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Targets Recommended: cell cycle arrest PARP Arp2/3 Complex PPAR Aromatase Arrestin IFNAR Arginase Aryl Hydrocarbon Receptor Monocarboxylate transporter Carbonic Anhydrase Stearoyl-CoA Desaturase (SCD) Decarboxylase Acetyl-CoA Carboxylase RAR/RXR SARS-CoV Parasite NMDAR Carboxypeptidase Molecular Glues Target Protein Ligand-Linker Conjugate Ligands for Target Protein for PROTAC GSK-3

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Cat. No.	Product Name	Form	Specificity Of Inhibition
CL0124	AMPAR antagonist/activator kit AMPAR antagonist/activator kit
CL0093	PARP inhibitor kit PARP inhibitor kit
CL0050	Antiparasitic compound kit Antiparasitic compound kit
C0113	Magrose Beads Heparin 肝素磁珠
CL0104	NMDAR agonist/antagonist kit NMDAR agonist/antagonist kit
CL0099	RAR/RXR agonist kit RAR/RXR agonist kit
CL0076	PPAR inhibitor/activator kit PPAR inhibitor/activator kit
CL0138	Carbonic Anhydrase inhibitor kit Carbonic Anhydrase inhibitor kit

Cat. No.	Product Name	Target	Signaling Pathways
T1881	AR-A014418 AR 0133418,GSK-3beta Inhibitor VIII,AR 014418,GSK 3β inhibitor VIII	GSK-3	PI3K/Akt/mTOR signaling; Stem Cells
	AR-A014418 (GSK 3β inhibitor VIII) 是选择性的，ATP 竞争性的 GSK3β抑制剂，其 IC50=104 nM，Ki=38 nM。
T14315	AR-9281 APAU	Epoxide Hydrolase	Metabolism
	AR-9281 (APAU) 是选择性的可溶性环氧化物水解酶抑制剂，可用于研究高血压和 2 型糖尿病。
T21646L	AR-M 1896 Acetate AR-M 1896 Acetate (367518-31-8 Free base)	Neuropeptide Y Receptor	GPCR/G Protein; Neuroscience
	AR-M 1896 Acetate 是 GalR2 的选择性激动剂。
T14316	AR-C155858	Monocarboxylate transporter	Membrane transporter/Ion channel
	AR-C155858 是单羧酸转运蛋白 MCT1 和 MCT2 的抑制剂，Ki 分别为2.3和 10 nM。
T8329	AR 231453	GPR	Endocrinology/Hormones; GPCR/G Protein
	AR 231453 是一种口服具有活性的、特异性的 GPR119激动剂。它能够刺激细胞增殖，改善胰岛 β 细胞的功能。
T26647	AR420626 AR 420626,AR-420626	Others	Others
	AR420626 是一种选择性脂肪酸 3 受体 (FA3R) 激动剂，对被选择性 FA3R 拮抗剂 β-羟基丁酸酯 (BHB) 完全阻断的猪甲酚 (SALS) 提供保护作用。
T10359	AR antagonist 1	Androgen Receptor; Ligand for E3 Ligase; Ligands for Target Protein for PROTAC	Endocrinology/Hormones; PROTAC
	AR antagonist 1 是 AR 拮抗剂，能够与 E3 连接酶配体结合，与 VHL 蛋白结合亲和力较弱，用于 PROTACARD-266 合成。
T4236	AR-M 1000390 hydrochloride ARM390 Hydrochloride,ARM-390 HCl	Opioid Receptor	Endocrinology/Hormones; GPCR/G Protein; Neuroscience
	AR-M 1000390 hydrochloride (ARM-390 HCl) 是选择性 δ 阿片受体激动剂，EC50为 7.2±0.9 nM。
T6392	AR42 OSU-HDAC42,AR-42,(S)-(+)-N-羟基-4-(3-甲基-2-苯基丁酰氨基)苯甲酰胺,AR 42,HDAC-42	HDAC	Chromatin/Epigenetic; DNA Damage/DNA Repair
	AR42 (OSU-HDAC42) 是一种 HDAC 抑制剂(IC50: 30 nM)。
T60924	Verosudil AR-12286	ROCK	Cell Cycle/Checkpoint; Cytoskeletal Signaling; Stem Cells
	Verosudil (AR-12286) 是一种高效的 Rho 激酶 (ROCK) 抑制剂，对 ROCK1 和 ROCK2 的 Ki 分别为 2 和 2 nM。AR-12286 可逆转类固醇诱导的小鼠眼内压，可通过增加眼房水通过小梁网流出来减缓眼压。
T10358	Netarsudil Dihydrochloride AR-13324 Dihydrochloride	ROCK	Cell Cycle/Checkpoint; Cytoskeletal Signaling; Stem Cells
	Netarsudil Dihydrochloride (AR-13324 Dihydrochloride) 是 Rho 相关蛋白激酶 (ROCK) 和去甲肾上腺素转运蛋白 (NET) 的抑制剂，可有效降低眼压 (IOP)。
T30110	AR 12456 AR12456,AR-12456
	AR-12456 is a Trapidil derivative that prevents serum hyperlipidemia in guinea pigs.
T39767	AR-C141990 hydrochloride AR-C141990 hydrochloride
	AR-C141990 hydrochloride is a potent inhibitor of lactate transporters known as monocarboxylate transporters (MCTs). It has pK i values of 7.6 and 6.6 for MCT-1 and MCT-2, respectively. Additionally, this compound exhibits immunosuppressive properties and effectively inhibits the graft versus host response.
