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Targets Recommended: Others

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Cat. No. Product Name Target Signaling Pathways
T11864 Iptacopan

LNP023

Others Others
Iptacopan (LNP023) 是一种与factor B 亲和力较高的抑制剂。
T9189 Iptacopan hydrochloride

Iptacopan HCl,LNP023 hydrochloride

Complement System Immunology/Inflammation
Iptacopan hydrochloride (LNP023 hydrochloride) 是一种可口服、高效和高选择性的因子 B 抑制剂,IC50 为 10 nM。 LNP023 显示与人因子 B 的直接、可逆和高亲和力结合,KD 为 7.9 nM。
T69628 Iptacopan hydrochloride hydrate

Iptacopan hydrochloride hydrate is a highly potent and highly selective factor B inhibitor.
T69627 Dapivirine HCl

Dapivirine HCl is the salt form of Dapivirine, also known as TMC120, a non-nucleoside inhibitor for HIV reverse transcriptase with IC50 of 24 nM. The HIV-1 replication inhibitor dapivirine (DPV) is one of the most promising drug candidates being used in topical microbicide products for prevention of HIV-1 sexual transmission.

化合物

Iptacopan
Cat.No: T11864
Synonym: LNP023
Target: Others
Iptacopan hydrochloride
Cat.No: T9189
Synonym: Iptacopan HCl,LNP023 hydrochloride
Target: Complement System
Iptacopan hydrochloride hydrate
Cat.No: T69628
Synonym:
Target:
Dapivirine HCl
Cat.No: T69627
Synonym:
Target:
TargetMol Loading
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