Cat. No. | Product Name | CAS No. | Purity | Chemical Structure |
---|---|---|---|---|
T0171 | Norethynodrel
异炔诺酮
|
68-23-5 |
|
|
Norethynodrel (Lynestrol) 是一种合成的孕激素,其作用和用途类似于孕酮。它已被用于治疗功能性子宫出血和子宫内膜异位症。它作为避孕药,通常与 MESTRANOL 联合使用。 | ||||
T77724 | OBHSA
化合物OBHSA
|
1404508-27-5 | 98% |
|
OBHSA(Oxabicycloheptane sulfonamide) 是一种新型选择性雌激素受体降解剂 (SERD),可用于研究乳腺癌。 | ||||
TN2045 | Pelargonidin-3-O-glucoside chloride
天竺葵素-3-氯化葡萄糖苷
|
18466-51-8 | 98% |
|
Pelargonidin-3-O-glucopyranoside is the glucoside of Pelargonidin, an potential antidiabetic agent. Pelargonidin-3-O-glucopyranoside has antioxidant, anti-inflam... | ||||
TQ0149 | Prinaberel
普林贝瑞
|
524684-52-4 | 98% |
|
Prinaberel (ERB-041) is an effective and selective ERβ agonist and >200-fold selective for ERβ. | ||||
TN2288 | Uralenol
化合物 TN2288
|
139163-15-8 | 98% |
|
Uralenol significantly shows the inhibitory activities against the PTP1B enzyme; it also shows inhibitory activities on mushroom tyrosinase using l-tyrosine as s... | ||||
T6404 | Bazedoxifene hydrochloride
盐酸巴多昔芬
|
198480-56-7 | 98% |
|
Bazedoxifene hydrochloride (TSE-424) 是一种 IL-6/GP130蛋白相互作用抑制剂,可用于胰腺癌的研究。它也是一种有口服活性的,能透过血脑屏障的,非甾体、选择性的雌激素受体调节剂 (SERM),对 ERα 和 ERβ 作用的 IC50值分别为 26 nM 和 99 nM,可用于研究骨... | ||||
T12278 | NXT629
化合物 T12278
|
1454925-59-7 | 98% |
|
NXT629 is a selective and competitive antagonist of PPAR-α(human PPARα with an IC50 of 77 nM). | ||||
TN2200 | Segetalin A
王不留行环肽 A
|
161875-97-4 | 98% |
|
Segetalin A has estrogen-like activity. | ||||
TN3802 | Dehydrodiconiferyl alcohol
去氢二松柏醇
|
4263-87-0 | 98% |
|
Dehydrodiconiferyl alcohol (DHCA) 是一种从葫芦中分离出来的木脂素,通过作为雌激素受体激动剂抑制破骨细胞分化和卵巢切除术诱导的骨质流失。 | ||||
T6827 | Endoxifen Z-isomer hydrochloride
Z-因多昔芬盐酸盐
|
1032008-74-4 | 98% |
|
Endoxifen Z-isomer hydrochloride (Endoxifen HCl) 是Tamoxifen 最重要的代谢产物, 在表达ERα的乳腺癌细胞中发挥抗雌激素作用, Endoxifen HCl 以浓度依赖的方式抑制hERG, IC50值为1.6μM。 | ||||
T5351 | PU-WS13
化合物PU-WS13
|
1454619-14-7 | 98% |
|
T21897 | Methylpiperidino pyrazole
甲基哌啶基吡唑
|
289726-02-9 | 98% |
|
Methylpiperidino pyrazole 是一种 ERα 抑制剂,可阻止 BPS 诱导的 Rb 磷酸化和细胞周期进程。 | ||||
TN1690 | Glabrene
光甘草素
|
60008-03-9 | 98% |
|
Glabrene, Liquiritin apioside, neolicuroside, and 18α²-glycyrrhetic acid are the predominant phenolic derivatives partitioning at the interface and most likely t... | ||||
TQ0163 | Sagittatoside A
箭藿苷 A
|
118525-35-2 | 98% |
|
Sagittatoside A selectively activates estrogen response element (ERE)-luciferase activity via ERα. | ||||
T16351 | NSC16168
化合物 T16351
|
6837-93-0 | 98% |
|
NSC16168 inhibits DNA repair and potentiates CDDP efficacy in cancer. NSC16168 is a specific ERCC1-XPF inhibitor (IC50: 0.42 μM). | ||||
T12329 | Ospemifene D4
化合物 T12329
|
T12329 | 98% |
|
Ospemifene D4 is a deuterium labeled Ospemifene. Ospemifene is a selective and orally active modulator of estrogen receptor. | ||||
T12312 | OP-1074
化合物 T12312
|
1443752-76-8 | 98% |
|
OP-1074 is a pure antiestrogen and a selective degrader of ER, shows specific antiestrogenic activity for ERα and ERβ. | ||||
TN1679 | Genistein 7,4'-di-O-β-D-glucoside
染料木素-7,4'-二-O-Β-D-葡萄糖苷
|
36190-98-4 | 98% |
|
Genistein 7,4'-di-O-beta-D-glucopyranoside shows significant estrogenic proliferative effect in MCF-7 cell in sub-cytotoxic concentration range. | ||||
T11222 | ERB-196
化合物 T11222
|
550997-55-2 | 98% |
|
Erb-196 is an estrogen receptor-receptor agonist with non-steroidal selectivity. | ||||
T11231 | ERRγ Inverse Agonist 1
化合物 T11231
|
2316832-86-5 | 98% |
|
ERRγ Inverse Agonist 1 (Compound 12) 是有效的、选择性的、口服生物可利用的雌激素相关受体 γ (ERRγ)的反向激动剂,IC50值为 40 nM。 |