboxamide	Others	Others
	12-oxo-N-[1-(propan-2-yl)piperidin-4-yl]-6H,7H,8H,9H,10H,12H-azepino[2,1-b]quinazoline-3-carboxamide 可用作分子结构单元，用于多种化合物的合成。
T0446	Naphazoline hydrochloride 盐酸萘甲唑啉,Albalon,Rhinantin,Naphazoline HCl	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Naphazoline hydrochloride (Naphazoline HCl) 是一种咪唑啉衍生物，是一种眼血管收缩剂。
T21445	Naphazoline AK-Con,Naphcon-a,Clear Eyes,All Clear,萘甲唑林	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Naphazoline (Naphcon-a) 是一种具有显着 α 肾上腺素能活性的拟交感神经化合物。萘甲唑啉可用作血管收缩剂，当应用于粘膜时可快速减少肿胀。
T9190	NAG-thiazoline GlcNAc-thiazoline,N-乙酰 - 葡糖胺基噻唑啉	Others	Others
	NAG-thiazoline (GlcNAc-thiazoline) 是一种 O-GlcNAcase 抑制剂，Ki 值为 180 nM。它对 V. campbellii 有效，MIC 值为 0.5 µM。
T71012	Nemazoline Free Base
	Nemazoline Free Base is a nasal decongestant. It has alpha 1-agonist/alpha 2-antagonist activity and was more effective and long-acting than oxymetazoline on canine nasal mucosa, in-vitro and in-vivo. Upon intranasal administration to dogs, the compound was devoid of systemic effects up to a concentration 1000 times that needed for local decongestant effect (1.65 micrograms, atomized from a 1 microgram mL-1 solution) suggesting limited mucosal absorption. After nasal administration to rats for 1...
T8615	ISOTHIAZOLINE 1,1-DIOXIDE 异噻唑烷 1,1-二氧化物,isothiazolidine 1,1-dioxide	Others	Others
	ISOTHIAZOLINE 1,1-DIOXIDE (isothiazolidine 1,1-dioxide) 是一种反应物，用于合成口服生物可利用的 hebatits B caspid 抑制剂，并用于制备隐花色素抑制剂作为抗糖尿病药物。
T0042	Xylometazoline hydrochloride 盐酸赛洛唑啉,Xylometazoline HCl	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Xylometazoline hydrochloride (Xylometazoline HCl) 是一种 α- 肾上腺素受体激动剂，是一种鼻血管收缩药。
T8513	Spastazoline	Others	Others
	Spastazoline 是spastin(一种微管切断AAA 蛋白) 的选择性抑制剂，对人 spastin 的IC50值为 99 nM。它不能影响重组人 VPS4 的 ATPase 活性。
T8565	N4-benzyl-N2-methylquinazoline-2,4-diamine hydrochloride	TRP/TRPV Channel	Membrane transporter/Ion channel
	N4-benzyl-N2-methylquinazoline-2,4-diamine hydrochloride 是 TRPC4 的抑制剂。
T72072	2-benzylsulfanyl-6-methoxy-4-methylquinazoline	ROS	Immunology/Inflammation
	2-benzylsulfanyl-6-methoxy-4-methylquinazoline 可作为TRPML 调节剂，可用于治疗与TRPML 活性相关的疾病，如溶酶体储存病、肌肉萎缩症、氧化应激或活性氧(ROS)相关疾病和衰老。
T0092	Antazoline hydrochloride 盐酸安他唑啉,Phenazocine HCl,Phenazoline hydrochloride,Antazoline HCl	Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Antazoline hydrochloride (Phenazoline hydrochloride) 是一种抗组胺药，可与组胺H1受体结合，阻断内源性组胺的作用。它也具有抗胆碱能特性，可缓解鼻塞，也可用作眼药水。
T65621	2-(Chloromethyl)-4-methylquinazoline
	2-(Chloromethyl)-4-methylquinazoline 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T65621，CAS号为 109113-72-6。
T14972	Cirazoline hydrochloride LD 3098 hydrochloride	Others	Others
	Cirazoline hydrochloride is a competitive full agonist of the α1A-adrenergic receptor (α1A-AR; Ki: 120 nM). It is a partial agonist at α1B-AR (Ki: 960 nM) and α1D-AR (Ki: 660 nM).
T36102	4-Chloro-6,7-bis(2-methoxyethoxy)quinazoline
	4-Chloro-6,7-bis(2-methoxyethoxy)quinazoline is a building block and synthetic intermediate.1,2,3,4,5It has been used as a precursor in the synthesis of receptor tyrosine kinase (RTK) inhibitors, dual RTK and histone deacetylase (HDAC) inhibitors, and anticancer compounds.1,2,3It is also a synthetic intermediate in the synthesis of EGFR inhibitors, including erlotinib , with antiproliferative activity.4,5
T70216	Clonazoline
	Clonazoline is a coronary vasodilator that is an imidazoline sympathomimetic, an alpha-adrenoreceptor agonist. It was used as a nasal decongestant and vasoconstrictor.
