Histamine Receptor

The histamine receptors are a class of G protein–coupled receptors which bind histamine as their primary endogenous ligand.

Cat. No.	Product Name	CAS No.	Purity
T10575	BMY-25271 化合物 T10575	78441-82-4	98%
T10575	BMY-25271 is an antagonist of histamine H2 receptor.
T11532	H4R antagonist 1 化合物 T11532	1429375-54-1	98%
T11532	H4R antagonist 1 is a highly selective histamine H4 receptor (H4R) antagonist (IC50: 27 nM). H4R antagonist 1 does not show any noticeable binding affinity to ot...
T19234	Cetirizine D8 dihydrochloride 盐酸西替利嗪 D8	2070015-04-0	98%
T19234	Cetirizine D8 dihydrochloride is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagoni...
TN5279	Zeorin 化合物 TN5279	22570-53-2	98%
TN5279	Zeorin shows strong inhibition activity against bacteria and fungi. It markedly exhibits inhibitory activity on histamine release from mast cell induced by DNP24...
T12756	ROS 234 dioxalate 化合物 T12756	1781941-93-2	98%
T12756	ROS 234 dioxalate is a potent antagonist of H3(pKB of 9.46 for Guinea-pig ileum H3-receptor)
T13040	SUN 1334H 化合物 T13040	607736-84-5	98%
T13040	SUN 1334H is a potent, orally active, highly selective antagonist of H1 receptor(Ki of 9.7 nM).
T11531	H3R-IN-1 Hydrochloride 化合物 T11531	2319790-07-1	98%
T11531	H3R-IN-1 Hydrochloride 是一种有效的组胺H3受体 (H3R) 的反向激动剂。
T21360	Asenapine 阿塞那平	65576-45-6	98%
T21360	Asenapine (Org 5222) 是5-HT受体、肾上腺素受体、多巴胺受体和组胺受体拮抗剂，具有抗精神病作用，可用于治疗精神分裂症和与双相 1 型障碍相关的躁狂或混合发作。
TN1913	Marmin 化合物Marmin	14957-38-1	98%
TN1913	Marmin have anti-ulcer effects, which are ascribed primarily to the maintenance of the mucosal barrier integrity and inhibition of gastric motor activity and sec...
T10769	Cetirizine D4 化合物 T10769	1219803-84-5	98%
T10769	Cetirizine D4 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
TN3062	4'-O-Methylnyasol 化合物 TN3062	79004-25-4	98%
TN3062	4'-O-Methylnyasol may have potential to be developed as medicines for the treatment of allergies by inhibiting the activation of mast cells.
T19604	WZ4141 化合物 T19604	1222776-76-2	98%
T19604	WZ4141 is an intermediate in compound synthesis.
T12054	MK-0249 化合物 T12054	862309-06-6	98%
T12054	MK-0249 is a potent antagonist of histamine H3 receptor (human H3, Ki : 1.7 nM).
T11324	FRG8701 化合物 T11324	108498-50-6	98%
T11324	FRG8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to 0.43 μM.
TN2895	3,5-Dicaffeoyl-epi-quinic acid 化合物 TN2895	879305-14-3	98%
TN2895	3,5-Dicaffeoyl-epi-quinic acid shows anti-inflammatory activity, it may improve mast cell-mediated inflammatory diseases.
T10911	H3 receptor antagonist 1 化合物 T10911	935840-13-4	98%
T10911	H3 receptor antagonist 1 is used in the study of neurological diseases, histamine H3 receptor antagonist.
T15565	Imetit dihydrobromide 化合物 T15565	32385-58-3	98%
T15565	Imetit dihydrobromide is a high affinity and effective agonist of histamine H3 and H4 receptors (Ki: 0.3 and 2.7 nM). Imetit mimics the histamine effect in trigg...
T4099	S 38093 化合物S38093	862896-30-8	99.98%
T4099	S 38093 是一种可透过大脑的，可口服的组胺 H3 受体拮抗剂，对大小鼠和人的 H3 受体具有不同的亲和力，Ki 值分别为 8.8、1.44 和 1.2 µM。
T1619	Trazodone hydrochloride 盐酸曲唑酮	25332-39-2	99.98%
T1619	Trazodone hydrochloride (Trazodone HCl) 是5 羟色胺受体拮抗剂和重吸收抑制剂，用作抗抑郁药，可治疗失眠和焦虑。
T4499	Mequitazine 美喹他嗪	29216-28-2	99.95%
T4499	Mequitazine (Virginan) 是一种有效的、非镇静剂和长效组胺 H1 拮抗剂。