T28881	Sulmazole Vardax,AR-L 115BS,AR-L 115-BS	PDE; Parasite; Adenosine Receptor	GPCR/G Protein; Metabolism; Microbiology/Virology; Neuroscience
	Sulmazole (AR-L 115-BS) 是一种小分子 cGMP-PDE抑制剂。Sulmazole 对 A1 腺苷受体具有竞争性抑制作用，可改善心脏指数，低肺毛细血管楔压，可用于研究心脏衰竭。
T10360	AR-A 2 AR-A 000002	Others	Others
	AR-A 2 is a selective 5-HT1B receptor antagonist, with a high affinity to guinea pig cortex 5HT1B/1D and recombinant guinea pig 5-HT1B receptors (Ki: 0.24 and 0.47 nM) and with 10-fold lower affinity to guinea pig 5-HT1D receptor (Ki: 5 nM).
TQ0113	Iclaprim 艾拉普林,AR-100	Antibacterial; Antibiotic	Microbiology/Virology
	Iclaprim (AR-100) 是一种细菌二氢叶酸的选择性新型抑制剂, 可抑制金黄色葡萄球菌的生长, 其 MIC90值为 0.06 μg/mL。
T30111	AR 12465 AR-12465
	AR 12465 is a trapidil derivative which may affect LDL receptor mediated uptake and degradation of 125 I-LDL by human skin fibroblasts (HSF) and human hepatic cells (HEP G2).
T23752	AR-C141990 ARC-141990,AR C141990,ARC141990,ARC 141990
	AR-C141990 is a lactate transporters inhibitor.
T30120	AR-C126313 ARC126313,AR C126313
	AR-C126313 is a thiouracil derivative.
T6320	GDC-0879 GDC 0879,AR-00341677,GDC0879	Raf	MAPK
	GDC-0879 (AR-00341677) 是一种选择性B-Raf 抑制剂，IC50为 0.13 nM。
T3955	AR7	Retinoid Receptor	Metabolism
	AR7 是一种非典型的 RARA/RARα(视黄酸受体 α) 拮抗剂，能够特异性激活伴侣介导的自噬活性，对自噬无影响。
T30112	AR 17048 AR17048,AR-17048
	AR-17048 is a potential anti-rheumatic drug.
T0371	Gliquidone AR-DF 26,格列喹酮,Glurenorm	Potassium Channel	Membrane transporter/Ion channel
	Gliquidone (AR-DF 26) 是一种磺酰脲类的抗糖尿病药物，可用于2型糖尿病的研究。
T2466	Osu03012 Osu-03012,Osu 03012,AR-12	PDK	PI3K/Akt/mTOR signaling
	Osu03012 (AR-12) 是一种口服生物可利用的小分子塞来昔布衍生的磷酸肌醇依赖性激酶 1(PDK1) 抑制剂，具有潜在的抗肿瘤活性。
T0080	Trapidil 唑嘧胺,乐可安,Rocornal,Trapymine,Avantrin,Trapymin,AR-12008	PDGFR; PDE	Angiogenesis; Metabolism; Tyrosine Kinase/Adaptors
	Trapidil (Avantrin) 是一种抗血小板药物，是一种血管扩张剂，有特异性血小板衍生生长因子。
T30133	AR-L 100 BS BRN 0842454,AR-L-100BS,AR-L100 BS
	AR-L 100 BS is a bioactive chemical with cardiovascular effects and blood pressure.
T26657	AR-H067637
	AR-H067637 is a rapid-binding, reversible and potent (inhibition constant K(i) = 2-4 nM), competitive inhibitor of thrombin, as well as of thrombin bound to fibrin (clot-bound thrombin) or to thrombomodulin. The total amount of free thrombin generated in
T10052	AR-08	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	AR-08 是一种有效的 α2 肾上腺素能受体 (α2-adrenergic receptor) 激动剂，可用于研究多动症与注意力缺陷。
T30191L	Atecegatran TFA Atecegatran TFA(917904-13-3 Free base）,AR-H067637 TFA	Others	Others
	Atecegatran TFA 常被当作一种抗凝血剂，可用来治疗心血管疾病。
T26652	AR-C67085 PSB0413,PSB 0413,PSB-0413
	AR-C67085 is a ADP receptor antagonist.
T37822	AR-C 141990 hydrochloride
	Monocarboxylate transporter (MCT1) inhibitor (pKi = 7.6. Exhibits approximately 10-fold selectivity for MCT1 over MCT2 and no significant activity against MCT3 or 4. Inhibits graft versus host response and prolongs cardiac graft survival in a rat model. Immunosuppressant. Also inhibits brain penetration of GHB analog HOCPCA.
T69853	AR-C117977
	AR-C117977 is a potent MCT1 inhibitor, which can reduce vimmune responses both in vitro and in vivo, maintains long-term graft survival, and induces operational tolerance.
T30114	AR-12463 AR12463
	AR 12463 是一种曲匹地尔衍生物，可显着减少血清总胆固醇的增加。
T69613	Ar-H047108 free base
	Ar-H047108 free base is an imidazopyridine potassium competitive acid blocker (P-CAB). This drug may be used to treat early stellate cell activation and veno-occlusive-disease (VOD)-like hepatotoxicity.
T21059	Ticagrelor metabolite M5 Ticagrelor metabolite M5,,T437700,替格瑞洛杂质H,AR-C133913XX	P2Y Receptor	GPCR/G Protein; Neuroscience
	Ticagrelor metabolite M5 (T437700) 是 Ticagrelor 的代谢物，是 P2Y12 受体的第一个可逆口服拮抗剂。与氯吡格雷相比，替格瑞洛对 ADP 受体具有更快和更一致的抑制作用。替格瑞洛用于治疗急性冠状动脉综合征(ACS)。
T30113	AR-102 UNII-54923Z352W
	AR-102 is a bio-active chemical.