T0446L	Naphazoline nitrate Benil,Sanorin Spofa,Rhinon,Rinazina,Clera
	Naphazoline nitrate is an α1-Adrenergic receptor agonist. It also induces autophagy and necrotic cell death in erythroleukemia cells and inhibits erythroid differentiation. It used to treat congestion and ocular pathologies.
T65018	2-Chloro-4-amino-6,7-dimethoxyquinazoline
	2-Chloro-4-amino-6,7-dimethoxyquinazoline 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T65018，CAS号为 23680-84-4。
T126280	Carnequinazoline A
	Carnequinazoline A 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T126280，CAS号为 1175962-86-3。
T32656	Lerimazoline ST-71,Trimizoline,Trimazoline,ST 71,ST71
	Lerimazoline(Trimazoline, Trimizoline, ST-71) is used in the form of tramazoline hydrochloride in nasal decongestant preparations. It is used to inhibits the secretion of nasal mucus as an α-adrenergic receptor agonist.
T69334	Coumazoline
	Coumazoline is a particular alpha-adrenergic agonist.
T69341	Tramazoline hydrochloride
	Tramazoline hydrochloride is commonly used in nasal spray as a nasal decongestant by acting as an α-adrenergic receptor agonist that inhibits secretion of nasal mucus.
T64314	OxyMetazoline
	OxyMetazoline 是一种 α-肾上腺素受体 (α-adrenoceptor) 激动剂，能够作用于 α1A (IC50: 0.02 μM)、α1B (IC50: 0.25 μM)、α2A (IC50: 0.58 μM) 和 α2C (IC50: 0.13 μM)。OxyMetazoline 能够用于研究缓解鼻黏膜充血。
T69031	Cirazoline (free base)
	Cirazoline (free base) is a full agonist at the α1A adrenergic receptor, a partial agonist at both the α1B and α1D adrenergic receptors, and a nonselective antagonist to the α₂ adrenergic receptor. It is believed that this combination of properties could make cirazoline an effective vasoconstricting agent.
T64861	2,4-Dichloro-6,7-dimethoxyquinazoline
	2,4-Dichloro-6,7-dimethoxyquinazoline 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T64861，CAS号为 27631-29-4。
T66340	4,6-Dichloro-7-methoxyquinazoline
	4,6-Dichloro-7-methoxyquinazoline 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T66340，CAS号为 205584-69-6。
T19371	Indanazoline	Others	Others
	Indanazoline is characterized by a pronounced vasoconstrictive action.
T66020	4-Chloroquinazoline-6,7-diol
	4-Chloroquinazoline-6,7-diol 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T66020，CAS号为 1145671-36-8。
T21020	Antazoline phosphate
	Antazoline phosphate is an antihistamine with anticholinergic properties. Antazoline prevents the typical allergic symptoms on capillaries, mucous membranes, skin, and gastrointestinal and bronchial smooth muscles by antagonizing the histamine H1 receptor
T125912	Fumiquinazoline A
	Fumiquinazoline A 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T125912，CAS号为 140715-85-1。
T66391	(S)-N4-(3-Chloro-4-fluorophenyl)-7-((tetrahydrofuran-3-yl)oxy)quinazoline-4,6-diamine
	(S)-N4-(3-Chloro-4-fluorophenyl)-7-((tetrahydrofuran-3-yl)oxy)quinazoline-4,6-diamine 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T66391，CAS号为 314771-76-1。
T69670	Clonazoline HCl
	Clonazoline HCl is the salt form of Clonazoline, a coronary vasodilator that is an imidazoline sympathomimetic, an alpha-adrenoreceptor agonist. It was used as a nasal decongestant and vasoconstrictor.
T71600	Benazoline oxalate salt
	Benazoline oxalate salt is a pharmacological active compound that inhibits casein kinase Iε (CKIε) or CKIδ phosphorylation of the PER2 protein.

