Cat. No. | Product Name | CAS No. | Purity | Chemical Structure |
---|---|---|---|---|
T13245 | UCSF924
化合物 T13245
|
1434515-70-4 | 98% |
|
UCSF924 is a potent and specific agonist of dopamine D4 receptor (DRD4) partial (EC50: 4.2 nM, Ki: 3 nM). | ||||
T12288 | Odapipam
化合物 T12288
|
131796-63-9 | 98% |
|
Odapipam is a selective and high affinity antagonist of benzazepine dopamine D1 receptor (Kd of 0.18 nM). | ||||
T1476L | Pramipexole dihydrochloride
盐酸普拉克索
|
104632-25-9 | 98% |
|
Pramipexole dihydrochloride could be used to treat Parkinson disease. | ||||
T22921 | LE 300
化合物LE 300
|
274694-98-3 | 98% |
|
LE 300 是选择性多巴胺 D1 样受体拮抗剂,作用于人多巴胺 D1 和 D5 受体的Kis 分别为 1.9 nM 和 7.5 nM。在大鼠尾动脉实验中,它作用于5-HT2A 受体的pA2 为 8.32。 | ||||
T10611 | Brexpiprazole S-oxide D8
化合物 T10611
|
2748605-29-8 | 98% |
|
Brexpiprazole S-oxide D8 (DM-3411 D8) is a deuterium labeled Brexpiprazole S-oxide. Brexpiprazole S-oxide is a main metabolite of Brexpiprazole. Brexpiprazole is... | ||||
T21360 | Asenapine
阿塞那平
|
65576-45-6 | 98% |
|
Asenapine (Org 5222) 是5-HT受体、肾上腺素受体、多巴胺受体和组胺受体拮抗剂,具有抗精神病作用,可用于治疗精神分裂症和与双相 1 型障碍相关的躁狂或混合发作。 | ||||
TQ0175 | Dexpramipexole
右旋普拉克索
|
104632-28-2 | 98% |
|
Dexpramipexole (KNS-760704, R-(+)-Pramipexole) is a neuroprotective agent and weak non-ergoline dopamine agonist. | ||||
TQ0140 | Sumanirole maleate
马来酸Sumanirole
|
179386-44-8 | 98% |
|
Sumanirole maleate (U-95666E) is a highly selective full agonist of the D2 receptor (ED50: 46 nM). | ||||
T7341 | Diclofensine
(+/-)-双氮奋兴
|
67165-56-4 | 98% |
|
Diclofensine (Ro 8-4650) 是一种高效单胺再摄取抑制剂,在大鼠脑突触体中能够阻断多巴胺 (IC50=0.74 nM)、去甲肾上腺素 (IC50=2.3 nM) 和 5-羟色胺 (IC50=3.7 nM)。 | ||||
T9540 | Phenelzine
苯乙肼
|
51-71-8 | 98% |
|
Phenelzine 是一种抗抑郁和躁狂症药物,是一种单胺氧化酶抑制剂。其抗抑郁作用与烟酰胺相似。可减少脑内儿茶酚胺(去甲肾上腺素、多巴胺、5-羟色胺)的降解,增加儿茶酚胺的含量。 ,并起到抗抑郁作用。对内源性抑郁症疗效较好,对外源性和反应性抑郁症疗效较差。 | ||||
T11799L | L-745870
化合物 T11799L
|
158985-00-3 | 98% |
|
L-745870 is a high-affinity and selective human dopamine D4 receptor antagonist (Ki: 0.43 nM). L-745870 has excellent brain penetration. It considerably weaker D... | ||||
T12476 | Pimozide-d4
化合物 T12476
|
1803193-57-8 | 98% |
|
Pimozide D4 is a deuterium labeled Pimozide. | ||||
T13463L | Dihydrexidine
化合物 T13463L
|
123039-93-0 | 98% |
|
Dihydrexidine is a full efficacy D1-like dopamine receptor (D1/D5) agonist (IC50: 10 nM for D1 receptor). It also shows potent antiparkinsonian activity. | ||||
T13898 | SPD-473 citrate
化合物 T13898
|
161190-26-7 | 98% |
|
SPD-473 citrate is an inhibitior of serotonin/dopamine/norepinephrine reuptake. | ||||
T10908 | CY 208-243
化合物 T10908
|
100999-26-6 | 98% |
|
CY 208-243 is a selective dopamine D1 receptor agonist with anti-Parkinson disease activity. | ||||
T12865 | SCH-23390 maleate
化合物SCH-23390 maleate
|
87134-87-0 | 98% |
|
SCH-23390 maleate (R-(+)-SCH-23390 maleate) 是多巴胺D1样受体选择性拮抗剂,与D1和D5受体结合的Ki 分别为 0.2 nM 和 0.3 nM。它也是人5-HT2C 受体激动剂,Ki 为 9.3 nM。它与5-HT2和5-HT1C 受体具有高亲和力。它还抑制 G 蛋白偶联的内向... | ||||
T13652 | Dicarbine
化合物 T13652
|
17411-19-7 | 98% |
|
Double carbene can be used for the study of schizophrenia and alcoholism. It can block dopamine receptors in various parts of the brain and prevent the reduction... | ||||
T68023 | Tolnapersine
托那哌嗪
|
70312-00-4 | 98% |
|
Tolnapersine 是混合多巴胺激动剂和α-肾上腺素受体拮抗剂。 | ||||
T10681 | Cariprazine D6
化合物 T10681
|
1308278-67-2 | 98% |
|
Cariprazine D6 (RGH-188 D6) is a deuterium-labeled Cariprazine. Cariprazine is an antipsychotic agent (D3 receptors, Ki: 0.085 nM; D2 receptors, Ki: 0.49 nM). | ||||
TN1424 | Bacopaside X
假马齿苋皂苷 VII
|
94443-88-6 | 98% |
|
Bacopaside X (9.06 μM) showed binding affinity towards the D1 receptor. |