T0179	Ticagrelor 替格瑞洛,替卡格雷,AR-C 126532XX,AZD6140	P450; P2Y Receptor	GPCR/G Protein; Metabolism; Neuroscience
	Ticagrelor (AR-C 126532XX) (AZD6140) 是可逆的，可口服的 P2Y12受体拮抗剂，可抑制血小板聚集。
T21857	AR-R 17779 hydrochloride
	AR-R17779 hydrochloride 是一种有效和选择性的 nAChR 完全激动剂，对α7和α4β2亚型的Ki 直分别为 92 和 16000 nM。AR-R17779 hydrochloride 可以改善大鼠的学习和记忆能力。AR-R17779 hydrochloride 也具有抗焦虑活性。AR-R17779 hydrochloride 可通过激活抗炎胆碱能（迷走神经）通路减轻炎症。
T22580	AR-C 102222	Others	Others
	AR-C 102222 is an iNOS inhibitor.
T10361	AR-C102222 hydrochloride	Others	Others
	AR-C102222 hydrochloride is a competitive, orally active, and highly selective inducible nitric oxide synthase (iNOS) inhibitor (IC50: 37 nM). It has antinociception and anti-inflammatory activities.
T70956	JNJ-pan-AR
	JNJ-pan-AR, a meylated analogue of JNJ-63576253, is a novel pan-AR antagonist with potent activity against wild-type and clinically relevant AR mutations including F877L. JNJ63576253, also known as TRC253, is a potent and orally active androgen receptor antagonist. TRC253 specifically binds to both wild-type and certain mutant forms of AR, thereby preventing androgen-induced receptor activation and facilitating the formation of inactive complexes that cannot translocate to the nucleus.
T11804	β3-AR agonist 2	Others	Others
	β3-AR agonist 2 is a potent and selective agonist of β3-adrenergic receptor (β3-AR with an EC50 of 8 nM).
T18596	PROTAC AR Degrader-4	Others	Others
	PROTAC AR Degrader-4 comprises a cIAP1 ligand binding group, a linker and an androgen receptor (AR) binding group. PROTAC AR Degrader-4 is an AR degrader. Degradation inducers based on cIAP1 are called specific and non-genetic IAP-dependent protein erasers (SNIPERs)[1].
T10523	β3-AR agonist 1	Others	Others
	β3-AR agonist 1 is a highly selective, and orally available agonist of β3-adrenergic receptor (EC50: 18 nM), being inactive to β1-, β2-, and α1A-AR (β1/β3, β2/β3, and α1A/β3>556-fold).
T10358L	AR-13324 M1 metabolite	Others	Others
	AR-13324 M1 metabolite is a hydrolysis metabolite of AR-13324 mesylate.
T30134	AR-L 57 CL
	AR-L 57 CL is a cardiotonic agent.
T10357	AR-13324 analog mesylate	Others	Others
	AR-13324 analog mesylate is an inhibitor of Rho-kinase and a norepinephrine transporter and reduces intraocular pressure in normotensive monkey eyes.
T30116	AR244555 AR-244555,AR 244555
	AR244555 is a bioactive chemical.
T126273	ar-Turmerol
	ar-Turmerol 是一种有用的有机化合物，可用于生命科学领域的相关研究，其产品编号为 T126273。
T26651	ARC-239 ARC239,AR C 239,AR C239,AR C-239
	ARC-239 is an agonist of α2-adrenergic receptor.

Cat. No.	Product Name	Target	Signaling Pathways
TN1507	Clematichinenoside AR	TNF; Autophagy	Apoptosis; Autophagy
	Clematichinenoside AR 是从中药威灵仙中提取的一种天然产物，具有抗炎和免疫抑制特性，对 PI3K/Akt 信号通路和与胶原诱导的关节炎相关的 TNF-α± 具有抗关节炎作用。
TN7022	Cymen-ar-ol	Antibacterial	Microbiology/Virology
	Cymen-ar-ol 是一种广谱高效的杀菌剂，可接触黏膜。
T14317	ar-Turmerone (+)-ar-Turmerone	Others	Others
	ar-Turmerone ((+)-ar-Turmerone) is a major bioactive compound of the herb Curcuma longa with anti-tumorigenesis and anti-inflammatory activities[1][2][3]. ar-Turmerone ((+)-ar-Turmerone) exerts positive modulation on murine DCs, induces NSC proliferation.
TN3436	ar-Curcumene	Others	Others
	ar-Curcumene has antiinflammatory activity, it could be used as antiinflammatory drugs in respiratory infections. ar-Curcumene is effective as oviposition deterrents against Anopheles stephensi, Aedes aegypti, and Culex quinquefasciatus, it can be conside
TN5371	8-Hydroxy-ar-turmerone
	8-Hydroxy-ar-turmerone may exhibit antitumor activity against breast cancer cells via cell death and cell cycle arrest.
T27282	Erucin AR 1G3839,AR-1G3839,CCRIS-9056,CCRIS9056,AR1G3839,CCRIS 9056
	Erucin is a sulforaphane analog found in cruciferous vegtables. Erucin is a telomerase inhibitor. It induces phase II enzyme activity, suppresses cellular proliferation in hepatocellular carcinoma cells, prevents 6-OHDA-induced neurodegenration, and inhib
T5711	Methylnissolin-3-O-glucoside (6aR, 11 aR)-3-hydroxy-9,l0-diMethoxy pt,美迪紫檀苷,黄芪异黄烷苷,7,2'-二羟基-3',4'-二甲氧基异黄烷	Others	Others
	Methylnissolin-3-O-glucoside ((6aR, 11 aR)-3-hydroxy-9,l0-diMethoxy pt) 是一种类黄酮，从黄芪的根中获得，具有抗炎活性。
TN2037	Paeonilactone C (3S,3AR,6S,7AR)-3-[(苯甲酰基氧基)甲基]四氢-6-羟基-6-甲基-2,5(3H,4H)-苯并呋喃二酮,芍药内苷 C	Others	Others
	Paeonilactone C significantly protects primary cultures of rat cortical cells against H2O2-induced neurotoxicity.
