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Estrogen/progestogen Receptor

Estrogen/progestogen Receptor

Estrogen receptors are a group of proteins found inside cells. They are receptors that are activated by the hormone estrogen (17β-estradiol). Two classes of estrogen receptor exist: ER, which is a member of the nuclear hormone family of intracellular receptors, and GPER (GPR30), which is a member of the rhodopsin-like family of G protein-coupled receptors.The progesterone receptor (PR), also known as NR3C3 or nuclear receptor subfamily 3, group C, member 3, is a protein found inside cells. It is activated by the steroid hormone progesterone.
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Cat. No. Product Name CAS No. Purity Chemical Structure
T0171 Norethynodrel
异炔诺酮
68-23-5
Norethynodrel (Lynestrol) 是一种合成的孕激素,其作用和用途类似于孕酮。它已被用于治疗功能性子宫出血和子宫内膜异位症。它作为避孕药,通常与 MESTRANOL 联合使用。
T77724 OBHSA
化合物OBHSA
1404508-27-5 98%
OBHSA(Oxabicycloheptane sulfonamide) 是一种新型选择性雌激素受体降解剂 (SERD),可用于研究乳腺癌。
TN2045 Pelargonidin-3-O-glucoside chloride
天竺葵素-3-氯化葡萄糖苷
18466-51-8 98%
Pelargonidin-3-O-glucopyranoside is the glucoside of Pelargonidin, an potential antidiabetic agent. Pelargonidin-3-O-glucopyranoside has antioxidant, anti-inflam...
TQ0149 Prinaberel
普林贝瑞
524684-52-4 98%
Prinaberel (ERB-041) is an effective and selective ERβ agonist and >200-fold selective for ERβ.
TN2288 Uralenol
化合物 TN2288
139163-15-8 98%
Uralenol significantly shows the inhibitory activities against the PTP1B enzyme; it also shows inhibitory activities on mushroom tyrosinase using l-tyrosine as s...
T6404 Bazedoxifene hydrochloride
盐酸巴多昔芬
198480-56-7 98%
Bazedoxifene hydrochloride (TSE-424) 是一种 IL-6/GP130蛋白相互作用抑制剂,可用于胰腺癌的研究。它也是一种有口服活性的,能透过血脑屏障的,非甾体、选择性的雌激素受体调节剂 (SERM),对 ERα 和 ERβ 作用的 IC50值分别为 26 nM 和 99 nM,可用于研究骨...
T12278 NXT629
化合物 T12278
1454925-59-7 98%
NXT629 is a selective and competitive antagonist of PPAR-α(human PPARα with an IC50 of 77 nM).
TN2200 Segetalin A
王不留行环肽 A
161875-97-4 98%
Segetalin A has estrogen-like activity.
TN3802 Dehydrodiconiferyl alcohol
去氢二松柏醇
4263-87-0 98%
Dehydrodiconiferyl alcohol (DHCA) 是一种从葫芦中分离出来的木脂素,通过作为雌激素受体激动剂抑制破骨细胞分化和卵巢切除术诱导的骨质流失。
T6827 Endoxifen Z-isomer hydrochloride
Z-因多昔芬盐酸盐
1032008-74-4 98%
Endoxifen Z-isomer hydrochloride (Endoxifen HCl) 是Tamoxifen 最重要的代谢产物, 在表达ERα的乳腺癌细胞中发挥抗雌激素作用, Endoxifen HCl 以浓度依赖的方式抑制hERG, IC50值为1.6μM。
T5351 PU-WS13
化合物PU-WS13
1454619-14-7 98%
T21897 Methylpiperidino pyrazole
甲基哌啶基吡唑
289726-02-9 98%
Methylpiperidino pyrazole 是一种 ERα 抑制剂,可阻止 BPS 诱导的 Rb 磷酸化和细胞周期进程。
TN1690 Glabrene
光甘草素
60008-03-9 98%
Glabrene, Liquiritin apioside, neolicuroside, and 18α²-glycyrrhetic acid are the predominant phenolic derivatives partitioning at the interface and most likely t...
TQ0163 Sagittatoside A
箭藿苷 A
118525-35-2 98%
Sagittatoside A selectively activates estrogen response element (ERE)-luciferase activity via ERα.
T16351 NSC16168
化合物 T16351
6837-93-0 98%
NSC16168 inhibits DNA repair and potentiates CDDP efficacy in cancer. NSC16168 is a specific ERCC1-XPF inhibitor (IC50: 0.42 μM).
T12329 Ospemifene D4
化合物 T12329
T12329 98%
Ospemifene D4 is a deuterium labeled Ospemifene. Ospemifene is a selective and orally active modulator of estrogen receptor.
T12312 OP-1074
化合物 T12312
1443752-76-8 98%
OP-1074 is a pure antiestrogen and a selective degrader of ER, shows specific antiestrogenic activity for ERα and ERβ.
