Cat. No. | Product Name | CAS No. | Purity | Chemical Structure |
---|---|---|---|---|
T11620 | IDO-IN-6
化合物 T11620
|
1402837-76-6 | 98% |
|
IDO-IN-6 is an indoleamine 2,3-dioxygenase (IDO) inhibitor. | ||||
T11626 | IACS-8968
化合物 T11626
|
2144425-14-7 | 98% |
|
IACS-8968 is a dual IDO and TDO inhibitor (pIC50s: 6.43 for IDO and <5 for TDO). | ||||
T8214 | Kushenol E
苦参醇E
|
99119-72-9 | 98% |
|
Kushenol E (Flemiphilippinin D) 是一种分离自Sophora flavescens 中的类黄酮,是一种IDO1的非竞争性抑制剂,其IC50=7.7 µM,Ki=为 9.5 µM,具有抗肿瘤特性。 | ||||
T11621 | IDO-IN-8
化合物 T11621
|
1402837-77-7 | 98% |
|
IDO-IN-8 is an indoleamine 2,3-dioxygenase (IDO) inhibitor (IC50: 1-10 μM). | ||||
T11619 | IDO-IN-5
化合物 T11619
|
1402837-79-9 | 98% |
|
IDO-IN-5 is an indoleamine 2,3-dioxygenase (IDO) inhibitor (IC50: 1-10 μM). | ||||
T11614 | IDO-IN-11
化合物 T11614
|
1888378-32-2 | 98% |
|
IDO-IN-11 is an indoleamine-2,3-dioxygenase (IDO) inhibitor with IC50s of 0.18 μM (Kinase) and 0.014 μM (Hela Cell). | ||||
T11627 | IACS-8968 R-enantiomer
化合物 T11627
|
2239305-67-8 | 98% |
|
IACS-8968 R-enantiomer is the R-enantiomer of IACS-8968. IACS-8968 is a dual IDO and TDO inhibitor (pIC50s: 6.43 for IDO and <5 for TDO). | ||||
T11617 | IDO-IN-3
化合物 T11617
|
2070018-30-1 | 98% |
|
IDO-IN-3 is a potent indoleamine 2,3-dioxygenase (IDO) inhibitor (IC50: 290 nM). | ||||
T11622 | IDO-IN-9
化合物 T11622
|
1888378-12-8 | 98% |
|
IDO-IN-9 is an indoleamine-2,3-dioxygenase (IDO) inhibitor with IC50s of 0.011 μM (Kinase) and 0.0018 μM (Hela Cell). | ||||
T11624 | IDO1-IN-2
化合物 T11624
|
2346614-58-0 | 98% |
|
IDO1-IN-2 is a potent and selective IDO1 inhibitor with IC50s of 81 nM, 59 nM (mouse), and 28 nM (rat), respectively. It has anti-cancer activity. | ||||
T11628 | IACS-8968 S-enantiomer
化合物 T11628
|
2239305-70-3 | 98% |
|
IACS-8968 S-enantiomer is the S-enantiomer of IACS-8968. IACS-8968 is a dual IDO and TDO inhibitor (pIC50s: 6.43 for IDO and <5 for TDO). | ||||
T4307 | PF-06840003
化合物PF06840003
|
198474-05-4 | 99.89% |
|
PF-06840003 (EOS200271) 是口服具有活力的、选择性的IDO-1抑制剂,抑制 hIDO-1, dIDO-1和 mIDO-1 的IC50分别为 0.41 μM, 0.59 μM,和 1.5 μM。 | ||||
T4532 | Linrodostat
化合物Linrodostat
|
1923833-60-6 | 99.84% |
|
Linrodostat (BMS-986205) 是选择性的、不可逆的吲哚胺 2,3-双加氧酶 1(IDO1) 抑制剂,能够有效抑制 IDO1-HEK293 细胞,其IC50=1.1 nM。它在晚期癌症中具有良好的药理特性。 | ||||
T6407 | β-Lapachone
化合物Beta-Lapachone
|
4707-32-8 | 99.72% |
|
β-Lapachone (ARQ-501) 是一种萘醌类天然产物,是拓扑异构酶 I 抑制剂,通过抑制细胞周期进程来诱导细胞凋亡。 | ||||
T20513 | IDO1-IN-1
2-肼基苯并噻唑
|
615-21-4 | 99.61% |
|
IDO1-IN-1 (2 HzBTZ) 是一种吲哚胺 2,3-双加氧酶 1 (IDO1) 抑制剂。 | ||||
T11615 | IDO-IN-12
化合物IDO-IN-12
|
1888341-29-4 | 99.61% |
|
IDO-IN-12 是吲哚胺 2,3-双加氧酶抑制剂。 | ||||
T11616 | IDO-IN-13
化合物IDO-IN-13
|
2291164-02-6 | 99.57% |
|
IDO-IN-13 (GS-4361) 是 indoleamine 2,3-dioxygenase 1 抑制剂,EC50=17 nM,摘自专利 WO2019040102A1,example 43。 | ||||
T10199 | GNF-PF-3777
化合物GNF-PF-3777
|
77603-42-0 | 99.47% |
|
GNF-PF-3777 (8-Nitrotryptanthrin) 是人吲哚胺2,3-双加氧酶 2 (hIDO2) 抑制剂,能够降低IDO2活性,Ki=为 0.97 μM。 | ||||
T9164 | BMS-986242
化合物BMS-986242
|
1923844-48-7 | 98.25% |
|
BMS-986242 是具有口服具有活力、强效的、选择性的 indoleamine-2,3-dioxygenase 1 抑制剂,可用于研究癌症。 | ||||
T3548 | Epacadostat
艾卡哚司他
|
1204669-58-8 | 98.08% |
|
Epacadostat (INCB 024360) 是选择性的IDO1抑制剂,IC50=71.8 nM。 |