TN2035	Paeonilactone A (3R,3AR,6S,7AR)-四氢-6-羟基-3,6-二甲基-2,5(3H,4H)-苯并呋喃二酮,芍药内苷A	Others	Others
	Paeonilactone A是一种天然产物，属于芍药科芍药属，其产品编号为 TN2035，CAS号为 98751-79-2。Paeonilactone A可用作对照参考。
TN2388	Cleroindicin C	Others	Others
	Cleroindicin C is a natural product from plants
T83554	(4R,4aS,5aS,6aR,6bS,7aR)-4-Hydroxy-3,6b-dimethyl-5-methylene-4,4a,5,5a,6,6a,7,7a-octahydrocyclopropa[2,3]indeno[5,6-b]furan-2(6bH)-one
	'(4R,4aS,5aS,6aR,6bS,7aR)-4-Hydroxy-3,6b-dimethyl-5-methylene-4,4a,5,5a,6,6a,7,7a-octahydrocyclopropa[2,3]indeno[5,6-b]furan-2(6bH)-one' 是倍半萜类内酯化合物。
T67200	(1R,4aS,10aR)-methyl 7-isopropyl-1,4a-dimethyl-1,2,3,4,4a,9,10,10a-octahydrophenanthrene-1-carboxylate
	(1R,4aS,10aR)-methyl 7-isopropyl-1,4a-dimethyl-1,2,3,4,4a,9,10,10a-octahydrophenanthrene-1-carboxylate 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 T67200，CAS号为 1235-74-1。
T83517	(Z)-(1R,3R,4R,4aS,8R,8aR)-3,4,8,8a-Tetramethyl-7-oxo-4-(2-(5-oxo-2,5-dihydrofuran-3-yl)ethyl)decahydronaphthalen-1-yl 2-methylbut-2-enoate
	(Z)-(1R,3R,4R,4aS,8R,8aR)-3,4,8,8a-Tetramethyl-7-oxo-4-(2-(5-oxo-2,5-dihydrofuran-3-yl)ethyl)decahydronaphthalen-1-yl 2-methylbut-2-enoate (compound 7a) 是一种特定立体化学配置的二萜类化合物。
TCS1372	Atraric acid	Phosphatase; Androgen Receptor	Endocrinology/Hormones; Metabolism
	Atraric acid 衍生物作为一种新的化学先导结构，用于作为 AR 拮抗剂的新型治疗化合物，可用于预防或治疗前列腺疾病。它以剂量依赖性方式抑制 PTP1B 活性，IC50 值为 51.5 uM，表明阿特拉酸具有治疗糖尿病的潜力。
T5656	(±)-Norcantharidin Endothall anhydride,去甲斑蝥素,Norcantharidin	EGFR; c-Met/HGFR	Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
	(±)-Norcantharidin (Endothall anhydride) 是一种人类结肠癌中 c-Met 和 EGFR 的双重抑制剂，可研究抗癌，具有抗血管生成活性。
T65128	Tartaric acid disodium dihydrate Disodium L-(＋)-Tartrate Dihydrate	Phosphatase; Endogenous Metabolite	Metabolism
	Tartaric acid disodium dihydrate (Disodium L-(＋)-Tartrate Dihydrate) 常用来制作分子生物学和细胞培养中的缓冲液,。Tartaric acid disodium dihydrate 是酸性磷酸酶抑制剂, 可增加秋水仙碱结合 tubulin1的概率。
T21665	DL-α-Hydroxyglutaric acid disodium salt disodium 2-hydroxypentanedioate,DL-Α-羟基戊二酸二钠	Others	Others
	DL-α-Hydroxyglutaric acid disodium salt (disodium 2-hydroxypentanedioate) 是一种 α-羟基酸，由 (R) -5-oxy-2-tetrahydrofuran 羧酸水解形成，在人类神经代谢疾病 D-α-羟基戊二酸尿症中过量产生。
TN6780	Carvacrol methyl ether Methyl carvacrol,Methyl carvacryl ether	Antibacterial	Microbiology/Virology
	Carvacrol methyl ether 来源于植物挥发油，具有抗菌活性。
T5559	Carboxin Carbathiin,Carboxine,Vitavax,Kisvax,萎锈灵	Others; Antibiotic; Antifungal	Microbiology/Virology; Others
	Carboxin (Kisvax)e 是一种内吸杀菌剂和种子保护剂。
T4814	(R)-5-Oxopyrrolidine-2-carboxylic acid D-Pyroglutamic acid,(R)-(+)-2-Pyrrolidone-5-carboxylic acid,D-焦谷氨酸	Others; Endogenous Metabolite	Metabolism; Others
	(R)-5-Oxopyrrolidine-2-carboxylic acid (D-Pyroglutamic acid) 是内源性代谢产物的一种。
TQ0172	2''-O-Rhamnosylicariside II	Others	Others
	2''-O-Rhamnosylicariside II 是天然来源的黄酮类糖苷化合物，可能对改善绝经后骨质疏松有益处。
TQ0024	3-Hydroxyglutaric acid	Endogenous Metabolite	Metabolism
	3-Hydroxyglutaric acid 是一种戊二酸的衍生物。
T5625	Zearalenone 玉米,Mycotoxin F2,玉米烯酮,RAL,F2 toxin,Toxin F2	Others	Others
	Zearalenone (F2 toxin) 是真菌毒素，主要由食物和饲料中的 Fusarium 产生。它会引起幼龄母猪乳房发育早熟或其它雌激素效应。它在猪、牛、羊体内具有雌激素活性，急性毒性低。
T2826	Asaraldehyde Asarylaldehyde,2,4,5-trimethoxy-Benzaldehyde,Asaronaldehyde,细辛醛	COX	Immunology/Inflammation; Neuroscience
	Asaraldehyde (2,4,5-trimethoxy-Benzaldehyde) 是COX-2抑制剂，能够明显降低环加氧酶 II (COX-2) 的活性(IC50:100 μg/mL)。