TN1679 Genistein 7,4'-di-O-β-D-glucoside
染料木素-7,4'-二-O-Β-D-葡萄糖苷
36190-98-4 98%
Genistein 7,4'-di-O-beta-D-glucopyranoside shows significant estrogenic proliferative effect in MCF-7 cell in sub-cytotoxic concentration range.
T11222 ERB-196
化合物 T11222
550997-55-2 98%
Erb-196 is an estrogen receptor-receptor agonist with non-steroidal selectivity.
T11231 ERRγ Inverse Agonist 1
化合物 T11231
2316832-86-5 98%
ERRγ Inverse Agonist 1 (Compound 12) 是有效的、选择性的、口服生物可利用的雌激素相关受体 γ (ERRγ)的反向激动剂,IC50值为 40 nM。
Norethynodrel
T0171
Norethynodrel (Lynestrol) 是一种合成的孕激素,其作用和用途类似于孕酮。它已被用于治疗功能性子宫出血和子宫内膜异位症。它作为避孕药,通常与 MESTRANOL 联合使用。
OBHSA
T77724
OBHSA(Oxabicycloheptane sulfonamide) 是一种新型选择性雌激素受体降解剂 (SERD),可用于研究乳腺癌。
Pelargonidin-3-O-glucoside chloride
TN2045
Pelargonidin-3-O-glucopyranoside is the glucoside of Pelargonidin, an potential antidiabetic agent. Pelargonidin-3-O-glucopyranoside has antioxidant, anti-inflam...
Prinaberel
TQ0149
Prinaberel (ERB-041) is an effective and selective ERβ agonist and >200-fold selective for ERβ.
Uralenol
TN2288
Uralenol significantly shows the inhibitory activities against the PTP1B enzyme; it also shows inhibitory activities on mushroom tyrosinase using l-tyrosine as s...
Bazedoxifene hydrochloride
T6404
Bazedoxifene hydrochloride (TSE-424) 是一种 IL-6/GP130蛋白相互作用抑制剂,可用于胰腺癌的研究。它也是一种有口服活性的,能透过血脑屏障的,非甾体、选择性的雌激素受体调节剂 (SERM),对 ERα 和 ERβ 作用的 IC50值分别为 26 nM 和 99 nM,可用于研究骨...
NXT629
T12278
NXT629 is a selective and competitive antagonist of PPAR-α(human PPARα with an IC50 of 77 nM).
Segetalin A
TN2200
Segetalin A has estrogen-like activity.
Dehydrodiconiferyl alcohol
TN3802
Dehydrodiconiferyl alcohol (DHCA) 是一种从葫芦中分离出来的木脂素,通过作为雌激素受体激动剂抑制破骨细胞分化和卵巢切除术诱导的骨质流失。
Endoxifen Z-isomer hydrochloride
T6827
Endoxifen Z-isomer hydrochloride (Endoxifen HCl) 是Tamoxifen 最重要的代谢产物, 在表达ERα的乳腺癌细胞中发挥抗雌激素作用, Endoxifen HCl 以浓度依赖的方式抑制hERG, IC50值为1.6μM。
PU-WS13
T5351
Methylpiperidino pyrazole
T21897
Methylpiperidino pyrazole 是一种 ERα 抑制剂,可阻止 BPS 诱导的 Rb 磷酸化和细胞周期进程。
Glabrene
TN1690
Glabrene, Liquiritin apioside, neolicuroside, and 18α²-glycyrrhetic acid are the predominant phenolic derivatives partitioning at the interface and most likely t...
Sagittatoside A
TQ0163
Sagittatoside A selectively activates estrogen response element (ERE)-luciferase activity via ERα.
NSC16168
T16351
NSC16168 inhibits DNA repair and potentiates CDDP efficacy in cancer. NSC16168 is a specific ERCC1-XPF inhibitor (IC50: 0.42 μM).
Ospemifene D4
T12329
Ospemifene D4 is a deuterium labeled Ospemifene. Ospemifene is a selective and orally active modulator of estrogen receptor.
OP-1074
T12312
OP-1074 is a pure antiestrogen and a selective degrader of ER, shows specific antiestrogenic activity for ERα and ERβ.
Genistein 7,4'-di-O-β-D-glucoside
TN1679
Genistein 7,4'-di-O-beta-D-glucopyranoside shows significant estrogenic proliferative effect in MCF-7 cell in sub-cytotoxic concentration range.
ERB-196
T11222
Erb-196 is an estrogen receptor-receptor agonist with non-steroidal selectivity.
ERRγ Inverse Agonist 1
T11231
ERRγ Inverse Agonist 1 (Compound 12) 是有效的、选择性的、口服生物可利用的雌激素相关受体 γ (ERRγ)的反向激动剂,IC50值为 40 nM。
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