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内质网应激化合物库

内质网应激化合物库

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产品编号 L9700 Endoplasmic Reticulum Stress Compound Library
  库化合物信息   Excel SDF

内质网应激(Endoplasmic Reticulum stress)是细胞为应对内质网腔内错误折叠与未折叠蛋白聚集以及钙离子平衡紊乱等状况,而激活未折叠蛋白反应、内质网超负荷反应和 caspase-12 介导的凋亡通路等信号途径的反应过程。内质网应激既能诱导葡糖调节蛋白(glucose-regulated protein)GRP78、GRP94 等内质网分子伴侣表达而产生保护效应,亦能独立地诱导内源性细胞凋亡,并影响应激细胞的转归,如适应、损伤或凋亡。 内质网应激是一种重要的防御机制,参与多种疾病进程,是一种泛在的病因机制。近年来的研究表明,癌症、炎症性疾病、代谢性疾病、骨质疏松症及神经退行性疾病等有内质网应激信号传递参与。 TargetMol 内质网应激化合物库收录了 193 个内质网应激相关的化合物,靶向 PERKIRE1、ATF6、GRP78等内质网应激信号通路相关靶点,是研究内质网应激及相关疾病的良好工具。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
咨询化合物库
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产品描述

  • 193 个内质网应激相关的化合物集合,可用于高通量和高内涵筛选;
  • 研究内质网应激及相关疾病的良好工具;
  • 靶点包含PERK、IRE1、ATF6、GRP78等内质网应激信号通路相关靶点;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;
  • 严格质检,保证产品结构准确,纯度高,保障实验顺利进行。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L9700)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

Apoptosis (63)
Autophagy (51)
HSP (34)
PERK (18)
JNK (15)
IRE1 (15)
Endogenous Metabolite (13)
Mitophagy (9)
AMPK (8)
NF-κB (7)
Antibiotic (7)
COX (7)
Antibacterial (7)
GPR (6)
Reactive Oxygen Species (6)
P450 (6)
p97 (5)
ERK (5)
HIV Protease (5)
Akt (4)
Phosphatase (4)
PPAR (4)
MEK (4)
DNA/RNA Synthesis (3)
Caspase (3)
Calcium Channel (3)
Prostaglandin Receptor (3)
MMP (3)
GABA Receptor (3)
HDAC (3)
Ferroptosis (3)
c-Kit (3)
5-HT Receptor (3)
Mitochondrial Metabolism (3)
FLT (2)
PDGFR (2)
Mdm2 (2)
Aurora Kinase (2)
Lipoxygenase (2)
Sodium Channel (2)
DUB (2)
SARS-CoV (2)
mTOR (2)
HIF (2)
TGF-beta/Smad (2)
Phospholipase (2)
MAPK (2)
AChE (2)
Casein Kinase (2)
ASK (2)
Sirtuin (2)
Proteasome (2)
CDK (2)
Chloride channel (2)
Estrogen/progestogen Receptor (2)
Antifungal (2)
VEGFR (2)
Antioxidant (2)
PI3K (2)
Glutathione Peroxidase (2)
Gamma-secretase (2)
Histamine Receptor (2)
Src (2)
NADPH (1)
PDK (1)
Histone Demethylase (1)
Dehydrogenase (1)
p38 MAPK (1)
Integrin (1)
HCV Protease (1)
Adenosine deaminase (1)
TNF (1)
Dopamine Receptor (1)
Microtubule Associated (1)
Kinesin (1)
p53 (1)
NOD-like Receptor (NLR) (1)
HIF/HIF Prolyl-Hydroxylase (1)
ATPase (1)
Tyrosinase (1)
HMG-CoA Reductase (1)
Beta Amyloid (1)
Transferase (1)
Monocarboxylate transporter (1)
ROR (1)
AChR (1)
Cannabinoid Receptor (1)
Potassium Channel (1)
GPX (1)
CETP (1)
IκB/IKK (1)
Androgen Receptor (1)
Hexokinase (1)
PROTAC Linker (1)
MTH1 (1)
Stearoyl-CoA Desaturase (SCD) (1)
HSV (1)
PTEN (1)
PDE (1)
UGT (1)
E1/E2/E3 Enzyme (1)
Epigenetic Reader Domain (1)
CaMK (1)
Topoisomerase (1)
Glucocorticoid Receptor (1)
RANKL/RANK (1)
TRP/TRPV Channel (1)
Influenza Virus (1)
Tyrosine Kinases (1)
Raf (1)
Nrf2 (1)
Trk receptor (1)
Melatonin Receptor (1)
MRP (1)
HBV (1)
P-gp (1)
Interleukin (1)
Parasite (1)
Cysteine Protease (1)
PGE Synthase (1)
Nucleoside Antimetabolite/Analog (1)
FXR (1)
ATP Citrate Lyase (1)
HER (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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