TJS1382	Taraxerone 蒲公英赛酮	Dehydrogenase	Metabolism
	Taraxerone 是分离自景天的天然产物。它可以增强乙醇脱氢酶和乙醛脱氢酶活性，EC50分别为 512.42 μM 和 500.16 μM。
T5781	taraxasteryl acetate 蒲公英甾醇醋酸酯,醋酸蒲公英酯	Antibacterial	Microbiology/Virology
	Taraxasteryl acetate 是分离自矢状疟原虫中，具有广谱的抗炎活性。它能够改善右旋糖酐、酵母聚糖及花生四烯酸诱导的大鼠后爪水肿。它可用于研究局部炎症。
T9510	1,2-Distearoyl-sn-glycero-3-phosphorylcholine DSPC,L-ALPHA-PHOSPHATIDYLCHOLINE, DISTEAROYL,1,2-Distearoyl-sn-glycero-3-PC,二硬脂酰磷脂酰胆碱	Others	Others
	1,2-Distearoyl-sn-glycero-3-phosphorylcholine (L-ALPHA-PHOSPHATIDYLCHOLINE, DISTEAROYL) 是一种脂质纳米颗粒(LNP) 系统中的脂质成分，可用于合成脂质体。
TN2279	Totarol (+)-Totarol,桃柁酚	Antibacterial; Antifection	Microbiology/Virology
	Totarol ((+)-Totarol) 对几种致病性革兰氏阳性细菌、结核分枝杆菌具有抗菌作用。
TN1918	Medicarpin 美迪紫檀素	Apoptosis; BCL; ROS; JNK	Apoptosis; Immunology/Inflammation; MAPK
	Medicarpin 是从紫花苜蓿中分离出的一种类黄酮。它通过调节 P-gp 介导的药物外流，诱导白血病 P388 细胞凋亡并克服多药耐药性。
T12581	Puerarin-4'-O-β-D-glucopyranoside Puerarin4'-O-glucoside,葛根素-4'-Β-D-葡萄糖苷	Others	Others
	Puerarin-4'-O-β-D-glucopyranoside (Puerarin4'-O-glucoside) 是一种从葛根 (PLR) 中提取的异黄酮。它具有雌激素活性和抗 MCF-7 人乳腺癌细胞增殖作用。
TQ0183	Narciclasine 水仙环素,Lycoricidinol	ROCK	Cell Cycle/Checkpoint; Cytoskeletal Signaling; Stem Cells
	Narciclasine (Lycoricidinol) 是一种植物生长调节剂。它通过调节Rho/Rho 激酶/LIM 激酶/cofilin 信号传导途径，大大增加GTP 酶RhoA 活性以及以RhoA 依赖性方式诱导肌动蛋白应力纤维形成。
TN1803	Isoscoparin	Antioxidant; TNF; NO Synthase; Fatty Acid Synthase	Apoptosis; Immunology/Inflammation; Metabolism; oxidation-reduction
	Isoscoparin 源自 Gentiana algida Pall，具有抗氧化和抗脂肪生成活性。Isoscoparin 可用于预防和治疗肥胖的研究。
TN1808	Isovitexin 2''-O-arabinoside	Others	Others
	Isovitexin 2''-O-arabinoside 是一种在紫花苜蓿植物中发现黄酮类化合物。
T37067	9-hydroxy Stearic Acid	HDAC	Chromatin/Epigenetic; DNA Damage/DNA Repair
	9-hydroxy Stearic Acid 是一种羟基脂肪酸，是9-PAHSA 的活性代谢物。9-hydroxy Stearic Acid 是由9-PAHSA 通过肝脏和胰腺的羧基酯脂肪酶形成的。9-hydroxy Stearic Acid (5 μM)抑制HT-29结肠癌细胞裂解物中组蛋白去乙酰化酶1 (HDAC1)的表达。3 .当浓度为100 μM.1时，可抑制HT-29细胞的增殖，并诱导细胞周期阻滞于G0/ g1期。
T8247	(+)-Aromadendrene	Anti-infection	Microbiology/Virology
	(+)-Aromadendrene 是一种天然产物，对革兰氏阳性菌和革兰氏阴性菌具有显着的抗菌活性。
TN2286	Tsugaric acid A	NO Synthase	Immunology/Inflammation
	Tsugaric acid A 能够显著抑制超氧阴离子的形成，还可以保护人类角质形成细胞，使其免受紫外线 B 诱导的损害。
T2O2731	L-Aspartic acid L-天冬氨酸,L-天冬氨酸；L-天冬碱;L-酰胺天冬酸；L-天冬酰胺一水物,Aspatofort,Asparagic acid	Others; Endogenous Metabolite	Metabolism; Others
	L-Aspartic acid (Aspatofort) 是一种氨基酸，是结肠特异性药物输送的前体药物。
TN1039	Tamarixetin 柽柳黄素,4'-O-Methyl Quercetin	Endogenous Metabolite; Immunology/Inflammation related	Immunology/Inflammation; Metabolism
	Tamarixetin (4'-O-Methyl Quercetin) 是一种槲皮素的天然类黄酮衍生物，具有抗氧化、抗炎作用，能够防止心肌肥厚。
T3778	3'-Hydroxypuerarin Pueraria glycoside,3'-hydroxy Puerarin,3'-羟基葛根素	Others	Others
	3'-Hydroxypuerarin (Pueraria glycoside) 是一种异黄酮，从 Pueraria lobata(Willd.) Ohwi 根部分离出来得到。它是抗氧化剂，具有显著的 ONOO(-)，NO•，总 ROS 清除活性。
T7030	anemarsaponin B 知母皂苷B,知母皂苷 B	p38 MAPK; NF-κB; MEK; COX; NO Synthase	Immunology/Inflammation; MAPK; Neuroscience; NF-κB
	Anemarsaponin B 是一种甾体皂苷，可降低iNOS 和COX-2的蛋白和 mRNA 水平，减少促炎细胞因子的表达和产生。它通过阻断 IκBα 的磷酸化来抑制NF-κB 的 p65 亚基的核转位，还抑制 MAP 激酶激酶 3/6 (MKK3/6) 和混合谱系激酶 3 的磷酸化。
T6S2023	Harpagoside	Others; COX; NO Synthase	Immunology/Inflammation; Neuroscience; Others
	Harpagoside 是从爪钩草中分离出来的一种天然产物，可抑制COX-1和COX-2活性，并抑制 NO 的产生。