化合物

Cat.No: T25982

Synonym: R-126638,R126638,R 126638,Azoline

Target: Antifungal

Cat.No: T7477

Target: Others

Cat.No: T21447

Synonym: Priscol,妥拉苏林,Priscoline,Pridazole,Divascol,Vasimid,Benzalolin

Target: Adrenergic Receptor

12-oxo-N-[1-(propan-2-yl)piperidin-4-yl]-6H,7H,8H,9H,10H,12H-azepino[2,1-b]quinazoline-3-carboxamide

Cat.No: T50083

Target: Others

Naphazoline hydrochloride

Cat.No: T0446

Synonym: 盐酸萘甲唑啉,Albalon,Rhinantin,Naphazoline HCl

Target: Adrenergic Receptor

Cat.No: T21445

Synonym: AK-Con,Naphcon-a,Clear Eyes,All Clear,萘甲唑林

Target: Adrenergic Receptor

Cat.No: T9190

Synonym: GlcNAc-thiazoline,N-乙酰 - 葡糖胺基噻唑啉

Target: Others

Nemazoline Free Base

Cat.No: T71012

ISOTHIAZOLINE 1,1-DIOXIDE

Cat.No: T8615

Synonym: 异噻唑烷 1,1-二氧化物,isothiazolidine 1,1-dioxide

Target: Others

Xylometazoline hydrochloride

Cat.No: T0042

Synonym: 盐酸赛洛唑啉,Xylometazoline HCl

Target: Adrenergic Receptor

Cat.No: T8513

Target: Others

N4-benzyl-N2-methylquinazoline-2,4-diamine hydrochloride

Cat.No: T8565

Target: TRP/TRPV Channel

2-benzylsulfanyl-6-methoxy-4-methylquinazoline

Cat.No: T72072

Target: ROS

Antazoline hydrochloride

Cat.No: T0092

Synonym: 盐酸安他唑啉,Phenazocine HCl,Phenazoline hydrochloride,Antazoline HCl

Target: Histamine Receptor

2-(Chloromethyl)-4-methylquinazoline

Cat.No: T65621

Cirazoline hydrochloride

Cat.No: T14972

Synonym: LD 3098 hydrochloride

Target: Others

4-Chloro-6,7-bis(2-methoxyethoxy)quinazoline

Cat.No: T36102

Cat.No: T70216

Naphazoline nitrate

Cat.No: T0446L

Synonym: Benil,Sanorin Spofa,Rhinon,Rinazina,Clera

2-Chloro-4-amino-6,7-dimethoxyquinazoline

Cat.No: T65018

Carnequinazoline A

Cat.No: T126280

Cat.No: T32656

Synonym: ST-71,Trimizoline,Trimazoline,ST 71,ST71

Cat.No: T69334

Tramazoline hydrochloride

Cat.No: T69341

Cat.No: T64314

Cirazoline (free base)

Cat.No: T69031

2,4-Dichloro-6,7-dimethoxyquinazoline

Cat.No: T64861

4,6-Dichloro-7-methoxyquinazoline

Cat.No: T66340

Cat.No: T19371

Target: Others

4-Chloroquinazoline-6,7-diol

Cat.No: T66020

Antazoline phosphate

Cat.No: T21020

Fumiquinazoline A

Cat.No: T125912

(S)-N4-(3-Chloro-4-fluorophenyl)-7-((tetrahydrofuran-3-yl)oxy)quinazoline-4,6-diamine

Cat.No: T66391

Clonazoline HCl

Cat.No: T69670

Benazoline oxalate salt

Cat.No: T71600

Cat. No.	Product Name	Target	Signaling Pathways
TN7192	7-Bromoquinazoline-2,4(1H,3H)-Dione 7-Bromo-2,4(1H,3H)-quinazolinedione,7-溴喹唑啉-(2,4)二酮,7-Bromo-1H-quinazoline-2,4-dione,7-bromoquinazoline-2,4-diol	Others	Others
	7-Bromoquinazoline-2,4(1H,3H)-Dione (7-Bromo-2,4(1H,3H)-quinazolinedione) 是一种海洋来源的天然产物，发现于 Pyura sacciformis。
T1680	Tolazoline hydrochloride Imidaline hydrochloride,苯甲唑啉盐酸盐,Imidaline (hydrochloride),Benzidazol hydrochloride,Tolazoline HCl,NSC35110 (hydrochloride)	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Tolazoline hydrochloride (NSC35110(hydrochloride)) 是一种 α 肾上腺素受体抑制剂。
T37712	Fumiquinazoline D
	Fumiquinazoline D is a fungal metabolite originally isolated from A. fumigatus that has activity against Gram-positive and Gram-negative bacteria (MICs = 8-16 μg/ml) as well as F. solani and C. albicans fungi (MICs = 32 and 64 μg/ml, respectively).

天然产物

7-Bromoquinazoline-2,4(1H,3H)-Dione

Cat.No: TN7192

Synonym: 7-Bromo-2,4(1H,3H)-quinazolinedione,7-溴喹唑啉-(2,4)二酮,7-Bromo-1H-quinazoline-2,4-dione,7-bromoquinazoline-2,4-diol

Target: Others

Tolazoline hydrochloride

Cat.No: T1680

Synonym: Imidaline hydrochloride,苯甲唑啉盐酸盐,Imidaline (hydrochloride),Benzidazol hydrochloride,Tolazoline HCl,NSC35110 (hydrochloride)

Target: Adrenergic Receptor

Fumiquinazoline D

Cat.No: T37712

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