T8249	Hexahydrofarnesyl acetone 植酮,Phytone	Others; Antibacterial	Microbiology/Virology; Others
	Hexahydrofarnesyl acetone (Phytone) 是从Launaea mucronata 中分离得到的倍半萜，具有抗菌和抗炎活性，可研究缓解疼痛。
T2972	Rutaecarpine Rutacarpine,吴茱萸次碱,Rhetine,Rutecarpine	COX	Immunology/Inflammation; Neuroscience
	Rutaecarpine (Rhetine) 是从槐木中提取的一种生物碱，是 COX-2的抑制剂，IC50值为0.28 μM。
T2729	Scoparone 滨蒿内酯,Escoparone,Scoparon,Aesculetin dimethyl ether,6,7-dimethoxycoumarin,6,7-Dimethylesculetin	Others	Others
	Scoparone (Aesculetin dimethyl ether) 是分离自毛蒿中，具有抗凝血，抗血管舒张作用和抗炎活性。
T4911	α-Arbutin 4-hydroxyphenyl-D-lucopyranoside,alpha-Arbutoside,α-熊果苷,alpha-Arbutin	Tyrosinase	Proteases/Proteasome
	α-Arbutin (4-hydroxyphenyl-D-lucopyranoside) 是一种流行的、有效的皮肤增白剂，也是一种酪氨酸酶 (tyrosinase) 抑制剂。
TQ0197	Acenocoumarol 醋硝香豆素,新抗凝
	Acenocoumarol 是一种抗凝血剂，与 Vitamin K 拮抗剂的功能相似。
T5041	Faropenem sodium 法罗培南,法罗培南钠	Antibacterial; Antibiotic	Microbiology/Virology
	Faropenem sodium 是一种口服生物可利用的青霉烯类抗生素，能有效杀灭结核分枝杆菌，治疗结核病和社区获得性肺炎。
T19564	Stearoylcarnitine Stearoyl-L-carnitine	Endogenous Metabolite	Metabolism
	Stearoylcarnitine (Stearoyl-L-carnitine) 是一种脂肪酯脂质分子，是一种人内源代谢产物，可作为早发型子痫前期和晚发性子痫前期的生物标志物。
T3S1944	Darutoside Darutin,豯莶苷	Others	Others
	Darutoside (Darutin) 是一种二萜化合物，提取自Siegesbeckia 中。
T4S1962	beta-Asarone β-细辛脑,(Z)-1,2,4-三甲氧基-5-丙烯基苯;顺式细辛脑,Cis-Isoasarone,Cis-Asarone,Cis-Isoelemicin	NF-κB; JNK	MAPK; NF-κB
	beta-Asarone (Cis-Isoelemicin) 是一种石菖蒲中的主要成分，具有免疫抑制、促进安定、中枢神经系统抑制、降温等功能。它可透过血脑屏障，能够预防帕金森病。
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Cat. No.	Product Name
L7000	活性脂质化合物库	385 compounds
	385 种生物活性小分子化合物，用于高通量、高内涵筛选；
L2620	神经退行性疾病化合物库	2154 compounds
	2154 种与神经退行性疾病相关的化合物，可用于高通量和高内涵筛选；
L5700	精选片段库	246 compounds
	246 个片段小分子的独特集合，可用于基于片段的筛选和药物发现（FBDD）；
L3980	DNA损伤/修复库Plus	667 compounds
	667 种 DNA 损伤/修复靶向、结构新颖的化合物；
L1020	EMA 上市药物库	657 compounds
	657个EMA批准药物的独特集合，可用于高通量筛选和高内涵筛选
L1510	核受体化合物库	531 compounds
	531 个核受体作用化合物的独特集合，可用于高通量筛选和高内涵筛选；
L1400	MAPK 抑制剂库	365 compounds
	365 种与MAPK 信号通路相关的生物活性小分子化合物的特有集合，可用于高通量筛选和高内涵筛选；
L2110	抗癌上市药物库	1779 compounds
	1779 个具有抗癌活性小分子的独特集合，所有化合物都经过了严格的临床前研究和临床试验，由FDA、EMA 或NMPA 批准上市，可用于高通量、高内涵筛选。
L2191	抗乳腺癌化合物库	1939 compounds
	1939 种与乳腺癌相关的化合物，可以用于抗乳腺癌药物研发和药理研究；
L2550	谷氨酰胺代谢化合物库	565 compounds
	565 种谷氨酰胺代谢相关的分子，可以用于高通量和高内涵筛选；
L2200	酪氨酸激酶分子库	1016 compounds
	1016 种酪氨酸激酶抑制剂的独特集合，可用于高通量筛选和高内涵筛选；
L3100	造血毒性小分子库	101 compounds
	101 种生物活性小分子化合物的特有集合，用于高通量、高内涵筛选；
L3800	NF-κB 通路分子库	729 compounds
	729 个 NF-κB 信号通路相关的小分子化合物的特有集合，用于高通量、高内涵筛选；
L4300	Wnt/Hedgehog/Notch 通路化合物库	237 compounds
	237 个Wnt & Hedgehog & Notch 靶点相关的生物活性小分子化合物的特有集合，用于相关通路的研究及药物的筛选，可用于高通量、高内涵筛选。
L4100	TGF-β/Smad靶点化合物库	184 compounds
	184 个 TGF-β/Smad 靶点相关的小分子化合物的特有集合，用于高通量、高内涵筛选；
L5900	血脑屏障通透化合物库	509 compounds
	509 个 CNS-Penetrant 生物活性小分子化合物的特有集合，用于高通量、高内涵筛选；
L3500	组蛋白修饰化合物库	469 compounds
	469 个组蛋白修饰相关的小分子化合物的特有集合，用于高通量、高内涵筛选；
L4510	抗寄生虫库	419 compounds
	419 种具有抗寄生虫活性的小分子化合物；
L6750	活血化瘀中药单体库	580 compounds
	580种来源于常见活血化瘀中药的单体化合物，是药物开发、药理研究等领域的有效工具。
L7500	凝血与抗凝化合物库	144 compounds
	144 个化合物的独特集合，可用于高通量筛选和高内涵筛选；

Cat. No.	Product Name	Species	Expression System
TMPK-00870	AREG Protein, Mouse, Recombinant (hFc) AR,MGC13647,CRDGF,AREG,Amphiregulin,SDGF,<...	Mouse	HEK293 Cells
	Amphiregulin (AREG) is a ligand of the epidermal growth factor receptor (EGFR), a widely expressed transmembrane tyrosine kinase. AREG is synthesized as a membrane-anchored precursor protein that can engage in juxtacrine signaling on adjacent cells. Alternatively, after proteolytic processing by cell membrane proteases, mainly TACE/ADAM17, AREG is secreted and behaves as an autocrine or paracrine factor.
TMPK-00820	AREG Protein, Human, Recombinant (hFc) SDGF,AR,MGC13647,AREGB,CRDGF,Amphiregulin,...	Human	HEK293 Cells
	Amphiregulin (AREG) is a member of the epidermal growth factor (EGF) family and is expressed in a plethora of cancers. Tumour growth and metastasis were decreased by AREG silencing in an orthotopic model of pancreatic cancer. AREG may play a critical role in cell migration, invasion, and EMT by activating the EGFR/ERK/NF‑κB signalling pathway in pancreatic cancer cells.
TMPJ-00859	AREG Protein, Human, Recombinant AR,CRDGF,Amphiregulin,Colorectum Cell-Derived Growt...	Human	E. coli
	Amphiregulin (AREG) is a single-pass membrane protein with 252 amino acids. AREG belongs to the amphiregulin family, which contains 1 EGF-like domain. AREG is expressed in a variety of tissues including ovary, placenta, lung, kidney, stomach, colon, and breast. It is related to Epidermal Growth Factor (EGF) and Transforming Growth Factor Alpha (TGF-alpha). As an EGF-related growth factor, AREG interacts with the EGF/TGF-alpha receptor to promote the growth of normal epithelial cells and inhibits...
TMPH-01294	EDNRA Protein, Human, Recombinant (His) ET-A,Endothelin-1 receptor,hET-AR,ETA-R,ETRA,EDNRA,...	Human	P. pastoris (Yeast)
	Receptor for endothelin-1. Mediates its action by association with G proteins that activate a phosphatidylinositol-calcium second messenger system. The rank order of binding affinities for ET-A is: ET1 > ET2 >> ET3.
TMPH-00287	Adrenodoxin reductase Protein, Bovine, Recombinant (E. coli, His) Ferredoxin--NADP(+) reductase,ADXR,NADPH:adrenodoxin oxidore...	Bovine	E. coli
	Serves as the first electron transfer protein in all the mitochondrial P450 systems including cholesterol side chain cleavage in all steroidogenic tissues, steroid 11-beta hydroxylation in the adrenal cortex, 25-OH-vitamin D3-24 hydroxylation in the kidney, and sterol C-27 hydroxylation in the liver. Adrenodoxin reductase Protein, Bovine, Recombinant (E. coli, His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 55.8 kDa and the accession number is ...
TMPH-00932	Androgen receptor Protein, Human, Recombinant (His & Myc & SUMO) Nuclear receptor subfamily 3 group C member 4,A...	Human	E. coli
	Androgen receptor Protein, Human, Recombinant (His & Myc & SUMO) is expressed in E. coli.
TMPH-00288	Adrenodoxin reductase Protein, Bovine, Recombinant (His) Ferredoxin reductase,Adrenodoxin reductase,Ferredoxin--NADP(...	Bovine	P. pastoris (Yeast)
	Serves as the first electron transfer protein in all the mitochondrial P450 systems including cholesterol side chain cleavage in all steroidogenic tissues, steroid 11-beta hydroxylation in the adrenal cortex, 25-OH-vitamin D3-24 hydroxylation in the kidney, and sterol C-27 hydroxylation in the liver. Adrenodoxin reductase Protein, Bovine, Recombinant (His) is expressed in yeast with N-10xHis tag. The predicted molecular weight is 52.8 kDa and the accession number is P08165.
TMPY-02438	AKR1B1 Protein, Human, Recombinant (His) ALDR1,AR,ADR,aldo-keto reductase family 1, member B...	Human	E. coli
	Aldose reductase (AKR1B1) belongs to the aldo/keto reductase superfamily. AKR1B1 is a NADPH-dependent aldo-keto reductase best known as the rate-limiting enzyme of the polyol pathway. Expression of AKR1B1 was the highest in lens and retina. It is the first enzyme in the polyol pathway through which glucose is converted to sorbitol which is important for the function of various organs in the body, and has been implicated in the etiology of diabetic complications. AKR1B1 is quite abundant in the c...
TMPK-00861	A2AR Protein-VLP, Human, Recombinant RDC8,Adenosine A2a R,ADORA2,ADORA 2,ADORA2A,A2aR	Human	HEK293 Cells
	Adenosine is a neuromodulator in the adult central nervous system. Membrane-bound receptors for adenosine have been identified and cDNAs for A1, A2a, A2b, and A3 adenosine receptor subtypes have been cloned recently.Expression of A2a adenosine receptor mRNA in cranial ganglia, carotid body, and intermediate lobe of the pituitary gland similarly suggests novel sites of adenosine action during development and in the adult.
TMPH-00892	A1AR Protein, Human, Recombinant (His) Adenosine receptor A1,ADORA1	Human	E. coli
	Receptor for adenosine. The activity of this receptor is mediated by G proteins which inhibit adenylyl cyclase. A1AR Protein, Human, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 39.3 kDa and the accession number is P30542.
TMPH-01022	C5AR1 Protein-VLP, Human, Recombinant (His) C5a anaphylatoxin chemotactic receptor 1,CD88,C5a anaphylato...	Human	HEK293 Cells
	Receptor for the chemotactic and inflammatory peptide anaphylatoxin C5a. The ligand interacts with at least two sites on the receptor: a high-affinity site on the extracellular N-terminus, and a second site in the transmembrane region which activates downstream signaling events. Receptor activation stimulates chemotaxis, granule enzyme release, intracellular calcium release and superoxide anion production. C5AR1 Protein-VLP, Human, Recombinant (His) is expressed in HEK293 mammalian cells with C-...
TMPH-01023	C5AR1 Protein, Human, Recombinant (Cell-Free, His) C5a anaphylatoxin chemotactic receptor 1,C5R1,C5a-R,C5a anap...	Human	E. coli
	Receptor for the chemotactic and inflammatory peptide anaphylatoxin C5a. The ligand interacts with at least two sites on the receptor: a high-affinity site on the extracellular N-terminus, and a second site in the transmembrane region which activates downstream signaling events. Receptor activation stimulates chemotaxis, granule enzyme release, intracellular calcium release and superoxide anion production. C5AR1 Protein, Human, Recombinant (Cell-Free, His) is expressed in E. coli expression syst...
TMPH-03765	Virus-Like Particles (VLPs) isotype control		HEK293
	Virus-Like Particles (VLPs) isotype control can be used as the control of VLP expressed proteins.
TMPY-01776	Carboxylesterase 2/CES2 Protein, Human, Recombinant (His) carboxylesterase 2,CES2A1,CE-2,PCE-2,iCE	Human	HEK293 Cells
	Carboxylesterase 2/CES2 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 60.4 kDa and the accession number is O00748-1.
TMPY-02130	Argonaute-2 Protein, Mouse, Recombinant (His) mKIAA4215,1110029L17Rik,2310051F07Rik,Ago2,argonaut...	Mouse	Baculovirus Insect Cells
	Argonaute-2 Protein, Mouse, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 99 kDa and the accession number is Q8CJG0.
TMPY-00144	Epstein-Barr virus (Herpesvirus 4) EBV Glycoprotein gp350/EBV GP350 Protein (His) BLLF1,gp22	EBV	Baculovirus Insect Cells
	Epstein-Barr virus (Herpesvirus 4) EBV Glycoprotein gp350/EBV GP350 Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 53.7 kDa and the accession number is A0A0B6VN60.
TMPY-00411	Influenza A H5N1 (A/bar-headed goose/Qinghai/1A/2005) Hemagglutinin/HA Protein (His) Harvey rat sarcoma viral oncogene homolog	H5N1	Baculovirus Insect Cells
	Influenza A H5N1 (A/bar-headed goose/Qinghai/1A/2005) Hemagglutinin/HA Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 59.6 kDa and the accession number is Q195D4.
TMPY-01188	PARP Protein, Human, Recombinant (His) ADPRT1,ADPRT,pADPRT-1,PPOL,ARTD1,PARP-1,po...	Human	Baculovirus Insect Cells
	PARP Protein, Human, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 114.5 kDa and the accession number is A0A024R3T8.
TMPY-02575	PPAR gamma/PPARG Protein, Human, Recombinant (His & GST) CIMT1,PPARγ,GLM1,PPARgamma,PPARG1...	Human	Baculovirus Insect Cells
	Peroxisome proliferator-activated receptor gamma (PPARG), a nuclear hormone receptor, plays a critical role in the lipid and glucose homeostasis, adipocyte differentiation, as well as intracellular insulin-signaling events. The peroxisome proliferator-activated receptor gamma (PPARgamma) regulates osteoblast and osteoclast differentiation, and is the molecular target of thiazolidinediones (TZDs), insulin sensitizers that enhance glucose utilization and adipocyte differentiation. Peroxisome proli...
TMPY-00694	Carbonic Anhydrase 12 Protein, Human, Recombinant (His) HsT18816,FLJ20151,carbonic anhydrase XII,CA12,CAXII	Human	HEK293 Cells
	Carbonic Anhydrase 12 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 31.6 kDa and the accession number is O43570-1.

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